Kristensen JL - Search Results

1

Correlating the metabolic stability of psychedelic 5-HT₂A agonists with anecdotal reports of human oral bioavailability.

Leth-Petersen S, Bundgaard C, Hansen M, Carnerup MA, Kehler J, Kristensen JL. Leth-Petersen S, et al. Among authors: kristensen jl. Neurochem Res. 2014 Oct;39(10):2018-23. doi: 10.1007/s11064-014-1253-y. Epub 2014 Feb 12. Neurochem Res. 2014. PMID: 24519542

2

Radiosynthesis and in vivo evaluation of a series of substituted 11C-phenethylamines as 5-HT (2A) agonist PET tracers.

Ettrup A, Hansen M, Santini MA, Paine J, Gillings N, Palner M, Lehel S, Herth MM, Madsen J, Kristensen J, Begtrup M, Knudsen GM. Ettrup A, et al. Eur J Nucl Med Mol Imaging. 2011 Apr;38(4):681-93. doi: 10.1007/s00259-010-1686-8. Epub 2010 Dec 21. Eur J Nucl Med Mol Imaging. 2011. PMID: 21174090

3

Synthesis and biological evaluation of 4-(aminomethyl)-1-hydroxypyrazole analogues of muscimol as γ-aminobutyric acid(a) receptor agonists.

Petersen JG, Bergmann R, Møller HA, Jørgensen CG, Nielsen B, Kehler J, Frydenvang K, Kristensen J, Balle T, Jensen AA, Kristiansen U, Frølund B. Petersen JG, et al. J Med Chem. 2013 Feb 14;56(3):993-1006. doi: 10.1021/jm301473k. Epub 2013 Jan 23. J Med Chem. 2013. PMID: 23294161

4

Preclinical safety assessment of the 5-HT2A receptor agonist PET radioligand [ 11C]Cimbi-36.

Ettrup A, Holm S, Hansen M, Wasim M, Santini MA, Palner M, Madsen J, Svarer C, Kristensen JL, Knudsen GM. Ettrup A, et al. Among authors: kristensen jl. Mol Imaging Biol. 2013 Aug;15(4):376-83. doi: 10.1007/s11307-012-0609-4. Mol Imaging Biol. 2013. PMID: 23306971

5

Structure-activity relationships of constrained phenylethylamine ligands for the serotonin 5-HT2 receptors.

Isberg V, Paine J, Leth-Petersen S, Kristensen JL, Gloriam DE. Isberg V, et al. Among authors: kristensen jl. PLoS One. 2013 Nov 7;8(11):e78515. doi: 10.1371/journal.pone.0078515. eCollection 2013. PLoS One. 2013. PMID: 24244317 Free PMC article.

6

Synthesis and structure-activity relationships of N-benzyl phenethylamines as 5-HT2A/2C agonists.

Hansen M, Phonekeo K, Paine JS, Leth-Petersen S, Begtrup M, Bräuner-Osborne H, Kristensen JL. Hansen M, et al. Among authors: kristensen jl. ACS Chem Neurosci. 2014 Mar 19;5(3):243-9. doi: 10.1021/cn400216u. Epub 2014 Jan 15. ACS Chem Neurosci. 2014. PMID: 24397362 Free PMC article.

7

Serotonin 2A receptor agonist binding in the human brain with [¹¹C]Cimbi-36.

Ettrup A, da Cunha-Bang S, McMahon B, Lehel S, Dyssegaard A, Skibsted AW, Jørgensen LM, Hansen M, Baandrup AO, Bache S, Svarer C, Kristensen JL, Gillings N, Madsen J, Knudsen GM. Ettrup A, et al. Among authors: kristensen jl. J Cereb Blood Flow Metab. 2014 Jul;34(7):1188-96. doi: 10.1038/jcbfm.2014.68. Epub 2014 Apr 30. J Cereb Blood Flow Metab. 2014. PMID: 24780897 Free PMC article. Clinical Trial.

8

Hallucinogen-like effects of 2-([2-(4-cyano-2,5-dimethoxyphenyl) ethylamino]methyl)phenol (25CN-NBOH), a novel N-benzylphenethylamine with 100-fold selectivity for 5-HT₂A receptors, in mice.

Fantegrossi WE, Gray BW, Bailey JM, Smith DA, Hansen M, Kristensen JL. Fantegrossi WE, et al. Among authors: kristensen jl. Psychopharmacology (Berl). 2015 Mar;232(6):1039-47. doi: 10.1007/s00213-014-3739-3. Epub 2014 Sep 17. Psychopharmacology (Berl). 2015. PMID: 25224567 Free PMC article.

9

Synthesis and pharmacological evaluation of N-benzyl substituted 4-bromo-2,5-dimethoxyphenethylamines as 5-HT2A/2C partial agonists.

Hansen M, Jacobsen SE, Plunkett S, Liebscher GE, McCorvy JD, Bräuner-Osborne H, Kristensen JL. Hansen M, et al. Among authors: kristensen jl. Bioorg Med Chem. 2015 Jul 15;23(14):3933-7. doi: 10.1016/j.bmc.2014.12.011. Epub 2014 Dec 17. Bioorg Med Chem. 2015. PMID: 25583099

10

Metabolic Fate of Hallucinogenic NBOMes.

Leth-Petersen S, Gabel-Jensen C, Gillings N, Lehel S, Hansen HD, Knudsen GM, Kristensen JL. Leth-Petersen S, et al. Among authors: kristensen jl. Chem Res Toxicol. 2016 Jan 19;29(1):96-100. doi: 10.1021/acs.chemrestox.5b00450. Epub 2015 Dec 29. Chem Res Toxicol. 2016. PMID: 26669514 Free article.

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