Bunch L - Search Results

1

Design, synthesis and pharmacological characterization of coumarin-based fluorescent analogs of excitatory amino acid transporter subtype 1 selective inhibitors, UCPH-101 and UCPH-102.

Huynh TH, Abrahamsen B, Madsen KK, Gonzalez-Franquesa A, Jensen AA, Bunch L. Huynh TH, et al. Among authors: bunch l. Bioorg Med Chem. 2012 Dec 1;20(23):6831-9. doi: 10.1016/j.bmc.2012.09.049. Epub 2012 Oct 2. Bioorg Med Chem. 2012. PMID: 23072958

2

Synthesis and receptor binding affinity of new selective GluR5 ligands.

Bunch L, Johansen TH, Bräuner-Osborne H, Stensbøl TB, Johansen TN, Krogsgaard-Larsen P, Madsen U. Bunch L, et al. Bioorg Med Chem. 2001 Apr;9(4):875-9. doi: 10.1016/s0968-0896(00)00304-7. Bioorg Med Chem. 2001. PMID: 11354670

3

Rational design, synthesis, and pharmacological evaluation of 2-azanorbornane-3-exo,5-endo-dicarboxylic acid: a novel conformationally restricted glutamic acid analogue.

Bunch L, Liljefors T, Greenwood JR, Frydenvang K, Bräuner-Osborne H, Krogsgaard-Larsen P, Madsen U. Bunch L, et al. J Org Chem. 2003 Feb 21;68(4):1489-95. doi: 10.1021/jo026509p. J Org Chem. 2003. PMID: 12585893

4

Azetidinic amino acids: stereocontrolled synthesis and pharmacological characterization as ligands for glutamate receptors and transporters.

Bräuner-Osborne H, Bunch L, Chopin N, Couty F, Evano G, Jensen AA, Kusk M, Nielsen B, Rabasso N. Bräuner-Osborne H, et al. Among authors: bunch l. Org Biomol Chem. 2005 Nov 7;3(21):3926-36. doi: 10.1039/b509514j. Epub 2005 Sep 29. Org Biomol Chem. 2005. PMID: 16240010

5

Chemoenzymatic synthesis of a series of 4-substituted glutamate analogues and pharmacological characterization at human glutamate transporters subtypes 1-3.

Alaux S, Kusk M, Sagot E, Bolte J, Jensen AA, Bräuner-Osborne H, Gefflaut T, Bunch L. Alaux S, et al. Among authors: bunch l. J Med Chem. 2005 Dec 15;48(25):7980-92. doi: 10.1021/jm050597z. J Med Chem. 2005. PMID: 16335922

6

Rational design and enantioselective synthesis of (1R,4S,5R,6S)-3-azabicyclo[3.3.0]octane-4,6-dicarboxylic acid - a novel inhibitor at human glutamate transporter subtypes 1, 2, and 3.

Bunch L, Nielsen B, Jensen AA, Bräuner-Osborne H. Bunch L, et al. J Med Chem. 2006 Jan 12;49(1):172-8. doi: 10.1021/jm0508336. J Med Chem. 2006. PMID: 16392801

7

Stereoselective chemoenzymatic synthesis of the four stereoisomers of l-2-(2-carboxycyclobutyl)glycine and pharmacological characterization at human excitatory amino acid transporter subtypes 1, 2, and 3.

Faure S, Jensen AA, Maurat V, Gu X, Sagot E, Aitken DJ, Bolte J, Gefflaut T, Bunch L. Faure S, et al. Among authors: bunch l. J Med Chem. 2006 Nov 2;49(22):6532-8. doi: 10.1021/jm060822s. J Med Chem. 2006. PMID: 17064071

8

Chemo-enzymatic synthesis of (2S,4R)-2-amino-4-(3-(2,2-diphenylethylamino)-3-oxopropyl)pentanedioic acid: a novel selective inhibitor of human excitatory amino acid transporter subtype 2.

Sagot E, Jensen AA, Pickering DS, Pu X, Umberti M, Stensbøl TB, Nielsen B, Assaf Z, Aboab B, Bolte J, Gefflaut T, Bunch L. Sagot E, et al. Among authors: bunch l. J Med Chem. 2008 Jul 24;51(14):4085-92. doi: 10.1021/jm800091e. Epub 2008 Jun 25. J Med Chem. 2008. PMID: 18578477 Free article.

9

Subtype selective kainic acid receptor agonists: discovery and approaches to rational design.

Bunch L, Krogsgaard-Larsen P. Bunch L, et al. Med Res Rev. 2009 Jan;29(1):3-28. doi: 10.1002/med.20133. Med Res Rev. 2009. PMID: 18623169 Review.

10

Discovery of the first selective inhibitor of excitatory amino acid transporter subtype 1.

Jensen AA, Erichsen MN, Nielsen CW, Stensbøl TB, Kehler J, Bunch L. Jensen AA, et al. Among authors: bunch l. J Med Chem. 2009 Feb 26;52(4):912-5. doi: 10.1021/jm8013458. J Med Chem. 2009. PMID: 19161278

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