Conte Camerino D - Search Results

1

Synthesis and toxicopharmacological evaluation of m-hydroxymexiletine, the first metabolite of mexiletine more potent than the parent compound on voltage-gated sodium channels.

Catalano A, Desaphy JF, Lentini G, Carocci A, Di Mola A, Bruno C, Carbonara R, De Palma A, Budriesi R, Ghelardini C, Perrone MG, Colabufo NA, Conte Camerino D, Franchini C. Catalano A, et al. Among authors: conte camerino d. J Med Chem. 2012 Feb 9;55(3):1418-22. doi: 10.1021/jm201197z. Epub 2012 Jan 31. J Med Chem. 2012. PMID: 22191686

2

Stereospecific synthesis of "para-hydroxymexiletine" and sodium channel blocking activity evaluation.

Catalano A, Carocci A, Fracchiolla G, Franchini C, Lentini G, Tortorella V, De Luca A, De Bellis M, Desaphy JF, Conte Camerino D. Catalano A, et al. Among authors: conte camerino d. Chirality. 2004 Feb;16(2):72-8. doi: 10.1002/chir.10307. Chirality. 2004. PMID: 14712469

3

Synthesis and in vitro sodium channel blocking activity evaluation of novel homochiral mexiletine analogs.

Carocci A, Catalano A, Bruno C, Lentini G, Franchini C, De Bellis M, De Luca A, Conte Camerino D. Carocci A, et al. Among authors: conte camerino d. Chirality. 2010 Mar;22(3):299-307. doi: 10.1002/chir.20741. Chirality. 2010. PMID: 19544349

4

N-aryl-2,6-dimethylbenzamides, a new generation of tocainide analogues as blockers of skeletal muscle voltage-gated sodium channels.

Muraglia M, De Bellis M, Catalano A, Carocci A, Franchini C, Carrieri A, Fortugno C, Bertucci C, Desaphy JF, De Luca A, Conte Camerino D, Corbo F. Muraglia M, et al. Among authors: conte camerino d. J Med Chem. 2014 Mar 27;57(6):2589-600. doi: 10.1021/jm401864b. Epub 2014 Mar 7. J Med Chem. 2014. PMID: 24568674

5

Homologation of mexiletine alkyl chain and stereoselective blockade of skeletal muscle sodium channels.

Duranti A, Franchini C, Lentini G, Loiodice F, Tortorella V, De Luca A, Pierno S, Conte Camerino D. Duranti A, et al. Among authors: conte camerino d. Eur J Med Chem. 2000 Jan;35(1):147-56. doi: 10.1016/s0223-5234(00)00115-x. Eur J Med Chem. 2000. PMID: 10733611

6

Synthesis of new 2,6-prolylxylidide analogues of tocainide as stereoselective blockers of voltage-gated Na(+) channels with increased potency and improved use-dependent activity.

Franchini C, Corbo F, Lentini G, Bruno G, Scilimati A, Tortorella V, Conte Camerino D, De Luca A. Franchini C, et al. Among authors: conte camerino d. J Med Chem. 2000 Oct 5;43(20):3792-8. doi: 10.1021/jm000931l. J Med Chem. 2000. PMID: 11020295

7

Inhibition of skeletal muscle sodium currents by mexiletine analogues: specific hydrophobic interactions rather than lipophilia per se account for drug therapeutic profile.

De Luca A, Talon S, De Bellis M, Desaphy JF, Franchini C, Lentini G, Catalano A, Corbo F, Tortorella V, Conte-Camerino D. De Luca A, et al. Among authors: conte camerino d. Naunyn Schmiedebergs Arch Pharmacol. 2003 Mar;367(3):318-27. doi: 10.1007/s00210-002-0669-0. Epub 2003 Jan 25. Naunyn Schmiedebergs Arch Pharmacol. 2003. PMID: 12644906

8

Hydroxylated analogs of mexiletine as tools for structural-requirements investigation of the sodium channel blocking activity.

Catalano A, Carocci A, Cavalluzzi MM, Di Mola A, Lentini G, Lovece A, Dipalma A, Costanza T, Desaphy JF, Conte Camerino D, Franchini C. Catalano A, et al. Among authors: conte camerino d. Arch Pharm (Weinheim). 2010 Jun;343(6):325-32. doi: 10.1002/ardp.200900218. Arch Pharm (Weinheim). 2010. PMID: 20509146

9

In vivo evaluation of antimyotonic efficacy of β-adrenergic drugs in a rat model of myotonia.

Desaphy JF, Costanza T, Carbonara R, Conte Camerino D. Desaphy JF, et al. Among authors: conte camerino d. Neuropharmacology. 2013 Feb;65:21-7. doi: 10.1016/j.neuropharm.2012.09.006. Epub 2012 Sep 18. Neuropharmacology. 2013. PMID: 23000075 Free PMC article.

10

Preclinical evaluation of marketed sodium channel blockers in a rat model of myotonia discloses promising antimyotonic drugs.

Desaphy JF, Carbonara R, Costanza T, Conte Camerino D. Desaphy JF, et al. Among authors: conte camerino d. Exp Neurol. 2014 May;255(100):96-102. doi: 10.1016/j.expneurol.2014.02.023. Epub 2014 Mar 5. Exp Neurol. 2014. PMID: 24613829 Free PMC article.

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