Cerchia C - Search Results

1

The antiproliferative and proapoptotic effects of cladosporols A and B are related to their different binding mode as PPARγ ligands.

Zurlo D, Ziccardi P, Votino C, Colangelo T, Cerchia C, Dal Piaz F, Dallavalle S, Moricca S, Novellino E, Lavecchia A, Colantuoni V, Lupo A. Zurlo D, et al. Among authors: cerchia c. Biochem Pharmacol. 2016 May 15;108:22-35. doi: 10.1016/j.bcp.2016.03.007. Epub 2016 Mar 17. Biochem Pharmacol. 2016. PMID: 26995279

2

Discovery of a novel small molecule inhibitor targeting the frataxin/ubiquitin interaction via structure-based virtual screening and bioassays.

Lavecchia A, Di Giovanni C, Cerchia C, Russo A, Russo G, Novellino E. Lavecchia A, et al. Among authors: cerchia c. J Med Chem. 2013 Apr 11;56(7):2861-73. doi: 10.1021/jm3017199. Epub 2013 Mar 29. J Med Chem. 2013. PMID: 23506486

3

Novel inhibitors of signal transducer and activator of transcription 3 signaling pathway: an update on the recent patent literature.

Lavecchia A, Di Giovanni C, Cerchia C. Lavecchia A, et al. Among authors: cerchia c. Expert Opin Ther Pat. 2014 Apr;24(4):383-400. doi: 10.1517/13543776.2014.877443. Epub 2014 Jan 16. Expert Opin Ther Pat. 2014. PMID: 24432979 Review.

4

Identification of a new series of amides as non-covalent proteasome inhibitors.

Scarbaci K, Troiano V, Micale N, Ettari R, Tamborini L, Di Giovanni C, Cerchia C, Grasso S, Novellino E, Schirmeister T, Lavecchia A, Zappalà M. Scarbaci K, et al. Among authors: cerchia c. Eur J Med Chem. 2014 Apr 9;76:1-9. doi: 10.1016/j.ejmech.2014.01.022. Epub 2014 Jan 25. Eur J Med Chem. 2014. PMID: 24561716

5

Development of novel selective peptidomimetics containing a boronic acid moiety, targeting the 20S proteasome as anticancer agents.

Scarbaci K, Troiano V, Ettari R, Pinto A, Micale N, Di Giovanni C, Cerchia C, Schirmeister T, Novellino E, Lavecchia A, Zappalà M, Grasso S. Scarbaci K, et al. Among authors: cerchia c. ChemMedChem. 2014 Aug;9(8):1801-16. doi: 10.1002/cmdc.201402075. Epub 2014 May 28. ChemMedChem. 2014. PMID: 24891205

6

Optimization of peptidomimetic boronates bearing a P3 bicyclic scaffold as proteasome inhibitors.

Troiano V, Scarbaci K, Ettari R, Micale N, Cerchia C, Pinto A, Schirmeister T, Novellino E, Grasso S, Lavecchia A, Zappalà M. Troiano V, et al. Among authors: cerchia c. Eur J Med Chem. 2014 Aug 18;83:1-14. doi: 10.1016/j.ejmech.2014.06.017. Epub 2014 Jun 10. Eur J Med Chem. 2014. PMID: 24946214

7

Ligand-based chemoinformatic discovery of a novel small molecule inhibitor targeting CDC25 dual specificity phosphatases and displaying in vitro efficacy against melanoma cells.

Capasso A, Cerchia C, Di Giovanni C, Granato G, Albano F, Romano S, De Vendittis E, Ruocco MR, Lavecchia A. Capasso A, et al. Among authors: cerchia c. Oncotarget. 2015 Nov 24;6(37):40202-22. doi: 10.18632/oncotarget.5473. Oncotarget. 2015. PMID: 26474275 Free PMC article.

8

In silico methods to address polypharmacology: current status, applications and future perspectives.

Lavecchia A, Cerchia C. Lavecchia A, et al. Among authors: cerchia c. Drug Discov Today. 2016 Feb;21(2):288-98. doi: 10.1016/j.drudis.2015.12.007. Epub 2015 Dec 29. Drug Discov Today. 2016. PMID: 26743596 Review.

9

Novel non-peptide small molecules preventing IKKβ/NEMO association inhibit NF-κB activation in LPS-stimulated J774 macrophages.

De Falco F, Di Giovanni C, Cerchia C, De Stefano D, Capuozzo A, Irace C, Iuvone T, Santamaria R, Carnuccio R, Lavecchia A. De Falco F, et al. Among authors: cerchia c. Biochem Pharmacol. 2016 Mar 15;104:83-94. doi: 10.1016/j.bcp.2016.01.008. Epub 2016 Jan 14. Biochem Pharmacol. 2016. PMID: 26776306

10

Structural basis for PPAR partial or full activation revealed by a novel ligand binding mode.

Capelli D, Cerchia C, Montanari R, Loiodice F, Tortorella P, Laghezza A, Cervoni L, Pochetti G, Lavecchia A. Capelli D, et al. Among authors: cerchia c. Sci Rep. 2016 Oct 6;6:34792. doi: 10.1038/srep34792. Sci Rep. 2016. PMID: 27708429 Free PMC article.

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