Spetea M - Search Results

1

Anti-inflammatory effect of dual nociceptin and opioid receptor agonist, BU08070, in experimental colitis in mice.

Zielińska M, Ben Haddou T, Cami-Kobeci G, Sałaga M, Jarmuż A, Padysz M, Kordek R, Spetea M, Husbands SM, Fichna J. Zielińska M, et al. Among authors: spetea m. Eur J Pharmacol. 2015 Oct 15;765:582-90. doi: 10.1016/j.ejphar.2015.09.021. Epub 2015 Sep 25. Eur J Pharmacol. 2015. PMID: 26404500 Free PMC article.

2

In vitro opioid activity profiles of 6-amino acid substituted derivatives of 14-O-methyloxymorphone.

Spetea M, Friedmann T, Riba P, Schütz J, Wunder G, Langer T, Schmidhammer H, Fürst S. Spetea M, et al. Eur J Pharmacol. 2004 Jan 12;483(2-3):301-8. doi: 10.1016/j.ejphar.2003.10.049. Eur J Pharmacol. 2004. PMID: 14729121

3

Local peripheral antinociceptive effects of 14-O-methyloxymorphone derivatives in inflammatory and neuropathic pain in the rat.

Obara I, Makuch W, Spetea M, Schütz J, Schmidhammer H, Przewlocki R, Przewlocka B. Obara I, et al. Among authors: spetea m. Eur J Pharmacol. 2007 Mar 8;558(1-3):60-7. doi: 10.1016/j.ejphar.2006.11.037. Epub 2006 Nov 25. Eur J Pharmacol. 2007. PMID: 17204264

4

Discovery and pharmacological evaluation of a diphenethylamine derivative (HS665), a highly potent and selective κ opioid receptor agonist.

Spetea M, Berzetei-Gurske IP, Guerrieri E, Schmidhammer H. Spetea M, et al. J Med Chem. 2012 Nov 26;55(22):10302-6. doi: 10.1021/jm301258w. Epub 2012 Nov 7. J Med Chem. 2012. PMID: 23134120

5

Pharmacological investigations of N-substituent variation in morphine and oxymorphone: opioid receptor binding, signaling and antinociceptive activity.

Ben Haddou T, Béni S, Hosztafi S, Malfacini D, Calo G, Schmidhammer H, Spetea M. Ben Haddou T, et al. Among authors: spetea m. PLoS One. 2014 Jun 11;9(6):e99231. doi: 10.1371/journal.pone.0099231. eCollection 2014. PLoS One. 2014. PMID: 24919067 Free PMC article.

6

Exploring pharmacological activities and signaling of morphinans substituted in position 6 as potent agonists interacting with the μ opioid receptor.

Ben Haddou T, Malfacini D, Calo G, Aceto MD, Harris LS, Traynor JR, Coop A, Schmidhammer H, Spetea M. Ben Haddou T, et al. Among authors: spetea m. Mol Pain. 2014 Jul 24;10:48. doi: 10.1186/1744-8069-10-48. Mol Pain. 2014. PMID: 25059282 Free PMC article.

7

Bifunctional peptide-based opioid agonist/nociceptin antagonist ligand for dual treatment of nociceptive and neuropathic pain.

Lagard C, Chevillard L, Guillemyn K, Risède P, Laplanche JL, Spetea M, Ballet S, Mégarbane B. Lagard C, et al. Among authors: spetea m. Pain. 2017 Mar;158(3):505-515. doi: 10.1097/j.pain.0000000000000790. Pain. 2017. PMID: 28135212 Free PMC article.

8

Selective κ receptor partial agonist HS666 produces potent antinociception without inducing aversion after i.c.v. administration in mice.

Spetea M, Eans SO, Ganno ML, Lantero A, Mairegger M, Toll L, Schmidhammer H, McLaughlin JP. Spetea M, et al. Br J Pharmacol. 2017 Aug;174(15):2444-2456. doi: 10.1111/bph.13854. Epub 2017 Jun 27. Br J Pharmacol. 2017. PMID: 28494108 Free PMC article.

9

Highly Potent and Selective New Diphenethylamines Interacting with the κ-Opioid Receptor: Synthesis, Pharmacology, and Structure-Activity Relationships.

Erli F, Guerrieri E, Ben Haddou T, Lantero A, Mairegger M, Schmidhammer H, Spetea M. Erli F, et al. Among authors: spetea m. J Med Chem. 2017 Sep 14;60(17):7579-7590. doi: 10.1021/acs.jmedchem.7b00981. Epub 2017 Aug 30. J Med Chem. 2017. PMID: 28825813 Free PMC article.

10

Synthesis, Pharmacology, and Molecular Docking Studies on 6-Desoxo-N-methylmorphinans as Potent μ-Opioid Receptor Agonists.

Dumitrascuta M, Ben Haddou T, Guerrieri E, Noha SM, Schläfer L, Schmidhammer H, Spetea M. Dumitrascuta M, et al. Among authors: spetea m. J Med Chem. 2017 Nov 22;60(22):9407-9412. doi: 10.1021/acs.jmedchem.7b01363. Epub 2017 Nov 3. J Med Chem. 2017. PMID: 29053268 Free PMC article.

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