Marco-Contelles J - Search Results

1

Tetrahydropyranodiquinolin-8-amines as new, non hepatotoxic, antioxidant, and acetylcholinesterase inhibitors for Alzheimer's disease therapy.

Dgachi Y, Sokolov O, Luzet V, Godyń J, Panek D, Bonet A, Martin H, Iriepa I, Moraleda I, García-Iriepa C, Janockova J, Richert L, Soukup O, Malawska B, Chabchoub F, Marco-Contelles J, Ismaili L. Dgachi Y, et al. Eur J Med Chem. 2017 Jan 27;126:576-589. doi: 10.1016/j.ejmech.2016.11.050. Epub 2016 Nov 23. Eur J Med Chem. 2017. PMID: 27918993

2

Synthesis, acetylcholinesterase inhibition and neuroprotective activity of new tacrine analogues.

León R, Marco-Contelles J, García AG, Villarroya M. León R, et al. Bioorg Med Chem. 2005 Feb 15;13(4):1167-75. doi: 10.1016/j.bmc.2004.11.020. Bioorg Med Chem. 2005. PMID: 15670925

3

New multipotent tetracyclic tacrines with neuroprotective activity.

Marco-Contelles J, León R, de los Ríos C, García AG, López MG, Villarroya M. Marco-Contelles J, et al. Bioorg Med Chem. 2006 Dec 15;14(24):8176-85. doi: 10.1016/j.bmc.2006.09.025. Epub 2006 Sep 26. Bioorg Med Chem. 2006. PMID: 17005406

4

Synthesis and biological evaluation of new 4H-pyrano[2,3-b]quinoline derivatives that block acetylcholinesterase and cell calcium signals, and cause neuroprotection against calcium overload and free radicals.

Marco-Contelles J, León R, López MG, García AG, Villarroya M. Marco-Contelles J, et al. Eur J Med Chem. 2006 Dec;41(12):1464-9. doi: 10.1016/j.ejmech.2006.06.016. Epub 2006 Oct 6. Eur J Med Chem. 2006. PMID: 17030484

5

Novel multipotent tacrine-dihydropyridine hybrids with improved acetylcholinesterase inhibitory and neuroprotective activities as potential drugs for the treatment of Alzheimer's disease.

Marco-Contelles J, León R, de Los Ríos C, Guglietta A, Terencio J, López MG, García AG, Villarroya M. Marco-Contelles J, et al. J Med Chem. 2006 Dec 28;49(26):7607-10. doi: 10.1021/jm061047j. J Med Chem. 2006. PMID: 17181144

6

Synthesis of 6-amino-1,4-dihydropyridines that prevent calcium overload and neuronal death.

León R, de Los Ríos C, Marco-Contelles J, López MG, García AG, Villarroya M. León R, et al. Eur J Med Chem. 2008 Mar;43(3):668-74. doi: 10.1016/j.ejmech.2007.06.001. Epub 2007 Jul 5. Eur J Med Chem. 2008. PMID: 17692434

7

New tacrine-dihydropyridine hybrids that inhibit acetylcholinesterase, calcium entry, and exhibit neuroprotection properties.

León R, de los Ríos C, Marco-Contelles J, Huertas O, Barril X, Luque FJ, López MG, García AG, Villarroya M. León R, et al. Bioorg Med Chem. 2008 Aug 15;16(16):7759-69. doi: 10.1016/j.bmc.2008.07.005. Epub 2008 Jul 8. Bioorg Med Chem. 2008. PMID: 18640842

8

Tacripyrines, the first tacrine-dihydropyridine hybrids, as multitarget-directed ligands for the treatment of Alzheimer's disease.

Marco-Contelles J, León R, de los Ríos C, Samadi A, Bartolini M, Andrisano V, Huertas O, Barril X, Luque FJ, Rodríguez-Franco MI, López B, López MG, García AG, Carreiras Mdo C, Villarroya M. Marco-Contelles J, et al. J Med Chem. 2009 May 14;52(9):2724-32. doi: 10.1021/jm801292b. J Med Chem. 2009. PMID: 19374444

9

Synthesis and biological evaluation of 3,6-diamino-1H-pyrazolo[3,4-b]pyridine derivatives as protein kinase inhibitors.

Chioua M, Samadi A, Soriano E, Lozach O, Meijer L, Marco-Contelles J. Chioua M, et al. Bioorg Med Chem Lett. 2009 Aug 15;19(16):4566-9. doi: 10.1016/j.bmcl.2009.06.099. Epub 2009 Jul 3. Bioorg Med Chem Lett. 2009. PMID: 19615897

10

Molecular modelling, synthesis and acetylcholinesterase inhibition of ethyl 5-amino-2-methyl-6,7,8,9-tetrahydrobenzo[b][1,8]naphthyridine-3-carboxylate.

Soriano E, Samadi A, Chioua M, de los Ríos C, Marco-Contelles J. Soriano E, et al. Bioorg Med Chem Lett. 2010 May 1;20(9):2950-3. doi: 10.1016/j.bmcl.2010.03.010. Epub 2010 Mar 4. Bioorg Med Chem Lett. 2010. PMID: 20350807

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