Hong KH - Search Results

1

Characterizing the Epothilone Binding Site on β-Tubulin by Photoaffinity Labeling: Identification of β-Tubulin Peptides TARGSQQY and TSRGSQQY as Targets of an Epothilone Photoprobe for Polymerized Tubulin.

Ranade AR, Higgins L, Markowski TW, Glaser N, Kashin D, Bai R, Hong KH, Hamel E, Höfle G, Georg GI. Ranade AR, et al. Among authors: hong kh. J Med Chem. 2016 Apr 14;59(7):3499-514. doi: 10.1021/acs.jmedchem.6b00188. Epub 2016 Mar 17. J Med Chem. 2016. PMID: 26986898 Free PMC article.

2

Synthesis and evaluation of the anti-proliferative and NF-κB activities of a library of simplified tylophorine analogs.

Niphakis MJ, Gay BC, Hong KH, Bleeker NP, Georg GI. Niphakis MJ, et al. Among authors: hong kh. Bioorg Med Chem. 2012 Oct 1;20(19):5893-900. doi: 10.1016/j.bmc.2012.07.044. Epub 2012 Aug 3. Bioorg Med Chem. 2012. PMID: 22910225

3

Discovery of 4-aminoquinazoline--urea derivatives as Aurora kinase inhibitors with antiproliferative activity.

Cai J, Li L, Hong KH, Wu X, Chen J, Wang P, Cao M, Zong X, Ji M. Cai J, et al. Among authors: hong kh. Bioorg Med Chem. 2014 Nov 1;22(21):5813-23. doi: 10.1016/j.bmc.2014.09.029. Epub 2014 Sep 19. Bioorg Med Chem. 2014. PMID: 25270403

4

Synthesis and biological evaluation of novel indole-pyrimidine hybrids bearing morpholine and thiomorpholine moieties.

Diao PC, Li Q, Hu MJ, Ma YF, You WW, Hong KH, Zhao PL. Diao PC, et al. Among authors: hong kh. Eur J Med Chem. 2017 Jul 7;134:110-118. doi: 10.1016/j.ejmech.2017.04.011. Epub 2017 Apr 7. Eur J Med Chem. 2017. PMID: 28410492

5

Structural Basis of ALDH1A2 Inhibition by Irreversible and Reversible Small Molecule Inhibitors.

Chen Y, Zhu JY, Hong KH, Mikles DC, Georg GI, Goldstein AS, Amory JK, Schönbrunn E. Chen Y, et al. Among authors: hong kh. ACS Chem Biol. 2018 Mar 16;13(3):582-590. doi: 10.1021/acschembio.7b00685. Epub 2018 Jan 3. ACS Chem Biol. 2018. PMID: 29240402 Free PMC article.

6

Design, Synthesis, and in Vitro and in Vivo Evaluation of Ouabain Analogues as Potent and Selective Na,K-ATPase α4 Isoform Inhibitors for Male Contraception.

Syeda SS, Sánchez G, Hong KH, Hawkinson JE, Georg GI, Blanco G. Syeda SS, et al. Among authors: hong kh. J Med Chem. 2018 Mar 8;61(5):1800-1820. doi: 10.1021/acs.jmedchem.7b00925. Epub 2018 Jan 19. J Med Chem. 2018. PMID: 29291372 Free PMC article.

7

Discovery and optimization of 3,4,5-trimethoxyphenyl substituted triazolylthioacetamides as potent tubulin polymerization inhibitors.

Yang F, He CP, Diao PC, Hong KH, Rao JJ, Zhao PL. Yang F, et al. Among authors: hong kh. Bioorg Med Chem Lett. 2019 Jan 1;29(1):22-27. doi: 10.1016/j.bmcl.2018.11.024. Epub 2018 Nov 13. Bioorg Med Chem Lett. 2019. PMID: 30448234

8

The Na+ and K+ transport system of sperm (ATP1A4) is essential for male fertility and an attractive target for male contraception†.

Syeda SS, Sánchez G, McDermott JP, Hong KH, Blanco G, Georg GI. Syeda SS, et al. Among authors: hong kh. Biol Reprod. 2020 Aug 4;103(2):343-356. doi: 10.1093/biolre/ioaa093. Biol Reprod. 2020. PMID: 32588885 Free PMC article. Review.

9

Tetrahydroindazole inhibitors of CDK2/cyclin complexes.

Lee JC, Hong KH, Becker A, Tash JS, Schönbrunn E, Georg GI. Lee JC, et al. Among authors: hong kh. Eur J Med Chem. 2021 Mar 15;214:113232. doi: 10.1016/j.ejmech.2021.113232. Epub 2021 Jan 31. Eur J Med Chem. 2021. PMID: 33550184 Free PMC article.

10

Screening through Lead Optimization of High Affinity, Allosteric Cyclin-Dependent Kinase 2 (CDK2) Inhibitors as Male Contraceptives That Reduce Sperm Counts in Mice.

Faber EB, Wang N, John K, Sun L, Wong HL, Burban D, Francis R, Tian D, Hong KH, Yang A, Wang L, Elsaid M, Khalid H, Levinson NM, Schönbrunn E, Hawkinson JE, Georg GI. Faber EB, et al. Among authors: hong kh. J Med Chem. 2023 Feb 9;66(3):1928-1940. doi: 10.1021/acs.jmedchem.2c01731. Epub 2023 Jan 26. J Med Chem. 2023. PMID: 36701569 Free PMC article.

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