Pocalyko DJ - Search Results

1

Discovery of a series of 2-(1H-pyrazol-1-yl)pyridines as ALK5 inhibitors with potential utility in the prevention of dermal scarring.

Boys ML, Bian F, Kramer JB, Chio CL, Ren XD, Chen H, Barrett SD, Sexton KE, Iula DM, Filzen GF, Nguyen MN, Angell P, Downs VL, Wang Z, Raheja N, Ellsworth EL, Fakhoury S, Bratton LD, Keller PR, Gowan R, Drummond EM, Maiti SN, Hena MA, Lu L, McConnell P, Knafels JD, Thanabal V, Sun F, Alessi D, McCarthy A, Zhang E, Finzel BC, Patel S, Ciotti SM, Eisma R, Payne NA, Gilbertsen RB, Kostlan CR, Pocalyko DJ, Lala DS. Boys ML, et al. Among authors: pocalyko dj. Bioorg Med Chem Lett. 2012 May 15;22(10):3392-7. doi: 10.1016/j.bmcl.2012.04.013. Epub 2012 Apr 10. Bioorg Med Chem Lett. 2012. PMID: 22542194

2

An activin receptor-like kinase 5 inhibitor reduces collagen deposition in a rat dermal incision wound healing model.

Bian F, Render J, Ren XD, Chio C, Chan K, Boys M, Lala DS, Pocalyko D. Bian F, et al. Plast Reconstr Surg. 2011 Nov;128(5):451e-459e. doi: 10.1097/PRS.0b013e31822b65c7. Plast Reconstr Surg. 2011. PMID: 22030504

3

Diphenyl ethers as androgen receptor antagonists for the topical suppression of sebum production.

Mitchell LH, Hu LY, Nguyen M, Fakhoury S, Smith Y, Iula D, Kostlan C, Carroll M, Dettling D, Du D, Pocalyko D, Wade K, Lefker B. Mitchell LH, et al. Bioorg Med Chem Lett. 2009 Apr 15;19(8):2176-8. doi: 10.1016/j.bmcl.2009.02.104. Epub 2009 Mar 3. Bioorg Med Chem Lett. 2009. PMID: 19286380

4

Pantolactams as androgen receptor antagonists for the topical suppression of sebum production.

Sexton KE, Barrett S, Bridgwood K, Carroll M, Dettling D, Du D, Fakhoury S, Fedij V, Hu LY, Kostlan C, Pocalyko D, Raheja N, Smith Y, Shanmugasundaram V, Wade K. Sexton KE, et al. Bioorg Med Chem Lett. 2011 Sep 15;21(18):5230-3. doi: 10.1016/j.bmcl.2011.07.048. Epub 2011 Jul 23. Bioorg Med Chem Lett. 2011. PMID: 21831636

5

Preparation of 4-aryl-2-trifluoromethylbenzonitrile derivatives as androgen receptor antagonists for topical suppression of sebum production.

Van Camp JA, Hu LY, Kostlan C, Lefker B, Li J, Mitchell L, Wang Z, Yue WS, Carroll M, Dettling D, Du D, Pocalyko D, Wade K. Van Camp JA, et al. Bioorg Med Chem Lett. 2007 Oct 15;17(20):5529-32. doi: 10.1016/j.bmcl.2007.08.034. Epub 2007 Aug 19. Bioorg Med Chem Lett. 2007. PMID: 17764935

6

Synthesis and biological evaluation of amino-pyridines as androgen receptor antagonists for stimulating hair growth and reducing sebum production.

Hu LY, Lei HJ, Du D, Johnson TR, Fedij V, Kostlan C, Yue WS, Lovdahl M, Li JJ, Carroll M, Dettling D, Asbill J, Fan C, Wade K, Pocalyko D, Lapham K, Yalamanchili R, Samas B, Vrieze D, Ciotti S, Krieger-Burke T, Sliskovic D, Welgus H. Hu LY, et al. Bioorg Med Chem Lett. 2007 Oct 15;17(20):5693-7. doi: 10.1016/j.bmcl.2007.07.059. Epub 2007 Aug 19. Bioorg Med Chem Lett. 2007. PMID: 17766112

7

(1R,2S)-4-(2-cyano-cyclohexyl-oxy)-2-trifluoromethyl-benzonitrile, a potent androgen receptor antagonist for stimulating hair growth and reducing sebum production.

Hu LY, Du D, Hoffman J, Smith Y, Fedij V, Kostlan C, Johnson TR, Huang Y, Kesten S, Harter W, Yue WS, Li JJ, Barvian N, Mitchell L, Lei HJ, Lefker B, Carroll M, Dettling D, Krieger-Burke T, Samas B, Yalamanchili R, Lapham K, Pocalyko D, Sliskovic D, Ciotti S, Stoller B, Hena MA, Ding Q, Maiti SN, Stier M, Welgus H. Hu LY, et al. Bioorg Med Chem Lett. 2007 Nov 1;17(21):5983-8. doi: 10.1016/j.bmcl.2007.07.075. Epub 2007 Aug 21. Bioorg Med Chem Lett. 2007. PMID: 17827000

8

4-(Alkylthio)- and 4-(arylthio)-benzonitrile derivatives as androgen receptor antagonists for the topical suppression of sebum production.

Mitchell L, Wang Z, Hu LY, Kostlan C, Carroll M, Dettling D, Du D, Pocalyko D, Wade K. Mitchell L, et al. Bioorg Med Chem Lett. 2009 Mar 1;19(5):1310-3. doi: 10.1016/j.bmcl.2009.01.063. Epub 2009 Jan 27. Bioorg Med Chem Lett. 2009. PMID: 19201190

9

Rational design of a topical androgen receptor antagonist for the suppression of sebum production with properties suitable for follicular delivery.

Mitchell LH, Johnson TR, Lu GW, Du D, Datta K, Grzemski F, Shanmugasundaram V, Spence J, Wade K, Wang Z, Sun K, Lin K, Hu LY, Sexton K, Raheja N, Kostlan C, Pocalyko D. Mitchell LH, et al. J Med Chem. 2010 Jun 10;53(11):4422-7. doi: 10.1021/jm9018004. J Med Chem. 2010. PMID: 20462217

10

Integrative Analysis of DiseaseLand Omics Database for Disease Signatures and Treatments: A Bipolar Case Study.

Wu C, Huang BE, Chen G, Lovenberg TW, Pocalyko DJ, Yao X. Wu C, et al. Among authors: pocalyko dj. Front Genet. 2019 Apr 30;10:396. doi: 10.3389/fgene.2019.00396. eCollection 2019. Front Genet. 2019. PMID: 31114610 Free PMC article.

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