Woster PM - Search Results

1

Cyclic peptide inhibitors of lysine-specific demethylase 1 with improved potency identified by alanine scanning mutagenesis.

Kumarasinghe IR, Woster PM. Kumarasinghe IR, et al. Among authors: woster pm. Eur J Med Chem. 2018 Mar 25;148:210-220. doi: 10.1016/j.ejmech.2018.01.098. Epub 2018 Feb 7. Eur J Med Chem. 2018. PMID: 29459279 Free PMC article.

2

(Bis)urea and (bis)thiourea inhibitors of lysine-specific demethylase 1 as epigenetic modulators.

Sharma SK, Wu Y, Steinbergs N, Crowley ML, Hanson AS, Casero RA, Woster PM. Sharma SK, et al. Among authors: woster pm. J Med Chem. 2010 Jul 22;53(14):5197-212. doi: 10.1021/jm100217a. J Med Chem. 2010. PMID: 20568780 Free PMC article.

3

Low molecular weight amidoximes that act as potent inhibitors of lysine-specific demethylase 1.

Hazeldine S, Pachaiyappan B, Steinbergs N, Nowotarski S, Hanson AS, Casero RA Jr, Woster PM. Hazeldine S, et al. Among authors: woster pm. J Med Chem. 2012 Sep 13;55(17):7378-91. doi: 10.1021/jm3002845. Epub 2012 Sep 4. J Med Chem. 2012. PMID: 22876979 Free PMC article.

4

Design of small molecule epigenetic modulators.

Pachaiyappan B, Woster PM. Pachaiyappan B, et al. Among authors: woster pm. Bioorg Med Chem Lett. 2014 Jan 1;24(1):21-32. doi: 10.1016/j.bmcl.2013.11.001. Epub 2013 Nov 13. Bioorg Med Chem Lett. 2014. PMID: 24300735 Free PMC article. Review.

5

Synthesis and evaluation of novel cyclic Peptide inhibitors of lysine-specific demethylase 1.

Kumarasinghe IR, Woster PM. Kumarasinghe IR, et al. Among authors: woster pm. ACS Med Chem Lett. 2013 Nov 8;5(1):29-33. doi: 10.1021/ml4002997. eCollection 2014 Jan 9. ACS Med Chem Lett. 2013. PMID: 24883177 Free PMC article.

6

Structure-activity study for (bis)ureidopropyl- and (bis)thioureidopropyldiamine LSD1 inhibitors with 3-5-3 and 3-6-3 carbon backbone architectures.

Nowotarski SL, Pachaiyappan B, Holshouser SL, Kutz CJ, Li Y, Huang Y, Sharma SK, Casero RA Jr, Woster PM. Nowotarski SL, et al. Among authors: woster pm. Bioorg Med Chem. 2015 Apr 1;23(7):1601-12. doi: 10.1016/j.bmc.2015.01.049. Epub 2015 Feb 7. Bioorg Med Chem. 2015. PMID: 25725609 Free PMC article.

7

Epigenetics: Novel Therapeutics Targeting Epigenetics.

Conway SJ, Woster PM, Greenlee WJ, Georg G, Wang S. Conway SJ, et al. Among authors: woster pm. J Med Chem. 2016 Feb 25;59(4):1247-8. doi: 10.1021/acs.jmedchem.6b00098. Epub 2016 Jan 29. J Med Chem. 2016. PMID: 26824165 No abstract available.

8

Antibacterial Diamines Targeting Bacterial Membranes.

Wang B, Pachaiyappan B, Gruber JD, Schmidt MG, Zhang YM, Woster PM. Wang B, et al. Among authors: woster pm. J Med Chem. 2016 Apr 14;59(7):3140-51. doi: 10.1021/acs.jmedchem.5b01912. Epub 2016 Mar 28. J Med Chem. 2016. PMID: 26964758 Free PMC article.

9

Inhibition of the histone demethylase KDM4B leads to activation of KDM1A, attenuates bacterial-induced pro-inflammatory cytokine release, and reduces osteoclastogenesis.

Kirkpatrick JE, Kirkwood KL, Woster PM. Kirkpatrick JE, et al. Among authors: woster pm. Epigenetics. 2018;13(5):557-572. doi: 10.1080/15592294.2018.1481703. Epub 2018 Aug 7. Epigenetics. 2018. PMID: 29927684 Free PMC article.

10

Synthesis and evaluation of small molecule inhibitors of LSD1 for use against MYCN-expressing neuroblastoma.

Mills CM, Turner J, Piña IC, Garrabrant KA, Geerts D, Bachmann AS, Peterson YK, Woster PM. Mills CM, et al. Among authors: woster pm. Eur J Med Chem. 2022 Dec 15;244:114818. doi: 10.1016/j.ejmech.2022.114818. Epub 2022 Oct 7. Eur J Med Chem. 2022. PMID: 36223680

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