Lacivita E - Search Results

1

Investigations on the 1-(2-biphenyl)piperazine motif: identification of new potent and selective ligands for the serotonin(7) (5-HT(7)) receptor with agonist or antagonist action in vitro or ex vivo.

Lacivita E, Patarnello D, Stroth N, Caroli A, Niso M, Contino M, De Giorgio P, Di Pilato P, Colabufo NA, Berardi F, Perrone R, Svenningsson P, Hedlund PB, Leopoldo M. Lacivita E, et al. J Med Chem. 2012 Jul 26;55(14):6375-80. doi: 10.1021/jm3003679. Epub 2012 Jul 11. J Med Chem. 2012. PMID: 22738316

2

trans-4-[4-(Methoxyphenyl)cyclohexyl]-1-arylpiperazines: a new class of potent and selective 5-HT(1A) receptor ligands as conformationally constrained analogues of 4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]-1-arylpiperazines.

Perrone R, Berardi F, Colabufo NA, Leopoldo M, Lacivita E, Tortorella V, Leonardi A, Poggesi E, Testa R. Perrone R, et al. Among authors: lacivita e. J Med Chem. 2001 Dec 6;44(25):4431-42. doi: 10.1021/jm010866v. J Med Chem. 2001. PMID: 11728188

3

Structure-affinity relationship study on N-[4-(4-arylpiperazin-1-yl)butyl]arylcarboxamides as potent and selective dopamine D(3) receptor ligands.

Leopoldo M, Berardi F, Colabufo NA, De Giorgio P, Lacivita E, Perrone R, Tortorella V. Leopoldo M, et al. Among authors: lacivita e. J Med Chem. 2002 Dec 19;45(26):5727-35. doi: 10.1021/jm020952a. J Med Chem. 2002. PMID: 12477356

4

Synthesis and structure-affinity relationships of 1-[omega-(4-aryl-1-piperazinyl)alkyl]-1-aryl ketones as 5-HT(7) receptor ligands.

Perrone R, Berardi F, Colabufo NA, Lacivita E, Leopoldo M, Tortorella V. Perrone R, et al. Among authors: lacivita e. J Med Chem. 2003 Feb 13;46(4):646-9. doi: 10.1021/jm020994z. J Med Chem. 2003. PMID: 12570387

5

Studies on 1-arylpiperazine derivatives with affinity for rat 5-HT7 and 5-HT1A receptors.

Leopoldo M, Berardi F, Colabufo NA, Contino M, Lacivita E, Perrone R, Tortorella V. Leopoldo M, et al. Among authors: lacivita e. J Pharm Pharmacol. 2004 Feb;56(2):247-55. doi: 10.1211/0022357022575. J Pharm Pharmacol. 2004. PMID: 15005884

6

Structure-affinity relationship study on N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4-aryl-1-piperazinealkylamides, a new class of 5-hydroxytryptamine7 receptor agents.

Leopoldo M, Berardi F, Colabufo NA, Contino M, Lacivita E, Niso M, Perrone R, Tortorella V. Leopoldo M, et al. Among authors: lacivita e. J Med Chem. 2004 Dec 16;47(26):6616-24. doi: 10.1021/jm049702f. J Med Chem. 2004. PMID: 15588097

7

11C-labeling of n-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]arylcarboxamide derivatives and evaluation as potential radioligands for PET imaging of dopamine D3 receptors.

Turolla EA, Matarrese M, Belloli S, Moresco RM, Simonelli P, Todde S, Fazio F, Magni F, Kienle MG, Leopoldo M, Berardi F, Colabufo NA, Lacivita E, Perrone R. Turolla EA, et al. Among authors: lacivita e. J Med Chem. 2005 Nov 3;48(22):7018-23. doi: 10.1021/jm050171k. J Med Chem. 2005. PMID: 16250661

8

Design and synthesis of long-chain arylpiperazines with mixed affinity for serotonin transporter (SERT) and 5-HT(1A) receptor.

Perrone R, Berardi F, Colabufo NA, Lacivita E, Larizza C, Leopoldo M, Tortorella V. Perrone R, et al. Among authors: lacivita e. J Pharm Pharmacol. 2005 Oct;57(10):1319-27. doi: 10.1211/jpp.57.10.0011. J Pharm Pharmacol. 2005. PMID: 16259761

9

First structure-activity relationship study on dopamine D3 receptor agents with N-[4-(4-arylpiperazin-1-yl)butyl]arylcarboxamide structure.

Leopoldo M, Lacivita E, Colabufo NA, Contino M, Berardi F, Perrone R. Leopoldo M, et al. Among authors: lacivita e. J Med Chem. 2005 Dec 15;48(25):7919-22. doi: 10.1021/jm050729o. J Med Chem. 2005. PMID: 16335915

10

Design, synthesis, and binding affinities of potential positron emission tomography (PET) ligands for visualization of brain dopamine D3 receptors.

Leopoldo M, Lacivita E, De Giorgio P, Colabufo NA, Niso M, Berardi F, Perrone R. Leopoldo M, et al. Among authors: lacivita e. J Med Chem. 2006 Jan 12;49(1):358-65. doi: 10.1021/jm050734s. J Med Chem. 2006. PMID: 16392820

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