Ejaz SA - Search Results

1

Chemoselective synthesis and biological evaluation of arylated 2-(Trifluoromethyl) quinolines as nucleotide pyrophosphatase (NPPs) inhibitors.

Kuhrt D, Ejaz SA, Afzal S, Khan SU, Lecka J, Sévigny J, Ehlers P, Spannenberg A, Iqbal J, Langer P. Kuhrt D, et al. Among authors: ejaz sa. Eur J Med Chem. 2017 Sep 29;138:816-829. doi: 10.1016/j.ejmech.2017.07.017. Epub 2017 Jul 13. Eur J Med Chem. 2017. PMID: 28735213

2

Diarylsulfonamides and their bioisosteres as dual inhibitors of alkaline phosphatase and carbonic anhydrase: Structure activity relationship and molecular modelling studies.

Al-Rashida M, Ejaz SA, Ali S, Shaukat A, Hamayoun M, Ahmed M, Iqbal J. Al-Rashida M, et al. Among authors: ejaz sa. Bioorg Med Chem. 2015 May 15;23(10):2435-44. doi: 10.1016/j.bmc.2015.03.054. Epub 2015 Mar 27. Bioorg Med Chem. 2015. PMID: 25865133

3

Efficient one-pot synthesis of 5-perfluoroalkylpyrazoles by cyclization of hydrazone dianions.

Ngo TN, Ejaz SA, Hung TQ, Dang TT, Iqbal J, Lecka J, Sévigny J, Langer P. Ngo TN, et al. Among authors: ejaz sa. Org Biomol Chem. 2015 Aug 14;13(30):8277-90. doi: 10.1039/c5ob01151e. Org Biomol Chem. 2015. PMID: 26140545

4

Synthesis of 3,3'-carbonyl-bis(chromones) and their activity as mammalian alkaline phosphatase inhibitors.

Miliutina M, Ejaz SA, Iaroshenko VO, Villinger A, Iqbal J, Langer P. Miliutina M, et al. Among authors: ejaz sa. Org Biomol Chem. 2016 Jan 14;14(2):495-502. doi: 10.1039/c5ob01350j. Org Biomol Chem. 2016. PMID: 26490672

5

2-Alkoxy-3-(sulfonylarylaminomethylene)-chroman-4-ones as potent and selective inhibitors of ectonucleotidases.

al-Rashida M, Batool G, Sattar A, Ejaz SA, Khan S, Lecka J, Sévigny J, Hameed A, Iqbal J. al-Rashida M, et al. Among authors: ejaz sa. Eur J Med Chem. 2016 Jun 10;115:484-94. doi: 10.1016/j.ejmech.2016.02.073. Epub 2016 Mar 3. Eur J Med Chem. 2016. PMID: 27054295

6

New one-pot synthesis of N-fused isoquinoline derivatives by palladium-catalyzed C-H arylation: potent inhibitors of nucleotide pyrophosphatase-1 and -3.

Ausekle E, Ejaz SA, Khan SU, Ehlers P, Villinger A, Lecka J, Sévigny J, Iqbal J, Langer P. Ausekle E, et al. Among authors: ejaz sa. Org Biomol Chem. 2016 Dec 28;14(48):11402-11414. doi: 10.1039/c6ob02236g. Epub 2016 Nov 18. Org Biomol Chem. 2016. PMID: 27858054

7

Cholinesterases inhibition and molecular modeling studies of piperidyl-thienyl and 2-pyrazoline derivatives of chalcones.

Shah MS, Khan SU, Ejaz SA, Afridi S, Rizvi SUF, Najam-Ul-Haq M, Iqbal J. Shah MS, et al. Among authors: ejaz sa. Biochem Biophys Res Commun. 2017 Jan 22;482(4):615-624. doi: 10.1016/j.bbrc.2016.11.082. Epub 2016 Nov 16. Biochem Biophys Res Commun. 2017. PMID: 27865835

8

Synthesis, alkaline phosphatase inhibition studies and molecular docking of novel derivatives of 4-quinolones.

Miliutina M, Ejaz SA, Khan SU, Iaroshenko VO, Villinger A, Iqbal J, Langer P. Miliutina M, et al. Among authors: ejaz sa. Eur J Med Chem. 2017 Jan 27;126:408-420. doi: 10.1016/j.ejmech.2016.11.036. Epub 2016 Nov 17. Eur J Med Chem. 2017. PMID: 27907877

9

Synthesis, functionalization and biological activity of arylated derivatives of (+)-estrone.

Ivanov A, Ejaz SA, Shah SJA, Ehlers P, Villinger A, Frank E, Schneider G, Wölfling J, Rahman Q, Iqbal J, Langer P. Ivanov A, et al. Among authors: ejaz sa. Bioorg Med Chem. 2017 Feb 1;25(3):949-962. doi: 10.1016/j.bmc.2016.12.009. Epub 2016 Dec 9. Bioorg Med Chem. 2017. PMID: 28034648

10

Synthesis, characterization and biological evaluation of novel chalcone sulfonamide hybrids as potent intestinal alkaline phosphatase inhibitors.

Ejaz SA, Saeed A, Siddique MN, Nisa ZU, Khan S, Lecka J, Sévigny J, Iqbal J. Ejaz SA, et al. Bioorg Chem. 2017 Feb;70:229-236. doi: 10.1016/j.bioorg.2017.01.003. Epub 2017 Jan 5. Bioorg Chem. 2017. PMID: 28110961

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