Salas-Sarduy E - Search Results

1

Rational design and synthesis of affinity matrices based on proteases immobilized onto cellulose membranes.

Del Monte-Martínez A, González-Bacerio J, Cutiño-Avila B, Rojas J, Chappé M, Salas-Sarduy E, Pascual I, Guisán JM. Del Monte-Martínez A, et al. Prep Biochem Biotechnol. 2017 Sep 14;47(8):745-753. doi: 10.1080/10826068.2017.1315600. Epub 2017 Apr 12. Prep Biochem Biotechnol. 2017. PMID: 28402172

2

Identification of (4-(9H-fluoren-9-yl) piperazin-1-yl) methanone derivatives as falcipain 2 inhibitors active against Plasmodium falciparum cultures.

Hernández-González JE, Salas-Sarduy E, Hernández Ramírez LF, Pascual MJ, Álvarez DE, Pabón A, Leite VBP, Pascutti PG, Valiente PA. Hernández-González JE, et al. Biochim Biophys Acta Gen Subj. 2018 Dec;1862(12):2911-2923. doi: 10.1016/j.bbagen.2018.09.015. Epub 2018 Sep 22. Biochim Biophys Acta Gen Subj. 2018. PMID: 30253205 Free article.

3

In silico identification of noncompetitive inhibitors targeting an uncharacterized allosteric site of falcipain-2.

Hernández González JE, Salas-Sarduy E, Hernández Alvarez L, Barreto Gomes DE, Pascutti PG, Oostenbrink C, Leite VBP. Hernández González JE, et al. Among authors: salas sarduy e. J Comput Aided Mol Des. 2021 Oct;35(10):1067-1079. doi: 10.1007/s10822-021-00420-7. Epub 2021 Oct 7. J Comput Aided Mol Des. 2021. PMID: 34617191

4

Tetracycline Derivatives Inhibit Plasmodial Cysteine Protease Falcipain-2 through Binding to a Distal Allosteric Site.

Hernández González JE, Alberca LN, Masforrol González Y, Reyes Acosta O, Talevi A, Salas-Sarduy E. Hernández González JE, et al. Among authors: salas sarduy e. J Chem Inf Model. 2022 Jan 10;62(1):159-175. doi: 10.1021/acs.jcim.1c01189. Epub 2021 Dec 28. J Chem Inf Model. 2022. PMID: 34962803

5

Identification of Tight-Binding Plasmepsin II and Falcipain 2 Inhibitors in Aqueous Extracts of Marine Invertebrates by the Combination of Enzymatic and Interaction-Based Assays.

Salas-Sarduy E, Guerra Y, Covaleda Cortés G, Avilés FX, Chávez Planes MA. Salas-Sarduy E, et al. Mar Drugs. 2017 Apr 21;15(4):123. doi: 10.3390/md15040123. Mar Drugs. 2017. PMID: 28430158 Free PMC article.

6

Novel scaffolds for inhibition of Cruzipain identified from high-throughput screening of anti-kinetoplastid chemical boxes.

Salas-Sarduy E, Landaburu LU, Karpiak J, Madauss KP, Cazzulo JJ, Agüero F, Alvarez VE. Salas-Sarduy E, et al. Sci Rep. 2017 Sep 21;7(1):12073. doi: 10.1038/s41598-017-12170-4. Sci Rep. 2017. PMID: 28935948 Free PMC article.

7

Potent and selective inhibitors for M32 metallocarboxypeptidases identified from high-throughput screening of anti-kinetoplastid chemical boxes.

Salas-Sarduy E, Landaburu LU, Carmona AK, Cazzulo JJ, Agüero F, Alvarez VE, Niemirowicz GT. Salas-Sarduy E, et al. PLoS Negl Trop Dis. 2019 Jul 22;13(7):e0007560. doi: 10.1371/journal.pntd.0007560. eCollection 2019 Jul. PLoS Negl Trop Dis. 2019. PMID: 31329594 Free PMC article.

8

Screening and Identification of Metacaspase Inhibitors: Evaluation of Inhibition Mechanism and Trypanocidal Activity.

Pérez B, Bouvier LA, Cazzulo JJ, Agüero F, Salas-Sarduy E, Alvarez VE. Pérez B, et al. Among authors: salas sarduy e. Antimicrob Agents Chemother. 2021 Feb 17;65(3):e01330-20. doi: 10.1128/AAC.01330-20. Print 2021 Feb 17. Antimicrob Agents Chemother. 2021. PMID: 33318019 Free PMC article.

9

Target-based Screening of the Chagas Box: Setting Up Enzymatic Assays to Discover Specific Inhibitors Across Bioactive Compounds.

Salas-Sarduy E, Niemirowicz GT, José Cazzulo J, Alvarez VE. Salas-Sarduy E, et al. Curr Med Chem. 2019;26(36):6672-6686. doi: 10.2174/0929867326666190705160637. Curr Med Chem. 2019. PMID: 31284853 Review.

10

Antiparasitic effect of a fraction enriched in tight-binding protease inhibitors isolated from the Caribbean coral Plexaura homomalla.

Salas-Sarduy E, Cabrera-Muñoz A, Cauerhff A, González-González Y, Trejo SA, Chidichimo A, Chávez-Planes Mde L, Cazzulo JJ. Salas-Sarduy E, et al. Exp Parasitol. 2013 Nov;135(3):611-22. doi: 10.1016/j.exppara.2013.09.013. Epub 2013 Sep 30. Exp Parasitol. 2013. PMID: 24090569

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