Kojetin D - Search Results

1

Synthesis and SAR of tetrahydroisoquinolines as Rev-erbα agonists.

Noel R, Song X, Shin Y, Banerjee S, Kojetin D, Lin L, Ruiz CH, Cameron MD, Burris TP, Kamenecka TM. Noel R, et al. Among authors: kojetin d. Bioorg Med Chem Lett. 2012 Jun 1;22(11):3739-42. doi: 10.1016/j.bmcl.2012.04.023. Epub 2012 Apr 13. Bioorg Med Chem Lett. 2012. PMID: 22560469 Free PMC article.

2

Implications of the binding of tamoxifen to the coactivator recognition site of the estrogen receptor.

Kojetin DJ, Burris TP, Jensen EV, Khan SA. Kojetin DJ, et al. Endocr Relat Cancer. 2008 Dec;15(4):851-70. doi: 10.1677/ERC-07-0281. Epub 2008 Aug 28. Endocr Relat Cancer. 2008. PMID: 18755852 Review.

3

Characterization of the core mammalian clock component, NPAS2, as a REV-ERBalpha/RORalpha target gene.

Crumbley C, Wang Y, Kojetin DJ, Burris TP. Crumbley C, et al. J Biol Chem. 2010 Nov 12;285(46):35386-92. doi: 10.1074/jbc.M110.129288. Epub 2010 Sep 3. J Biol Chem. 2010. PMID: 20817722 Free PMC article.

4

Identification of SR8278, a synthetic antagonist of the nuclear heme receptor REV-ERB.

Kojetin D, Wang Y, Kamenecka TM, Burris TP. Kojetin D, et al. ACS Chem Biol. 2011 Feb 18;6(2):131-4. doi: 10.1021/cb1002575. Epub 2010 Nov 10. ACS Chem Biol. 2011. PMID: 21043485 Free PMC article.

5

Identification of SR3335 (ML-176): a synthetic RORα selective inverse agonist.

Kumar N, Kojetin DJ, Solt LA, Kumar KG, Nuhant P, Duckett DR, Cameron MD, Butler AA, Roush WR, Griffin PR, Burris TP. Kumar N, et al. Among authors: kojetin dj. ACS Chem Biol. 2011 Mar 18;6(3):218-22. doi: 10.1021/cb1002762. Epub 2010 Dec 6. ACS Chem Biol. 2011. PMID: 21090593 Free PMC article.

6

A role for rev-erbα ligands in regulation of adipogenesis.

Kojetin DJ, Burris TP. Kojetin DJ, et al. Curr Pharm Des. 2011;17(4):320-4. doi: 10.2174/138161211795164211. Curr Pharm Des. 2011. PMID: 21375499 Review.

7

DNA binding alters coactivator interaction surfaces of the intact VDR-RXR complex.

Zhang J, Chalmers MJ, Stayrook KR, Burris LL, Wang Y, Busby SA, Pascal BD, Garcia-Ordonez RD, Bruning JB, Istrate MA, Kojetin DJ, Dodge JA, Burris TP, Griffin PR. Zhang J, et al. Among authors: kojetin dj. Nat Struct Mol Biol. 2011 May;18(5):556-63. doi: 10.1038/nsmb.2046. Epub 2011 Apr 10. Nat Struct Mol Biol. 2011. PMID: 21478866 Free PMC article.

8

The REV-ERBs and RORs: molecular links between circadian rhythms and lipid homeostasis.

Solt LA, Kojetin DJ, Burris TP. Solt LA, et al. Future Med Chem. 2011 Apr;3(5):623-38. doi: 10.4155/fmc.11.9. Future Med Chem. 2011. PMID: 21526899 Free PMC article. Review.

9

Structural and biophysical insights into the ligand-free Pitx2 homeodomain and a ring dermoid of the cornea inducing homeodomain mutant.

Doerdelmann T, Kojetin DJ, Baird-Titus JM, Solt LA, Burris TP, Rance M. Doerdelmann T, et al. Biochemistry. 2012 Jan 17;51(2):665-76. doi: 10.1021/bi201639x. Epub 2012 Jan 6. Biochemistry. 2012. PMID: 22224469 Free PMC article.

10

Ligand and receptor dynamics contribute to the mechanism of graded PPARγ agonism.

Hughes TS, Chalmers MJ, Novick S, Kuruvilla DS, Chang MR, Kamenecka TM, Rance M, Johnson BA, Burris TP, Griffin PR, Kojetin DJ. Hughes TS, et al. Structure. 2012 Jan 11;20(1):139-50. doi: 10.1016/j.str.2011.10.018. Structure. 2012. PMID: 22244763 Free PMC article.

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