Haufe G - Search Results

1

Fluorescent non-peptidic RGD mimetics with high selectivity for αVβ3 vs αIIbβ3 integrin receptor: novel probes for in vivo optical imaging.

Alsibai W, Hahnenkamp A, Eisenblätter M, Riemann B, Schäfers M, Bremer C, Haufe G, Höltke C. Alsibai W, et al. Among authors: haufe g. J Med Chem. 2014 Dec 11;57(23):9971-82. doi: 10.1021/jm501197c. Epub 2014 Nov 21. J Med Chem. 2014. PMID: 25384028

2

Novel fluorinated derivatives of the broad-spectrum MMP inhibitors N-hydroxy-2(R)-[[(4-methoxyphenyl)sulfonyl](benzyl)- and (3-picolyl)-amino]-3-methyl-butanamide as potential tools for the molecular imaging of activated MMPs with PET.

Wagner S, Breyholz HJ, Law MP, Faust A, Höltke C, Schröer S, Haufe G, Levkau B, Schober O, Schäfers M, Kopka K. Wagner S, et al. Among authors: haufe g. J Med Chem. 2007 Nov 15;50(23):5752-64. doi: 10.1021/jm0708533. Epub 2007 Oct 23. J Med Chem. 2007. PMID: 17956082

3

Fluorinated isatin derivatives. Part 1: synthesis of new N-substituted (S)-5-[1-(2-methoxymethylpyrrolidinyl)sulfonyl]isatins as potent caspase-3 and -7 inhibitors.

Podichetty AK, Faust A, Kopka K, Wagner S, Schober O, Schäfers M, Haufe G. Podichetty AK, et al. Among authors: haufe g. Bioorg Med Chem. 2009 Apr 1;17(7):2680-8. doi: 10.1016/j.bmc.2009.02.048. Epub 2009 Mar 1. Bioorg Med Chem. 2009. PMID: 19299147

4

Fluorinated isatin derivatives. Part 2. New N-substituted 5-pyrrolidinylsulfonyl isatins as potential tools for molecular imaging of caspases in apoptosis.

Podichetty AK, Wagner S, Schröer S, Faust A, Schäfers M, Schober O, Kopka K, Haufe G. Podichetty AK, et al. Among authors: haufe g. J Med Chem. 2009 Jun 11;52(11):3484-95. doi: 10.1021/jm8015014. J Med Chem. 2009. PMID: 19445513

5

Synthesis of geminal difluorides by oxidative desulfurization-difluorination of alkyl aryl thioethers with halonium electrophiles in the presence of fluorinating reagents and its application for 18F-radiolabeling.

Hugenberg V, Wagner S, Kopka K, Schober O, Schäfers M, Haufe G. Hugenberg V, et al. Among authors: haufe g. J Org Chem. 2010 Sep 17;75(18):6086-95. doi: 10.1021/jo100689v. J Org Chem. 2010. PMID: 20738143

6

Fluorinated isatin derivatives. Part 3. New side-chain fluoro-functionalized pyrrolidinyl sulfonyl isatins as potent caspase-3 and -7 inhibitors.

Podichetty AK, Wagner S, Faust A, Schäfers M, Schober O, Kopka K, Haufe G. Podichetty AK, et al. Among authors: haufe g. Future Med Chem. 2009 Aug;1(5):969-89. doi: 10.4155/fmc.09.66. Future Med Chem. 2009. PMID: 21426092

7

A new generation of radiofluorinated pyrimidine-2,4,6-triones as MMP-targeted radiotracers for positron emission tomography.

Schrigten D, Breyholz HJ, Wagner S, Hermann S, Schober O, Schäfers M, Haufe G, Kopka K. Schrigten D, et al. Among authors: haufe g. J Med Chem. 2012 Jan 12;55(1):223-32. doi: 10.1021/jm201142w. Epub 2011 Dec 13. J Med Chem. 2012. PMID: 22118188

8

Synthesis of new fluorinated, 2-substituted 5-pyrrolidinylsulfonyl isatin derivatives as caspase-3 and caspase-7 inhibitors: nonradioactive counterparts of putative PET-compatible apoptosis imaging agents.

Limpachayaporn P, Schäfers M, Schober O, Kopka K, Haufe G. Limpachayaporn P, et al. Among authors: haufe g. Bioorg Med Chem. 2013 Apr 1;21(7):2025-36. doi: 10.1016/j.bmc.2013.01.011. Epub 2013 Jan 16. Bioorg Med Chem. 2013. PMID: 23411396

9

Synthesis, 18F-radiolabeling, and in vivo biodistribution studies of N-fluorohydroxybutyl isatin sulfonamides using positron emission tomography.

Limpachayaporn P, Wagner S, Kopka K, Hermann S, Schäfers M, Haufe G. Limpachayaporn P, et al. Among authors: haufe g. J Med Chem. 2013 Jun 13;56(11):4509-20. doi: 10.1021/jm400257a. Epub 2013 May 29. J Med Chem. 2013. PMID: 23656488

10

Influence of 4- or 5-substituents on the pyrrolidine ring of 5-[1-(2-methoxymethylpyrrolidinyl)sulfonyl]isatin derivatives on their inhibitory activities towards caspases-3 and -7.

Limpachayaporn P, Riemann B, Kopka K, Schober O, Schäfers M, Haufe G. Limpachayaporn P, et al. Among authors: haufe g. Eur J Med Chem. 2013 Jun;64:562-78. doi: 10.1016/j.ejmech.2013.04.011. Epub 2013 Apr 11. Eur J Med Chem. 2013. PMID: 23685941

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