Depreux P - Search Results

1

DNA Methylation Targeting: The DNMT/HMT Crosstalk Challenge.

Castillo-Aguilera O, Depreux P, Halby L, Arimondo PB, Goossens L. Castillo-Aguilera O, et al. Among authors: depreux p. Biomolecules. 2017 Jan 5;7(1):3. doi: 10.3390/biom7010003. Biomolecules. 2017. PMID: 28067760 Free PMC article. Review.

2

Quinazoline derivatives as anticancer drugs: a patent review (2011 - present).

Ravez S, Castillo-Aguilera O, Depreux P, Goossens L. Ravez S, et al. Among authors: depreux p. Expert Opin Ther Pat. 2015 Jul;25(7):789-804. doi: 10.1517/13543776.2015.1039512. Epub 2015 Apr 24. Expert Opin Ther Pat. 2015. PMID: 25910402 Review.

3

Synthesis and biological evaluation of di-aryl urea derivatives as c-Kit inhibitors.

Ravez S, Arsenlis S, Barczyk A, Dupont A, Frédérick R, Hesse S, Kirsch G, Depreux P, Goossens L. Ravez S, et al. Among authors: depreux p. Bioorg Med Chem. 2015 Nov 15;23(22):7340-7. doi: 10.1016/j.bmc.2015.10.035. Epub 2015 Oct 24. Bioorg Med Chem. 2015. PMID: 26526740

4

Design, synthesis, and DNA-binding of N-alkyl(anilino)quinazoline derivatives.

Garofalo A, Goossens L, Baldeyrou B, Lemoine A, Ravez S, Six P, David-Cordonnier MH, Bonte JP, Depreux P, Lansiaux A, Goossens JF. Garofalo A, et al. Among authors: depreux p. J Med Chem. 2010 Nov 25;53(22):8089-103. doi: 10.1021/jm1009605. Epub 2010 Oct 29. J Med Chem. 2010. PMID: 21033670

5

Inhibition of tumor cell growth and angiogenesis by 7-aminoalkoxy-4-aryloxy-quinazoline ureas, a novel series of multi-tyrosine kinase inhibitors.

Ravez S, Barczyk A, Six P, Cagnon A, Garofalo A, Goossens L, Depreux P. Ravez S, et al. Among authors: depreux p. Eur J Med Chem. 2014 May 22;79:369-81. doi: 10.1016/j.ejmech.2014.04.007. Epub 2014 Apr 5. Eur J Med Chem. 2014. PMID: 24747748

6

Impact of aryloxy-linked quinazolines: a novel series of selective VEGFR-2 receptor tyrosine kinase inhibitors.

Garofalo A, Goossens L, Six P, Lemoine A, Ravez S, Farce A, Depreux P. Garofalo A, et al. Among authors: depreux p. Bioorg Med Chem Lett. 2011 Apr 1;21(7):2106-12. doi: 10.1016/j.bmcl.2011.01.137. Epub 2011 Feb 3. Bioorg Med Chem Lett. 2011. PMID: 21353546

7

Synthesis and structure-activity relationships of (aryloxy)quinazoline ureas as novel, potent, and selective vascular endothelial growth factor receptor-2 inhibitors.

Garofalo A, Farce A, Ravez S, Lemoine A, Six P, Chavatte P, Goossens L, Depreux P. Garofalo A, et al. Among authors: depreux p. J Med Chem. 2012 Feb 9;55(3):1189-204. doi: 10.1021/jm2013453. Epub 2012 Jan 25. J Med Chem. 2012. PMID: 22229669

8

Amine coupling versus biotin capture for the assessment of sulfonamide as ligands of hCA isoforms.

Rogez-Florent T, Goossens L, Drucbert AS, Duban-Deweer S, Six P, Depreux P, Danzé PM, Goossens JF, Foulon C. Rogez-Florent T, et al. Among authors: depreux p. Anal Biochem. 2016 Oct 15;511:42-51. doi: 10.1016/j.ab.2016.07.029. Epub 2016 Jul 30. Anal Biochem. 2016. PMID: 27485269

9

Chiral separation of new sulfonamide derivatives and evaluation of their enantioselective affinity for human carbonic anhydrase II by microscale thermophoresis and surface plasmon resonance.

Rogez-Florent T, Foulon C, Drucbert AS, Schifano N, Six P, Devassine S, Depreux P, Danzé PM, Goossens L, Danel C, Goossens JF. Rogez-Florent T, et al. Among authors: depreux p. J Pharm Biomed Anal. 2017 Apr 15;137:113-122. doi: 10.1016/j.jpba.2017.01.023. Epub 2017 Jan 9. J Pharm Biomed Anal. 2017. PMID: 28110167

10

Design, solid-phase synthesis, and biological evaluation of novel 1,5-diarylpyrrole-3-carboxamides as carbonic anhydrase IX inhibitors.

Gluszok S, Frédérick R, Foulon C, Klupsch F, Supuran CT, Vullo D, Scozzafava A, Goossens JF, Masereel B, Depreux P, Goossens L. Gluszok S, et al. Among authors: depreux p. Bioorg Med Chem. 2010 Nov 1;18(21):7392-401. doi: 10.1016/j.bmc.2010.09.007. Epub 2010 Sep 7. Bioorg Med Chem. 2010. PMID: 20880712

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