Roush WR - Search Results

1

Identification of SR3335 (ML-176): a synthetic RORα selective inverse agonist.

Kumar N, Kojetin DJ, Solt LA, Kumar KG, Nuhant P, Duckett DR, Cameron MD, Butler AA, Roush WR, Griffin PR, Burris TP. Kumar N, et al. Among authors: roush wr. ACS Chem Biol. 2011 Mar 18;6(3):218-22. doi: 10.1021/cb1002762. Epub 2010 Dec 6. ACS Chem Biol. 2011. PMID: 21090593 Free PMC article.

2

Synthesis of small molecule inhibitors of the orphan nuclear receptor steroidogenic factor-1 (NR5A1) based on isoquinolinone scaffolds.

Roth J, Madoux F, Hodder P, Roush WR. Roth J, et al. Among authors: roush wr. Bioorg Med Chem Lett. 2008 Apr 15;18(8):2628-32. doi: 10.1016/j.bmcl.2008.03.027. Epub 2008 Mar 14. Bioorg Med Chem Lett. 2008. PMID: 18374567 Free PMC article.

3

A novel and specific NADPH oxidase-1 (Nox1) small-molecule inhibitor blocks the formation of functional invadopodia in human colon cancer cells.

Gianni D, Taulet N, Zhang H, DerMardirossian C, Kister J, Martinez L, Roush WR, Brown SJ, Bokoch GM, Rosen H. Gianni D, et al. Among authors: roush wr. ACS Chem Biol. 2010 Oct 15;5(10):981-93. doi: 10.1021/cb100219n. ACS Chem Biol. 2010. PMID: 20715845 Free PMC article.

4

Identification of SR1078, a synthetic agonist for the orphan nuclear receptors RORα and RORγ.

Wang Y, Kumar N, Nuhant P, Cameron MD, Istrate MA, Roush WR, Griffin PR, Burris TP. Wang Y, et al. Among authors: roush wr. ACS Chem Biol. 2010 Nov 19;5(11):1029-34. doi: 10.1021/cb100223d. ACS Chem Biol. 2010. PMID: 20735016 Free PMC article.

5

Enantio- and diastereoselective synthesis of (E)-1,5-syn-diols: application to the synthesis of the C(23)-C(40) fragment of tetrafibricin.

Kister J, Nuhant P, Lira R, Sorg A, Roush WR. Kister J, et al. Among authors: roush wr. Org Lett. 2011 Apr 1;13(7):1868-71. doi: 10.1021/ol2003836. Epub 2011 Mar 4. Org Lett. 2011. PMID: 21375316 Free PMC article.

6

Identification of a novel non-retinoid pan inverse agonist of the retinoic acid receptors.

Busby SA, Kumar N, Kuruvilla DS, Istrate MA, Conkright JJ, Wang Y, Kamenecka TM, Cameron MD, Roush WR, Burris TP, Griffin PR. Busby SA, et al. Among authors: roush wr. ACS Chem Biol. 2011 Jun 17;6(6):618-27. doi: 10.1021/cb100396s. Epub 2011 Mar 17. ACS Chem Biol. 2011. PMID: 21381756 Free PMC article.

7

Suppression of TH17 differentiation and autoimmunity by a synthetic ROR ligand.

Solt LA, Kumar N, Nuhant P, Wang Y, Lauer JL, Liu J, Istrate MA, Kamenecka TM, Roush WR, Vidović D, Schürer SC, Xu J, Wagoner G, Drew PD, Griffin PR, Burris TP. Solt LA, et al. Among authors: roush wr. Nature. 2011 Apr 28;472(7344):491-4. doi: 10.1038/nature10075. Epub 2011 Apr 17. Nature. 2011. PMID: 21499262 Free PMC article.

8

Development of a Double Allylboration Reagent Targeting 1,5-syn-(E)-Diols: Application to the Synthesis of the C(23)-C(40) Fragment of Tetrafibricin.

Nuhant P, Kister J, Lira R, Sorg A, Roush WR. Nuhant P, et al. Among authors: roush wr. Tetrahedron. 2011 Sep 2;67(35):6497-6512. doi: 10.1016/j.tet.2011.06.008. Tetrahedron. 2011. PMID: 21857752 Free PMC article.

9

Enantio- and diastereoselective synthesis of N-acetyl dihydrotetrafibricin methyl ester.

Nuhant P, Roush WR. Nuhant P, et al. Among authors: roush wr. J Am Chem Soc. 2013 Apr 10;135(14):5340-3. doi: 10.1021/ja401918r. Epub 2013 Mar 26. J Am Chem Soc. 2013. PMID: 23530855 Free PMC article.

10

Development of highly selective casein kinase 1δ/1ε (CK1δ/ε) inhibitors with potent antiproliferative properties.

Bibian M, Rahaim RJ, Choi JY, Noguchi Y, Schürer S, Chen W, Nakanishi S, Licht K, Rosenberg LH, Li L, Feng Y, Cameron MD, Duckett DR, Cleveland JL, Roush WR. Bibian M, et al. Among authors: roush wr. Bioorg Med Chem Lett. 2013 Aug 1;23(15):4374-80. doi: 10.1016/j.bmcl.2013.05.075. Epub 2013 May 31. Bioorg Med Chem Lett. 2013. PMID: 23787102 Free PMC article.

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