Nettekoven M - Search Results

1

Rational design of novel pyrrolidine derivatives as orally active neurokinin-3 receptor antagonists.

Ratni H, Ballard TM, Bissantz C, Hoffmann T, Jablonski P, Knoflach F, Knust H, Malherbe P, Nettekoven M, Patiny-Adam A, Riemer C, Schmitt M, Spooren W. Ratni H, et al. Among authors: nettekoven m. Bioorg Med Chem Lett. 2010 Nov 15;20(22):6735-8. doi: 10.1016/j.bmcl.2010.08.138. Epub 2010 Sep 17. Bioorg Med Chem Lett. 2010. PMID: 20850972

2

Combinatorial synthesis of libraries of indole derivatives.

Nettekoven M. Nettekoven M. Bioorg Med Chem Lett. 2001 Aug 20;11(16):2169-71. doi: 10.1016/s0960-894x(01)00393-6. Bioorg Med Chem Lett. 2001. PMID: 11514162

3

Comparison of inhibitory activity of isomeric triazolopyridine derivatives towards adenosine receptor subtypes or do similar structures reveal similar bioactivities?

Guba W, Nettekoven M, Püllmann B, Riemer C, Schmitt S. Guba W, et al. Among authors: nettekoven m. Bioorg Med Chem Lett. 2004 Jun 21;14(12):3307-12. doi: 10.1016/j.bmcl.2004.03.104. Bioorg Med Chem Lett. 2004. PMID: 15149696

4

Novel and potent NPY5 receptor antagonists derived from virtual screening and iterative parallel chemistry design.

Guba W, Neidhart W, Nettekoven M. Guba W, et al. Among authors: nettekoven m. Bioorg Med Chem Lett. 2005 Mar 15;15(6):1599-603. doi: 10.1016/j.bmcl.2005.01.063. Bioorg Med Chem Lett. 2005. PMID: 15745805

5

Isomeric thiazole derivatives as ligands for the neuropeptide Y5 receptor.

Nettekoven M, Guba W, Neidhart W, Mattei P, Pflieger P, Roche O, Taylor S. Nettekoven M, et al. Bioorg Med Chem Lett. 2005 Jul 15;15(14):3446-9. doi: 10.1016/j.bmcl.2005.05.009. Bioorg Med Chem Lett. 2005. PMID: 15951170

6

Benzodioxoles: novel cannabinoid-1 receptor inverse agonists for the treatment of obesity.

Alig L, Alsenz J, Andjelkovic M, Bendels S, Bénardeau A, Bleicher K, Bourson A, David-Pierson P, Guba W, Hildbrand S, Kube D, Lübbers T, Mayweg AV, Narquizian R, Neidhart W, Nettekoven M, Plancher JM, Rocha C, Rogers-Evans M, Röver S, Schneider G, Taylor S, Waldmeier P. Alig L, et al. Among authors: nettekoven m. J Med Chem. 2008 Apr 10;51(7):2115-27. doi: 10.1021/jm701487t. Epub 2008 Mar 13. J Med Chem. 2008. PMID: 18335976

7

Refinement of histamine H3 ligands pharmacophore model leads to a new class of potent and selective naphthalene inverse agonists.

Roche O, Nettekoven M, Vifian W, Sarmiento RM. Roche O, et al. Among authors: nettekoven m. Bioorg Med Chem Lett. 2008 Aug 1;18(15):4377-9. doi: 10.1016/j.bmcl.2008.06.062. Epub 2008 Jun 21. Bioorg Med Chem Lett. 2008. PMID: 18606542

8

Discovery of benzoylpiperazines as a novel class of potent and selective GlyT1 inhibitors.

Pinard E, Alberati D, Borroni E, Fischer H, Hainzl D, Jolidon S, Moreau JL, Narquizian R, Nettekoven M, Norcross RD, Stalder H, Thomas AW. Pinard E, et al. Among authors: nettekoven m. Bioorg Med Chem Lett. 2008 Sep 15;18(18):5134-9. doi: 10.1016/j.bmcl.2008.07.086. Epub 2008 Jul 24. Bioorg Med Chem Lett. 2008. PMID: 18752953

9

5-hydroxyindole-2-carboxylic acid amides: novel histamine-3 receptor inverse agonists for the treatment of obesity.

Pierson PD, Fettes A, Freichel C, Gatti-McArthur S, Hertel C, Huwyler J, Mohr P, Nakagawa T, Nettekoven M, Plancher JM, Raab S, Richter H, Roche O, Rodríguez Sarmiento RM, Schmitt M, Schuler F, Takahashi T, Taylor S, Ullmer C, Wiegand R. Pierson PD, et al. Among authors: nettekoven m. J Med Chem. 2009 Jul 9;52(13):3855-68. doi: 10.1021/jm900409x. J Med Chem. 2009. PMID: 19456097

10

Selective naphthalene H(3) receptor inverse agonists with reduced potential to induce phospholipidosis and their quinoline analogs.

Rodríguez Sarmiento RM, Nettekoven MH, Taylor S, Plancher JM, Richter H, Roche O. Rodríguez Sarmiento RM, et al. Bioorg Med Chem Lett. 2009 Aug 1;19(15):4495-500. doi: 10.1016/j.bmcl.2009.03.100. Epub 2009 Mar 26. Bioorg Med Chem Lett. 2009. PMID: 19524437

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