Díaz JF - Search Results

1

Synthesis and biological evaluation of colchicine C-ring analogues tethered with aliphatic linkers suitable for prodrug derivatisation.

Fournier-Dit-Chabert J, Vinader V, Santos AR, Redondo-Horcajo M, Dreneau A, Basak R, Cosentino L, Marston G, Abdel-Rahman H, Loadman PM, Shnyder SD, Díaz JF, Barasoain I, Falconer RA, Pors K. Fournier-Dit-Chabert J, et al. Among authors: diaz jf. Bioorg Med Chem Lett. 2012 Dec 15;22(24):7693-6. doi: 10.1016/j.bmcl.2012.09.104. Epub 2012 Oct 10. Bioorg Med Chem Lett. 2012. PMID: 23103097

2

Fast kinetics of Taxol binding to microtubules. Effects of solution variables and microtubule-associated proteins.

Díaz JF, Barasoain I, Andreu JM. Díaz JF, et al. J Biol Chem. 2003 Mar 7;278(10):8407-19. doi: 10.1074/jbc.M211163200. Epub 2002 Dec 20. J Biol Chem. 2003. PMID: 12496245 Free article.

3

Macromolecular accessibility of fluorescent taxoids bound at a paclitaxel binding site in the microtubule surface.

Díaz JF, Barasoain I, Souto AA, Amat-Guerri F, Andreu JM. Díaz JF, et al. J Biol Chem. 2005 Feb 4;280(5):3928-37. doi: 10.1074/jbc.M407816200. Epub 2004 Nov 18. J Biol Chem. 2005. PMID: 15550392 Free article.

4

Design, synthesis and biological evaluation of novel, simplified analogues of laulimalide: modification of the side chain.

Paterson I, Menche D, Håkansson AE, Longstaff A, Wong D, Barasoain I, Buey RM, Díaz JF. Paterson I, et al. Among authors: diaz jf. Bioorg Med Chem Lett. 2005 May 2;15(9):2243-7. doi: 10.1016/j.bmcl.2005.03.018. Bioorg Med Chem Lett. 2005. PMID: 15837302

5

Microtubule interactions with chemically diverse stabilizing agents: thermodynamics of binding to the paclitaxel site predicts cytotoxicity.

Buey RM, Barasoain I, Jackson E, Meyer A, Giannakakou P, Paterson I, Mooberry S, Andreu JM, Díaz JF. Buey RM, et al. Among authors: diaz jf. Chem Biol. 2005 Dec;12(12):1269-79. doi: 10.1016/j.chembiol.2005.09.010. Chem Biol. 2005. PMID: 16356844

6

Overcoming tumor drug resistance with high-affinity taxanes: a SAR study of C2-modified 7-acyl-10-deacetyl cephalomannines.

Yang CG, Barasoain I, Li X, Matesanz R, Liu R, Sharom FJ, Yin DL, Díaz JF, Fang WS. Yang CG, et al. Among authors: diaz jf. ChemMedChem. 2007 May;2(5):691-701. doi: 10.1002/cmdc.200700002. ChemMedChem. 2007. PMID: 17385753

7

Synthesis, biological evaluations, and tubulin binding poses of C-2alpha sulfur linked taxol analogues.

Wang L, Alcaraz AA, Matesanz R, Yang CG, Barasoain I, Díaz JF, Li YZ, Snyder JP, Fang WS. Wang L, et al. Among authors: diaz jf. Bioorg Med Chem Lett. 2007 Jun 1;17(11):3191-4. doi: 10.1016/j.bmcl.2007.03.026. Epub 2007 Mar 14. Bioorg Med Chem Lett. 2007. PMID: 17395465

8

Arylthioindole inhibitors of tubulin polymerization. 3. Biological evaluation, structure-activity relationships and molecular modeling studies.

La Regina G, Edler MC, Brancale A, Kandil S, Coluccia A, Piscitelli F, Hamel E, De Martino G, Matesanz R, Díaz JF, Scovassi AI, Prosperi E, Lavecchia A, Novellino E, Artico M, Silvestri R. La Regina G, et al. Among authors: diaz jf. J Med Chem. 2007 Jun 14;50(12):2865-74. doi: 10.1021/jm061479u. Epub 2007 May 12. J Med Chem. 2007. PMID: 17497841

9

The total synthesis and biological properties of the cytotoxic macrolide FD-891 and its non-natural (Z)-C12 isomer.

García-Fortanet J, Murga J, Carda M, Marco JA, Matesanz R, Díaz JF, Barasoain I. García-Fortanet J, et al. Among authors: diaz jf. Chemistry. 2007;13(18):5060-74. doi: 10.1002/chem.200700342. Chemistry. 2007. PMID: 17516610

10

Optimization of taxane binding to microtubules: binding affinity dissection and incremental construction of a high-affinity analog of paclitaxel.

Matesanz R, Barasoain I, Yang CG, Wang L, Li X, de Inés C, Coderch C, Gago F, Barbero JJ, Andreu JM, Fang WS, Díaz JF. Matesanz R, et al. Among authors: diaz jf. Chem Biol. 2008 Jun;15(6):573-85. doi: 10.1016/j.chembiol.2008.05.008. Chem Biol. 2008. PMID: 18559268

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