Bazgier V - Search Results

1

Novel N-substituted indole Schiff bases as dual inhibitors of cyclooxygenase-2 and 5-lipoxygenase enzymes: Synthesis, biological activities in vitro and docking study.

Lamie PF, Ali WAM, Bazgier V, Rárová L. Lamie PF, et al. Among authors: bazgier v. Eur J Med Chem. 2016 Nov 10;123:803-813. doi: 10.1016/j.ejmech.2016.08.013. Epub 2016 Aug 10. Eur J Med Chem. 2016. PMID: 27541263

2

A novel series of highly potent 2,6,9-trisubstituted purine cyclin-dependent kinase inhibitors.

Gucký T, Jorda R, Zatloukal M, Bazgier V, Berka K, Řezníčková E, Béres T, Strnad M, Kryštof V. Gucký T, et al. Among authors: bazgier v. J Med Chem. 2013 Aug 8;56(15):6234-47. doi: 10.1021/jm4006884. Epub 2013 Jul 24. J Med Chem. 2013. PMID: 23829517

3

Synthesis and kinase inhibitory activity of new sulfonamide derivatives of pyrazolo[4,3-e][1,2,4]triazines.

Mojzych M, Šubertová V, Bielawska A, Bielawski K, Bazgier V, Berka K, Gucký T, Fornal E, Kryštof V. Mojzych M, et al. Among authors: bazgier v. Eur J Med Chem. 2014 May 6;78:217-24. doi: 10.1016/j.ejmech.2014.03.054. Epub 2014 Mar 18. Eur J Med Chem. 2014. PMID: 24681986

4

Biological activities of new monohydroxylated brassinosteroid analogues with a carboxylic group in the side chain.

Kvasnica M, Oklestkova J, Bazgier V, Rarova L, Berka K, Strnad M. Kvasnica M, et al. Among authors: bazgier v. Steroids. 2014 Jul;85:58-64. doi: 10.1016/j.steroids.2014.04.007. Epub 2014 Apr 21. Steroids. 2014. PMID: 24769247

5

Synthesis, biological evaluation and molecular modeling of a novel series of 7-azaindole based tri-heterocyclic compounds as potent CDK2/Cyclin E inhibitors.

Baltus CB, Jorda R, Marot C, Berka K, Bazgier V, Kryštof V, Prié G, Viaud-Massuard MC. Baltus CB, et al. Among authors: bazgier v. Eur J Med Chem. 2016 Jan 27;108:701-719. doi: 10.1016/j.ejmech.2015.12.023. Epub 2015 Dec 19. Eur J Med Chem. 2016. PMID: 26741853

6

Design, synthesis and biological activities of new brassinosteroid analogues with a phenyl group in the side chain.

Kvasnica M, Oklestkova J, Bazgier V, Rárová L, Korinkova P, Mikulík J, Budesinsky M, Béres T, Berka K, Lu Q, Russinova E, Strnad M. Kvasnica M, et al. Among authors: bazgier v. Org Biomol Chem. 2016 Sep 21;14(37):8691-8701. doi: 10.1039/c6ob01479h. Org Biomol Chem. 2016. PMID: 27714217

7

Synthesis of novel aryl brassinosteroids through alkene cross-metathesis and preliminary biological study.

Korinkova P, Bazgier V, Oklestkova J, Rarova L, Strnad M, Kvasnica M. Korinkova P, et al. Among authors: bazgier v. Steroids. 2017 Nov;127:46-55. doi: 10.1016/j.steroids.2017.08.010. Epub 2017 Aug 31. Steroids. 2017. PMID: 28837783

8

Discovery of N²-(4-Amino-cyclohexyl)-9-cyclopentyl- N⁶-(4-morpholin-4-ylmethyl-phenyl)- 9H-purine-2,6-diamine as a Potent FLT3 Kinase Inhibitor for Acute Myeloid Leukemia with FLT3 Mutations.

Gucký T, Řezníčková E, Radošová Muchová T, Jorda R, Klejová Z, Malínková V, Berka K, Bazgier V, Ajani H, Lepšík M, Divoký V, Kryštof V. Gucký T, et al. Among authors: bazgier v. J Med Chem. 2018 May 10;61(9):3855-3869. doi: 10.1021/acs.jmedchem.7b01529. Epub 2018 Apr 30. J Med Chem. 2018. PMID: 29672049

9

Synthesis of novel galeterone derivatives and evaluation of their in vitro activity against prostate cancer cell lines.

Jorda R, Řezníčková E, Kiełczewska U, Maj J, Morzycki JW, Siergiejczyk L, Bazgier V, Berka K, Rárová L, Wojtkielewicz A. Jorda R, et al. Among authors: bazgier v. Eur J Med Chem. 2019 Oct 1;179:483-492. doi: 10.1016/j.ejmech.2019.06.040. Epub 2019 Jun 18. Eur J Med Chem. 2019. PMID: 31271960

10

Novel thiazolidinedione-hydroxamates as inhibitors of Mycobacterium tuberculosis virulence factor Zmp1.

Šlachtová V, Šebela M, Torfs E, Oorts L, Cappoen D, Berka K, Bazgier V, Brulíková L. Šlachtová V, et al. Among authors: bazgier v. Eur J Med Chem. 2020 Jan 1;185:111812. doi: 10.1016/j.ejmech.2019.111812. Epub 2019 Nov 5. Eur J Med Chem. 2020. PMID: 31703818

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