Stewart EL - Search Results

1

Rational design of potent non-nucleoside inhibitors of HIV-1 reverse transcriptase.

Chong P, Sebahar P, Youngman M, Garrido D, Zhang H, Stewart EL, Nolte RT, Wang L, Ferris RG, Edelstein M, Weaver K, Mathis A, Peat A. Chong P, et al. Among authors: stewart el. J Med Chem. 2012 Dec 13;55(23):10601-9. doi: 10.1021/jm301294g. Epub 2012 Nov 26. J Med Chem. 2012. PMID: 23137340

2

2-Amino-4,6-diarylpyridines as novel ligands for the estrogen receptor.

Henke BR, Drewry DH, Jones SA, Stewart EL, Weaver SL, Wiethe RW. Henke BR, et al. Among authors: stewart el. Bioorg Med Chem Lett. 2001 Jul 23;11(14):1939-42. doi: 10.1016/s0960-894x(01)00321-3. Bioorg Med Chem Lett. 2001. PMID: 11459665

3

A new series of estrogen receptor modulators that display selectivity for estrogen receptor beta.

Henke BR, Consler TG, Go N, Hale RL, Hohman DR, Jones SA, Lu AT, Moore LB, Moore JT, Orband-Miller LA, Robinett RG, Shearin J, Spearing PK, Stewart EL, Turnbull PS, Weaver SL, Williams SP, Wisely GB, Lambert MH. Henke BR, et al. Among authors: stewart el. J Med Chem. 2002 Dec 5;45(25):5492-505. doi: 10.1021/jm020291h. J Med Chem. 2002. PMID: 12459017

4

Progesterone receptor ligand binding pocket flexibility: crystal structures of the norethindrone and mometasone furoate complexes.

Madauss KP, Deng SJ, Austin RJ, Lambert MH, McLay I, Pritchard J, Short SA, Stewart EL, Uings IJ, Williams SP. Madauss KP, et al. Among authors: stewart el. J Med Chem. 2004 Jun 17;47(13):3381-7. doi: 10.1021/jm030640n. J Med Chem. 2004. PMID: 15189034

5

Discovery of non-steroidal mifepristone mimetics: pyrazoline-based PR antagonists.

Jones DG, Liang X, Stewart EL, Noe RA, Kallander LS, Madauss KP, Williams SP, Thompson SK, Gray DW, Hoekstra WJ. Jones DG, et al. Among authors: stewart el. Bioorg Med Chem Lett. 2005 Jul 1;15(13):3203-6. doi: 10.1016/j.bmcl.2005.05.001. Bioorg Med Chem Lett. 2005. PMID: 15925510

6

Array synthesis of progesterone receptor antagonists: 3-aryl-1,2-diazepines.

Wiethe RW, Stewart EL, Drewry DH, Gray DW, Mehbob A, Hoekstra WJ. Wiethe RW, et al. Among authors: stewart el. Bioorg Med Chem Lett. 2006 Jul 15;16(14):3777-9. doi: 10.1016/j.bmcl.2006.04.055. Epub 2006 May 5. Bioorg Med Chem Lett. 2006. PMID: 16678409

7

Structure-guided design of N-phenyl tertiary amines as transrepression-selective liver X receptor modulators with anti-inflammatory activity.

Chao EY, Caravella JA, Watson MA, Campobasso N, Ghisletti S, Billin AN, Galardi C, Wang P, Laffitte BA, Iannone MA, Goodwin BJ, Nichols JA, Parks DJ, Stewart E, Wiethe RW, Williams SP, Smallwood A, Pearce KH, Glass CK, Willson TM, Zuercher WJ, Collins JL. Chao EY, et al. J Med Chem. 2008 Sep 25;51(18):5758-65. doi: 10.1021/jm800612u. J Med Chem. 2008. PMID: 18800767

8

The first X-ray crystal structure of the glucocorticoid receptor bound to a non-steroidal agonist.

Madauss KP, Bledsoe RK, Mclay I, Stewart EL, Uings IJ, Weingarten G, Williams SP. Madauss KP, et al. Among authors: stewart el. Bioorg Med Chem Lett. 2008 Dec 1;18(23):6097-9. doi: 10.1016/j.bmcl.2008.10.021. Epub 2008 Oct 8. Bioorg Med Chem Lett. 2008. PMID: 18952422

9

Discovery of tertiary sulfonamides as potent liver X receptor antagonists.

Zuercher WJ, Buckholz RG, Campobasso N, Collins JL, Galardi CM, Gampe RT, Hyatt SM, Merrihew SL, Moore JT, Oplinger JA, Reid PR, Spearing PK, Stanley TB, Stewart EL, Willson TM. Zuercher WJ, et al. Among authors: stewart el. J Med Chem. 2010 Apr 22;53(8):3412-6. doi: 10.1021/jm901797p. J Med Chem. 2010. PMID: 20345102

10

Structure guided design of 5-arylindazole glucocorticoid receptor agonists and antagonists.

Yates CM, Brown PJ, Stewart EL, Patten C, Austin RJ, Holt JA, Maglich JM, Angell DC, Sasse RZ, Taylor SJ, Uings IJ, Trump RP. Yates CM, et al. Among authors: stewart el. J Med Chem. 2010 Jun 10;53(11):4531-44. doi: 10.1021/jm100447c. J Med Chem. 2010. PMID: 20469868

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