Miah AH - Search Results

1

Lead identification and structure-activity relationships of heteroarylpyrazole arylsulfonamides as allosteric CC-chemokine receptor 4 (CCR4) antagonists.

Miah AH, Copley RC, O'Flynn D, Percy JM, Procopiou PA. Miah AH, et al. Org Biomol Chem. 2014 Mar 21;12(11):1779-92. doi: 10.1039/c3ob42443j. Org Biomol Chem. 2014. PMID: 24515101 Free article.

2

A potentially divergent and rapid route to analogues of deoxycyclitols, pentopyranoses, 6-deoxyhexoses, and hexoses.

Audouard C, Fawcett J, Griffith GA, Kérourédan E, Miah A, Percy JM, Yang H. Audouard C, et al. Org Lett. 2004 Nov 11;6(23):4269-72. doi: 10.1021/ol0482902. Org Lett. 2004. PMID: 15524460

3

Syntheses of difluorinated carbasugar phosphates from trifluoroethanol.

Anderl T, Audouard C, Miah A, Percy JM, Rinaudo G, Singh K. Anderl T, et al. Org Biomol Chem. 2009 Dec 21;7(24):5200-6. doi: 10.1039/b914068a. Epub 2009 Oct 20. Org Biomol Chem. 2009. PMID: 20024116

4

Synthesis and structure-activity relationships of indazole arylsulfonamides as allosteric CC-chemokine receptor 4 (CCR4) antagonists.

Procopiou PA, Barrett JW, Barton NP, Begg M, Clapham D, Copley RC, Ford AJ, Graves RH, Hall DA, Hancock AP, Hill AP, Hobbs H, Hodgson ST, Jumeaux C, Lacroix YM, Miah AH, Morriss KM, Needham D, Sheriff EB, Slack RJ, Smith CE, Sollis SL, Staton H. Procopiou PA, et al. Among authors: miah ah. J Med Chem. 2013 Mar 14;56(5):1946-60. doi: 10.1021/jm301572h. Epub 2013 Feb 27. J Med Chem. 2013. PMID: 23409871

5

Lead identification of benzimidazolone and azabenzimidazolone arylsulfonamides as CC-chemokine receptor 4 (CCR4) antagonists.

Miah AH, Abas H, Begg M, Marsh BJ, O'Flynn DE, Ford AJ, Percy JM, Procopiou PA, Richards SA, Rumley SA. Miah AH, et al. Bioorg Med Chem. 2014 Aug 1;22(15):4298-311. doi: 10.1016/j.bmc.2014.05.021. Epub 2014 May 21. Bioorg Med Chem. 2014. PMID: 24909677 Free article.

6

2,8-Diazaspiro[4.5]decan-8-yl)pyrimidin-4-amine potent CCR4 antagonists capable of inducing receptor endocytosis.

Shukla L, Ajram LA, Begg M, Evans B, Graves RH, Hodgson ST, Lynn SM, Miah AH, Percy JM, Procopiou PA, Richards SA, Slack RJ. Shukla L, et al. Among authors: miah ah. Eur J Med Chem. 2016 Jun 10;115:14-25. doi: 10.1016/j.ejmech.2016.02.058. Epub 2016 Feb 27. Eur J Med Chem. 2016. PMID: 26991939 Free article.

7

Identification of pyrazolopyrimidine arylsulfonamides as CC-chemokine receptor 4 (CCR4) antagonists.

Miah AH, Champigny AC, Graves RH, Hodgson ST, Percy JM, Procopiou PA. Miah AH, et al. Bioorg Med Chem. 2017 Oct 15;25(20):5327-5340. doi: 10.1016/j.bmc.2017.07.052. Epub 2017 Jul 29. Bioorg Med Chem. 2017. PMID: 28801066

8

Structure-based optimisation of orally active & reversible MetAP-2 inhibitors maintaining a tight 'molecular budget'.

Hirst DJ, Brandt M, Bruton G, Christodoulou E, Cutler L, Deeks N, Goodacre JD, Jack T, Lindon M, Miah A, Page K, Parr N, Shukla L, Sims M, Thomas P, Thorpe J, Holmes DS. Hirst DJ, et al. Bioorg Med Chem Lett. 2020 Nov 1;30(21):127533. doi: 10.1016/j.bmcl.2020.127533. Epub 2020 Sep 10. Bioorg Med Chem Lett. 2020. PMID: 32919012

9

Identification of PDE4B Over 4D subtype-selective inhibitors revealing an unprecedented binding mode.

Kranz M, Wall M, Evans B, Miah A, Ballantine S, Delves C, Dombroski B, Gross J, Schneck J, Villa JP, Neu M, Somers DO. Kranz M, et al. Bioorg Med Chem. 2009 Jul 15;17(14):5336-41. doi: 10.1016/j.bmc.2009.03.061. Epub 2009 Apr 5. Bioorg Med Chem. 2009. PMID: 19525117

10

Optimization of a Series of RIPK2 PROTACs.

Miah AH, Smith IED, Rackham M, Mares A, Thawani AR, Nagilla R, Haile PA, Votta BJ, Gordon LJ, Watt G, Denyer J, Fisher DT, Dace P, Giffen P, Goncalves A, Churcher I, Scott-Stevens P, Harling JD. Miah AH, et al. J Med Chem. 2021 Sep 9;64(17):12978-13003. doi: 10.1021/acs.jmedchem.1c01118. Epub 2021 Aug 25. J Med Chem. 2021. PMID: 34432979

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

38 results

Search Page

Filters