Desmet T - Search Results

1

Synthesis of functionalized 3-, 5-, 6- and 8-aminoquinolines via intermediate (3-pyrrolin-1-yl)- and (2-oxopyrrolidin-1-yl)quinolines and evaluation of their antiplasmodial and antifungal activity.

Vandekerckhove S, Van Herreweghe S, Willems J, Danneels B, Desmet T, de Kock C, Smith PJ, Chibale K, D'hooghe M. Vandekerckhove S, et al. Among authors: desmet t. Eur J Med Chem. 2015 Mar 6;92:91-102. doi: 10.1016/j.ejmech.2014.12.020. Epub 2014 Dec 12. Eur J Med Chem. 2015. PMID: 25544689

2

Chemoenzymatic Syntheses of Fluorine-18-Labeled Disaccharides from [¹⁸F] FDG Yield Potent Sensors of Living Bacteria In Vivo.

Sorlin AM, López-Álvarez M, Rabbitt SJ, Alanizi AA, Shuere R, Bobba KN, Blecha J, Sakhamuri S, Evans MJ, Bayles KW, Flavell RR, Rosenberg OS, Sriram R, Desmet T, Nidetzky B, Engel J, Ohliger MA, Fraser JS, Wilson DM. Sorlin AM, et al. Among authors: desmet t. J Am Chem Soc. 2023 Aug 16;145(32):17632-17642. doi: 10.1021/jacs.3c03338. Epub 2023 Aug 3. J Am Chem Soc. 2023. PMID: 37535945 Free PMC article.

3

Biocatalytic production of novel glycolipids with cellodextrin phosphorylase.

Tran HG, Desmet T, Saerens K, Waegeman H, Vandekerckhove S, D'hooghe M, Van Bogaert I, Soetaert W. Tran HG, et al. Among authors: desmet t. Bioresour Technol. 2012 Jul;115:84-7. doi: 10.1016/j.biortech.2011.09.085. Epub 2011 Sep 25. Bioresour Technol. 2012. PMID: 22000964

4

Synthesis of 2-aminomethyl-4-phenyl-1-azabicyclo[2.2.1]heptanes via LiAlH₄-induced reductive cyclization of 2-(4-chloro-2-cyano-2-phenylbutyl)aziridines and evaluation of their antimalarial activity.

D'hooghe M, Vervisch K, Törnroos KW, Verhaeghe T, Desmet T, Lategan C, Smith PJ, Chibale K, De Kimpe N. D'hooghe M, et al. Among authors: desmet t. Bioorg Med Chem Lett. 2013 Mar 1;23(5):1507-10. doi: 10.1016/j.bmcl.2012.12.029. Epub 2012 Dec 20. Bioorg Med Chem Lett. 2013. PMID: 23347684

5

Potent and selective HDAC6 inhibitory activity of N-(4-hydroxycarbamoylbenzyl)-1,2,4,9-tetrahydro-3-thia-9-azafluorenes as novel sulfur analogues of Tubastatin A.

De Vreese R, Verhaeghe T, Desmet T, D'hooghe M. De Vreese R, et al. Among authors: desmet t. Chem Commun (Camb). 2013 May 8;49(36):3775-7. doi: 10.1039/c3cc41422a. Epub 2013 Mar 28. Chem Commun (Camb). 2013. PMID: 23538448

6

Evaluation of (4-aminobutyloxy)quinolines as a novel class of antifungal agents.

Vandekerckhove S, Tran HG, Desmet T, D'hooghe M. Vandekerckhove S, et al. Among authors: desmet t. Bioorg Med Chem Lett. 2013 Aug 15;23(16):4641-3. doi: 10.1016/j.bmcl.2013.06.014. Epub 2013 Jun 13. Bioorg Med Chem Lett. 2013. PMID: 23838261

7

Synthesis of halogenated 4-quinolones and evaluation of their antiplasmodial activity.

Vandekerckhove S, Desmet T, Tran HG, de Kock C, Smith PJ, Chibale K, D'hooghe M. Vandekerckhove S, et al. Among authors: desmet t. Bioorg Med Chem Lett. 2014 Feb 15;24(4):1214-7. doi: 10.1016/j.bmcl.2013.12.067. Epub 2014 Jan 4. Bioorg Med Chem Lett. 2014. PMID: 24468411

8

Engineering the specificity of trehalose phosphorylase as a general strategy for the production of glycosyl phosphates.

Chen C, Van der Borght J, De Vreese R, D'hooghe M, Soetaert W, Desmet T. Chen C, et al. Among authors: desmet t. Chem Commun (Camb). 2014 Jul 25;50(58):7834-6. doi: 10.1039/c4cc02202e. Chem Commun (Camb). 2014. PMID: 24909572

9

Synthesis of 2-aryl-3-(2-cyanoethyl)aziridines and their chemical and enzymatic hydrolysis towards γ-lactams and γ-lactones.

Mollet K, Decuyper L, Vander Meeren S, Piens N, De Winter K, Desmet T, D'hooghe M. Mollet K, et al. Among authors: desmet t. Org Biomol Chem. 2015 Mar 7;13(9):2716-25. doi: 10.1039/c4ob02615b. Org Biomol Chem. 2015. PMID: 25598487

10

Synthesis of benzothiophene-based hydroxamic acids as potent and selective HDAC6 inhibitors.

De Vreese R, Van Steen N, Verhaeghe T, Desmet T, Bougarne N, De Bosscher K, Benoy V, Haeck W, Van Den Bosch L, D'hooghe M. De Vreese R, et al. Among authors: desmet t. Chem Commun (Camb). 2015 Jun 18;51(48):9868-71. doi: 10.1039/c5cc03295d. Chem Commun (Camb). 2015. PMID: 25994553

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