Misawa T - Search Results

1

Structural development of stapled short helical peptides as vitamin D receptor (VDR)-coactivator interaction inhibitors.

Misawa T, Demizu Y, Kawamura M, Yamagata N, Kurihara M. Misawa T, et al. Bioorg Med Chem. 2015 Mar 1;23(5):1055-61. doi: 10.1016/j.bmc.2015.01.007. Epub 2015 Jan 12. Bioorg Med Chem. 2015. PMID: 25637122

2

Discovery and structural development of small molecules that enhance transport activity of bile salt export pump mutant associated with progressive familial intrahepatic cholestasis type 2.

Misawa T, Hayashi H, Sugiyama Y, Hashimoto Y. Misawa T, et al. Bioorg Med Chem. 2012 May 1;20(9):2940-9. doi: 10.1016/j.bmc.2012.03.016. Epub 2012 Mar 14. Bioorg Med Chem. 2012. PMID: 22464344

3

E297G mutated bile salt export pump (BSEP) function enhancers derived from GW4064: structural development study and separation from farnesoid X receptor-agonistic activity.

Misawa T, Hayashi H, Makishima M, Sugiyama Y, Hashimoto Y. Misawa T, et al. Bioorg Med Chem Lett. 2012 Jun 15;22(12):3962-6. doi: 10.1016/j.bmcl.2012.04.099. Epub 2012 Apr 30. Bioorg Med Chem Lett. 2012. PMID: 22583617

4

Structure-activity relationship-guided development of retinoic acid receptor-related orphan receptor gamma (RORγ)-selective inverse agonists with a phenanthridin-6(5H)-one skeleton from a liver X receptor ligand.

Nishiyama Y, Nakamura M, Misawa T, Nakagomi M, Makishima M, Ishikawa M, Hashimoto Y. Nishiyama Y, et al. Among authors: misawa t. Bioorg Med Chem. 2014 May 1;22(9):2799-808. doi: 10.1016/j.bmc.2014.03.007. Epub 2014 Mar 17. Bioorg Med Chem. 2014. PMID: 24702856

5

Development of cell-penetrating R7 fragment-conjugated helical peptides as inhibitors of estrogen receptor-mediated transcription.

Nagakubo T, Demizu Y, Kanda Y, Misawa T, Shoda T, Okuhira K, Sekino Y, Naito M, Kurihara M. Nagakubo T, et al. Among authors: misawa t. Bioconjug Chem. 2014 Nov 19;25(11):1921-4. doi: 10.1021/bc500480e. Epub 2014 Nov 7. Bioconjug Chem. 2014. PMID: 25375254

6

Effects of D-Leu residues on the helical secondary structures of L-Leu-based nonapeptides.

Demizu Y, Yamashita H, Misawa T, Doi M, Tanaka M, Kurihara M. Demizu Y, et al. Among authors: misawa t. Chem Pharm Bull (Tokyo). 2015;63(3):218-24. doi: 10.1248/cpb.c14-00760. Chem Pharm Bull (Tokyo). 2015. PMID: 25757493 Free article.

7

Structure-activity relationships of benzhydrol derivatives based on 1'-acetoxychavicol acetate (ACA) and their inhibitory activities on multiple myeloma cell growth via inactivation of the NF-κB pathway.

Misawa T, Dodo K, Ishikawa M, Hashimoto Y, Sagawa M, Kizaki M, Aoyama H. Misawa T, et al. Bioorg Med Chem. 2015 May 1;23(9):2241-6. doi: 10.1016/j.bmc.2015.02.039. Epub 2015 Mar 7. Bioorg Med Chem. 2015. PMID: 25801158

8

A preorganized β-amino acid bearing a guanidinium side chain and its use in cell-penetrating peptides.

Demizu Y, Oba M, Okitsu K, Yamashita H, Misawa T, Tanaka M, Kurihara M, Gellman SH. Demizu Y, et al. Among authors: misawa t. Org Biomol Chem. 2015 May 28;13(20):5617-20. doi: 10.1039/c5ob00389j. Epub 2015 Apr 21. Org Biomol Chem. 2015. PMID: 25897867

9

Design, synthesis, and anti-HIV-1 activity of 1-aromatic methyl-substituted 3-(3,5-dimethylbenzyl)uracil and N-3,5-dimethylbenzyl-substituted urea derivatives.

Sakakibara N, Baba M, Okamoto M, Toyama M, Demizu Y, Misawa T, Kurihara M, Irie K, Kato Y, Maruyama T. Sakakibara N, et al. Among authors: misawa t. Antivir Chem Chemother. 2015 Feb;24(1):3-18. doi: 10.1177/2040206614566584. Antivir Chem Chemother. 2015. PMID: 26149262 Free PMC article.

10

Structural development of stabilized helical peptides as inhibitors of estrogen receptor (ER)-mediated transcription.

Demizu Y, Misawa T, Nagakubo T, Kanda Y, Okuhira K, Sekino Y, Naito M, Kurihara M. Demizu Y, et al. Among authors: misawa t. Bioorg Med Chem. 2015 Aug 1;23(15):4132-4138. doi: 10.1016/j.bmc.2015.06.067. Epub 2015 Jul 2. Bioorg Med Chem. 2015. PMID: 26183544

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