Rennie PS - Search Results

1

In silico discovery and validation of potent small-molecule inhibitors targeting the activation function 2 site of human oestrogen receptor α.

Singh K, Munuganti RS, Leblanc E, Lin YL, Leung E, Lallous N, Butler M, Cherkasov A, Rennie PS. Singh K, et al. Among authors: rennie ps. Breast Cancer Res. 2015 Feb 25;17(1):27. doi: 10.1186/s13058-015-0529-8. Breast Cancer Res. 2015. PMID: 25848700 Free PMC article.

2

Targeting the binding function 3 (BF3) site of the human androgen receptor through virtual screening.

Lack NA, Axerio-Cilies P, Tavassoli P, Han FQ, Chan KH, Feau C, LeBlanc E, Guns ET, Guy RK, Rennie PS, Cherkasov A. Lack NA, et al. Among authors: rennie ps. J Med Chem. 2011 Dec 22;54(24):8563-73. doi: 10.1021/jm201098n. Epub 2011 Nov 18. J Med Chem. 2011. PMID: 22047606 Free PMC article.

3

Discovery of 1H-indole-2-carboxamides as novel inhibitors of the androgen receptor binding function 3 (BF3).

Ban F, Leblanc E, Li H, Munuganti RS, Frewin K, Rennie PS, Cherkasov A. Ban F, et al. Among authors: rennie ps. J Med Chem. 2014 Aug 14;57(15):6867-72. doi: 10.1021/jm500684r. Epub 2014 Jul 25. J Med Chem. 2014. PMID: 25025737

4

Discovery of small-molecule inhibitors selectively targeting the DNA-binding domain of the human androgen receptor.

Li H, Ban F, Dalal K, Leblanc E, Frewin K, Ma D, Adomat H, Rennie PS, Cherkasov A. Li H, et al. Among authors: rennie ps. J Med Chem. 2014 Aug 14;57(15):6458-67. doi: 10.1021/jm500802j. Epub 2014 Aug 4. J Med Chem. 2014. PMID: 25062331

5

Drug-Discovery Pipeline for Novel Inhibitors of the Androgen Receptor.

Dalal K, Munuganti R, Morin H, Lallous N, Rennie PS, Cherkasov A. Dalal K, et al. Among authors: rennie ps. Methods Mol Biol. 2016;1443:31-54. doi: 10.1007/978-1-4939-3724-0_4. Methods Mol Biol. 2016. PMID: 27246333

6

Targeting Binding Function-3 of the Androgen Receptor Blocks Its Co-Chaperone Interactions, Nuclear Translocation, and Activation.

Lallous N, Leblanc E, Munuganti RS, Hassona MD, Nakouzi NA, Awrey S, Morin H, Roshan-Moniri M, Singh K, Lawn S, Yamazaki T, Adomat HH, Andre C, Daugaard M, Young RN, Guns ES, Rennie PS, Cherkasov A. Lallous N, et al. Among authors: rennie ps. Mol Cancer Ther. 2016 Dec;15(12):2936-2945. doi: 10.1158/1535-7163.MCT-16-0354. Epub 2016 Oct 7. Mol Cancer Ther. 2016. PMID: 27765852 Free PMC article.

7

Computer-Aided Discovery of Small Molecule Inhibitors of Transcriptional Activity of TLX (NR2E1) Nuclear Receptor.

Dueva E, Singh K, Kalyta A, LeBlanc E, Rennie PS, Cherkasov A. Dueva E, et al. Among authors: rennie ps. Molecules. 2018 Nov 14;23(11):2967. doi: 10.3390/molecules23112967. Molecules. 2018. PMID: 30441799 Free PMC article.

8

Computer-Aided Ligand Discovery for Estrogen Receptor Alpha.

Bafna D, Ban F, Rennie PS, Singh K, Cherkasov A. Bafna D, et al. Among authors: rennie ps. Int J Mol Sci. 2020 Jun 12;21(12):4193. doi: 10.3390/ijms21124193. Int J Mol Sci. 2020. PMID: 32545494 Free PMC article. Review.

9

Development of Novel Inhibitors Targeting the D-Box of the DNA Binding Domain of Androgen Receptor.

Radaeva M, Ban F, Zhang F, LeBlanc E, Lallous N, Rennie PS, Gleave ME, Cherkasov A. Radaeva M, et al. Among authors: rennie ps. Int J Mol Sci. 2021 Mar 2;22(5):2493. doi: 10.3390/ijms22052493. Int J Mol Sci. 2021. PMID: 33801338 Free PMC article.

10

Inhibitors of androgen receptor activation function-2 (AF2) site identified through virtual screening.

Axerio-Cilies P, Lack NA, Nayana MR, Chan KH, Yeung A, Leblanc E, Guns ES, Rennie PS, Cherkasov A. Axerio-Cilies P, et al. Among authors: rennie ps. J Med Chem. 2011 Sep 22;54(18):6197-205. doi: 10.1021/jm200532b. Epub 2011 Aug 29. J Med Chem. 2011. PMID: 21846139

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