Franchetti P - Search Results

1

5'-C-Ethyl-tetrazolyl-N(6)-substituted adenosine and 2-chloro-adenosine derivatives as highly potent dual acting A1 adenosine receptor agonists and A3 adenosine receptor antagonists.

Petrelli R, Torquati I, Kachler S, Luongo L, Maione S, Franchetti P, Grifantini M, Novellino E, Lavecchia A, Klotz KN, Cappellacci L. Petrelli R, et al. Among authors: franchetti p. J Med Chem. 2015 Mar 12;58(5):2560-6. doi: 10.1021/acs.jmedchem.5b00074. Epub 2015 Feb 27. J Med Chem. 2015. PMID: 25699637

2

Ribose-modified nucleosides as ligands for adenosine receptors: synthesis, conformational analysis, and biological evaluation of 1'-C-methyl adenosine analogues.

Cappellacci L, Barboni G, Palmieri M, Pasqualini M, Grifantini M, Costa B, Martini C, Franchetti P. Cappellacci L, et al. Among authors: franchetti p. J Med Chem. 2002 Mar 14;45(6):1196-202. doi: 10.1021/jm0102755. J Med Chem. 2002. PMID: 11881988

3

Synthesis, biological evaluation, and molecular modeling of ribose-modified adenosine analogues as adenosine receptor agonists.

Cappellacci L, Franchetti P, Pasqualini M, Petrelli R, Vita P, Lavecchia A, Novellino E, Costa B, Martini C, Klotz KN, Grifantini M. Cappellacci L, et al. Among authors: franchetti p. J Med Chem. 2005 Mar 10;48(5):1550-62. doi: 10.1021/jm049408n. J Med Chem. 2005. PMID: 15743197

4

Antitumor activity of C-methyl-beta-D-ribofuranosyladenine nucleoside ribonucleotide reductase inhibitors.

Franchetti P, Cappellacci L, Pasqualini M, Petrelli R, Vita P, Jayaram HN, Horvath Z, Szekeres T, Grifantini M. Franchetti P, et al. J Med Chem. 2005 Jul 28;48(15):4983-9. doi: 10.1021/jm048944c. J Med Chem. 2005. PMID: 16033277

5

5'-Carbamoyl derivatives of 2'-C-methyl-purine nucleosides as selective A1 adenosine receptor agonists: affinity, efficacy, and selectivity for A1 receptor from different species.

Cappellacci L, Franchetti P, Vita P, Petrelli R, Lavecchia A, Costa B, Spinetti F, Martini C, Klotz KN, Grifantini M. Cappellacci L, et al. Among authors: franchetti p. Bioorg Med Chem. 2008 Jan 1;16(1):336-53. doi: 10.1016/j.bmc.2007.09.035. Epub 2007 Sep 22. Bioorg Med Chem. 2008. PMID: 17933541

6

Ribose-modified purine nucleosides as ribonucleotide reductase inhibitors. Synthesis, antitumor activity, and molecular modeling of N6-substituted 3'-C-methyladenosine derivatives.

Cappellacci L, Franchetti P, Vita P, Petrelli R, Lavecchia A, Jayaram HN, Saiko P, Graser G, Szekeres T, Grifantini M. Cappellacci L, et al. Among authors: franchetti p. J Med Chem. 2008 Jul 24;51(14):4260-9. doi: 10.1021/jm800205c. Epub 2008 Jun 28. J Med Chem. 2008. PMID: 18588281

7

N6-Cycloalkyl- and N6-bicycloalkyl-C5'(C2')-modified adenosine derivatives as high-affinity and selective agonists at the human A1 adenosine receptor with antinociceptive effects in mice.

Franchetti P, Cappellacci L, Vita P, Petrelli R, Lavecchia A, Kachler S, Klotz KN, Marabese I, Luongo L, Maione S, Grifantini M. Franchetti P, et al. J Med Chem. 2009 Apr 23;52(8):2393-406. doi: 10.1021/jm801456g. J Med Chem. 2009. PMID: 19317449

8

Synthesis and biological activity of novel N6-substituted and 2,N6-disubstituted adenine ribo- and 3'-C-methyl-ribonucleosides as antitumor agents.

Cappellacci L, Petrelli R, Franchetti P, Vita P, Kusumanchi P, Kumar M, Jayaram HN, Zhou B, Yen Y, Grifantini M. Cappellacci L, et al. Among authors: franchetti p. Eur J Med Chem. 2011 May;46(5):1499-504. doi: 10.1016/j.ejmech.2011.01.055. Epub 2011 Feb 3. Eur J Med Chem. 2011. PMID: 21349610

9

From the covalent linkage of drugs to novel inhibitors of ribonucleotide reductase: synthesis and biological evaluation of valproic esters of 3'-C-methyladenosine.

Petrelli R, Meli M, Vita P, Torquati I, Ferro A, Vodnala M, D'Alessandro N, Tolomeo M, Del Bello F, Kusumanchi P, Franchetti P, Grifantini M, Jayaram HN, Hofer A, Cappellacci L. Petrelli R, et al. Among authors: franchetti p. Bioorg Med Chem Lett. 2014 Nov 15;24(22):5304-9. doi: 10.1016/j.bmcl.2014.09.046. Epub 2014 Sep 28. Bioorg Med Chem Lett. 2014. PMID: 25304896

10

Adenosine receptor agonists: synthesis and biological evaluation of 1-deaza analogues of adenosine derivatives.

Cristalli G, Franchetti P, Grifantini M, Vittori S, Klotz KN, Lohse MJ. Cristalli G, et al. Among authors: franchetti p. J Med Chem. 1988 Jun;31(6):1179-83. doi: 10.1021/jm00401a018. J Med Chem. 1988. PMID: 3373486

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