Scapozza L - Search Results

1

Naphthoquinone derivatives exert their antitrypanosomal activity via a multi-target mechanism.

Pieretti S, Haanstra JR, Mazet M, Perozzo R, Bergamini C, Prati F, Fato R, Lenaz G, Capranico G, Brun R, Bakker BM, Michels PA, Scapozza L, Bolognesi ML, Cavalli A. Pieretti S, et al. Among authors: scapozza l. PLoS Negl Trop Dis. 2013;7(1):e2012. doi: 10.1371/journal.pntd.0002012. Epub 2013 Jan 17. PLoS Negl Trop Dis. 2013. PMID: 23350008 Free PMC article.

2

Single-molecule pulling simulations can discern active from inactive enzyme inhibitors.

Colizzi F, Perozzo R, Scapozza L, Recanatini M, Cavalli A. Colizzi F, et al. Among authors: scapozza l. J Am Chem Soc. 2010 Jun 2;132(21):7361-71. doi: 10.1021/ja100259r. J Am Chem Soc. 2010. PMID: 20462212

3

Crystal structures of T. b. rhodesiense adenosine kinase complexed with inhibitor and activator: implications for catalysis and hyperactivation.

Kuettel S, Greenwald J, Kostrewa D, Ahmed S, Scapozza L, Perozzo R. Kuettel S, et al. Among authors: scapozza l. PLoS Negl Trop Dis. 2011 May;5(5):e1164. doi: 10.1371/journal.pntd.0001164. Epub 2011 May 24. PLoS Negl Trop Dis. 2011. PMID: 21629723 Free PMC article.

4

Design, synthesis, and biological and crystallographic evaluation of novel inhibitors of Plasmodium falciparum enoyl-ACP-reductase (PfFabI).

Belluti F, Perozzo R, Lauciello L, Colizzi F, Kostrewa D, Bisi A, Gobbi S, Rampa A, Bolognesi ML, Recanatini M, Brun R, Scapozza L, Cavalli A. Belluti F, et al. Among authors: scapozza l. J Med Chem. 2013 Oct 10;56(19):7516-26. doi: 10.1021/jm400637m. Epub 2013 Sep 25. J Med Chem. 2013. PMID: 24063369

5

Adenosine Kinase of T. b. Rhodesiense identified as the putative target of 4-[5-(4-phenoxyphenyl)-2H-pyrazol-3-yl]morpholine using chemical proteomics.

Kuettel S, Mosimann M, Mäser P, Kaiser M, Brun R, Scapozza L, Perozzo R. Kuettel S, et al. Among authors: scapozza l. PLoS Negl Trop Dis. 2009 Aug 25;3(8):e506. doi: 10.1371/journal.pntd.0000506. PLoS Negl Trop Dis. 2009. PMID: 19707572 Free PMC article.

6

Inhibition of Plasmodium falciparum fatty acid biosynthesis: evaluation of FabG, FabZ, and FabI as drug targets for flavonoids.

Tasdemir D, Lack G, Brun R, Rüedi P, Scapozza L, Perozzo R. Tasdemir D, et al. Among authors: scapozza l. J Med Chem. 2006 Jun 1;49(11):3345-53. doi: 10.1021/jm0600545. J Med Chem. 2006. PMID: 16722653

7

Synthesis and evaluation of antiparasitic activities of new 4-[5-(4-phenoxyphenyl)-2H-pyrazol-3-yl]morpholine derivatives.

Kuettel S, Zambon A, Kaiser M, Brun R, Scapozza L, Perozzo R. Kuettel S, et al. Among authors: scapozza l. J Med Chem. 2007 Nov 15;50(23):5833-9. doi: 10.1021/jm700938n. Epub 2007 Oct 20. J Med Chem. 2007. PMID: 17949068

8

Structure-based drug design and in vitro testing reveal new inhibitors of enoyl-acyl carrier protein reductases.

Ghattas MA, Eissa NA, Tessaro F, Perozzo R, Scapozza L, Obaid D, Atatreh N. Ghattas MA, et al. Among authors: scapozza l. Chem Biol Drug Des. 2019 Aug;94(2):1545-1555. doi: 10.1111/cbdd.13536. Epub 2019 Jun 2. Chem Biol Drug Des. 2019. PMID: 31063658

9

Expression, purification and biochemical characterization of recombinant Ca-dependent protein kinase 2 of the malaria parasite Plasmodium falciparum.

Lauciello L, Kappes B, Scapozza L, Perozzo R. Lauciello L, et al. Among authors: scapozza l. Protein Expr Purif. 2013 Aug;90(2):170-7. doi: 10.1016/j.pep.2013.06.006. Epub 2013 Jun 18. Protein Expr Purif. 2013. PMID: 23792132

10

Synthesis of 3-azabicyclo[3.2.2]nonanes and their antiprotozoal activities.

Seebacher W, Wolkinger V, Faist J, Kaiser M, Brun R, Saf R, Bucar F, Gröblacher B, Brantner A, Merino V, Kalia Y, Scapozza L, Perozzo R, Weis R. Seebacher W, et al. Among authors: scapozza l. Bioorg Med Chem Lett. 2015 Apr 1;25(7):1390-3. doi: 10.1016/j.bmcl.2015.02.044. Epub 2015 Feb 28. Bioorg Med Chem Lett. 2015. PMID: 25746816

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