Kaiser M - Search Results

1

Optimization of triazine nitriles as rhodesain inhibitors: structure-activity relationships, bioisosteric imidazopyridine nitriles, and X-ray crystal structure analysis with human cathepsin L.

Ehmke V, Winkler E, Banner DW, Haap W, Schweizer WB, Rottmann M, Kaiser M, Freymond C, Schirmeister T, Diederich F. Ehmke V, et al. Among authors: kaiser m. ChemMedChem. 2013 Jun;8(6):967-75. doi: 10.1002/cmdc.201300112. Epub 2013 May 9. ChemMedChem. 2013. PMID: 23658062

2

Betraying the parasite's redox system: diaryl sulfide-based inhibitors of trypanothione reductase: subversive substrates and antitrypanosomal properties.

Stump B, Kaiser M, Brun R, Krauth-Siegel RL, Diederich F. Stump B, et al. Among authors: kaiser m. ChemMedChem. 2007 Dec;2(12):1708-12. doi: 10.1002/cmdc.200700172. ChemMedChem. 2007. PMID: 17918760 No abstract available.

3

Diaryl sulfide-based inhibitors of trypanothione reductase: inhibition potency, revised binding mode and antiprotozoal activities.

Stump B, Eberle C, Kaiser M, Brun R, Krauth-Siegel RL, Diederich F. Stump B, et al. Among authors: kaiser m. Org Biomol Chem. 2008 Nov 7;6(21):3935-47. doi: 10.1039/b806371k. Epub 2008 Sep 9. Org Biomol Chem. 2008. PMID: 18931800

4

Pentafluorosulfanyl as a novel building block for enzyme inhibitors: trypanothione reductase inhibition and antiprotozoal activities of diarylamines.

Stump B, Eberle C, Schweizer WB, Kaiser M, Brun R, Krauth-Siegel RL, Lentz D, Diederich F. Stump B, et al. Among authors: kaiser m. Chembiochem. 2009 Jan 5;10(1):79-83. doi: 10.1002/cbic.200800565. Chembiochem. 2009. PMID: 19058274 No abstract available.

5

Synthesis, inhibition potency, binding mode, and antiprotozoal activities of fluorescent inhibitors of trypanothione reductase based on mepacrine-conjugated diaryl sulfide scaffolds.

Eberle C, Burkhard JA, Stump B, Kaiser M, Brun R, Krauth-Siegel RL, Diederich F. Eberle C, et al. Among authors: kaiser m. ChemMedChem. 2009 Dec;4(12):2034-44. doi: 10.1002/cmdc.200900327. ChemMedChem. 2009. PMID: 19847846

6

Improved inhibitors of trypanothione reductase by combination of motifs: synthesis, inhibitory potency, binding mode, and antiprotozoal activities.

Eberle C, Lauber BS, Fankhauser D, Kaiser M, Brun R, Krauth-Siegel RL, Diederich F. Eberle C, et al. Among authors: kaiser m. ChemMedChem. 2011 Feb 7;6(2):292-301. doi: 10.1002/cmdc.201000420. Epub 2010 Dec 16. ChemMedChem. 2011. PMID: 21275053

7

Identification of 1,3-diiminoisoindoline carbohydrazides as potential antimalarial candidates.

Mombelli P, Witschel MC, van Zijl AW, Geist JG, Rottmann M, Freymond C, Röhl F, Kaiser M, Illarionova V, Fischer M, Siepe I, Schweizer WB, Brun R, Diederich F. Mombelli P, et al. Among authors: kaiser m. ChemMedChem. 2012 Jan 2;7(1):151-8. doi: 10.1002/cmdc.201100441. Epub 2011 Nov 16. ChemMedChem. 2012. PMID: 22095896

8

Antiparasitic agents: new drugs on the horizon.

Mäser P, Wittlin S, Rottmann M, Wenzler T, Kaiser M, Brun R. Mäser P, et al. Among authors: kaiser m. Curr Opin Pharmacol. 2012 Oct;12(5):562-6. doi: 10.1016/j.coph.2012.05.001. Epub 2012 May 29. Curr Opin Pharmacol. 2012. PMID: 22652215 Review.

9

Agrochemicals against malaria, sleeping sickness, leishmaniasis and Chagas disease.

Witschel M, Rottmann M, Kaiser M, Brun R. Witschel M, et al. Among authors: kaiser m. PLoS Negl Trop Dis. 2012;6(10):e1805. doi: 10.1371/journal.pntd.0001805. Epub 2012 Oct 25. PLoS Negl Trop Dis. 2012. PMID: 23145187 Free PMC article.

10

Binding to large enzyme pockets: small-molecule inhibitors of trypanothione reductase.

Persch E, Bryson S, Todoroff NK, Eberle C, Thelemann J, Dirdjaja N, Kaiser M, Weber M, Derbani H, Brun R, Schneider G, Pai EF, Krauth-Siegel RL, Diederich F. Persch E, et al. Among authors: kaiser m. ChemMedChem. 2014 Aug;9(8):1880-91. doi: 10.1002/cmdc.201402032. Epub 2014 Apr 30. ChemMedChem. 2014. PMID: 24788386

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

2,133 results

Search Page

Filters