Gomaa MS - Search Results

1

Synthesis, biological evaluation, and molecular docking investigation of benzhydrol- and indole-based dual PPAR-γ/FFAR1 agonists.

Darwish KM, Salama I, Mostafa S, Gomaa MS, Khafagy ES, Helal MA. Darwish KM, et al. Among authors: gomaa ms. Bioorg Med Chem Lett. 2018 May 15;28(9):1595-1602. doi: 10.1016/j.bmcl.2018.03.051. Epub 2018 Mar 21. Bioorg Med Chem Lett. 2018. PMID: 29615345

2

Small molecule inhibitors of retinoic acid 4-hydroxylase (CYP26): synthesis and biological evaluation of imidazole methyl 3-(4-(aryl-2-ylamino)phenyl)propanoates.

Gomaa MS, Bridgens CE, Aboraia AS, Veal GJ, Redfern CP, Brancale A, Armstrong JL, Simons C. Gomaa MS, et al. J Med Chem. 2011 Apr 28;54(8):2778-91. doi: 10.1021/jm101583w. Epub 2011 Mar 23. J Med Chem. 2011. PMID: 21428449

3

Synthesis and CYP26A1 inhibitory activity of novel methyl 3-[4-(arylamino)phenyl]-3-(azole)-2,2-dimethylpropanoates.

Gomaa MS, Lim AS, Lau SC, Watts AM, Illingworth NA, Bridgens CE, Veal GJ, Redfern CP, Brancale A, Armstrong JL, Simons C. Gomaa MS, et al. Bioorg Med Chem. 2012 Oct 15;20(20):6080-8. doi: 10.1016/j.bmc.2012.08.044. Epub 2012 Aug 30. Bioorg Med Chem. 2012. PMID: 22989911

4

Design, synthesis, and biological evaluation of novel thiazolidinediones as PPARγ/FFAR1 dual agonists.

Darwish KM, Salama I, Mostafa S, Gomaa MS, Helal MA. Darwish KM, et al. Among authors: gomaa ms. Eur J Med Chem. 2016 Feb 15;109:157-72. doi: 10.1016/j.ejmech.2015.12.049. Epub 2015 Dec 31. Eur J Med Chem. 2016. PMID: 26774923

5

Design, selective alkylation and X-ray crystal structure determination of dihydro-indolyl-1,2,4-triazole-3-thione and its 3-benzylsulfanyl analogue as potent anticancer agents.

Boraei AT, Gomaa MS, El Ashry ES, Duerkop A. Boraei AT, et al. Among authors: gomaa ms. Eur J Med Chem. 2017 Jan 5;125:360-371. doi: 10.1016/j.ejmech.2016.09.046. Epub 2016 Sep 15. Eur J Med Chem. 2017. PMID: 27688190

6

Design, synthesis and 2D QSAR study of novel pyridine and quinolone hydrazone derivatives as potential antimicrobial and antitubercular agents.

Abdelrahman MA, Salama I, Gomaa MS, Elaasser MM, Abdel-Aziz MM, Soliman DH. Abdelrahman MA, et al. Among authors: gomaa ms. Eur J Med Chem. 2017 Sep 29;138:698-714. doi: 10.1016/j.ejmech.2017.07.004. Epub 2017 Jul 4. Eur J Med Chem. 2017. PMID: 28715707

7

Design and synthesis of new phthalazine-based derivatives as potential EGFR inhibitors for the treatment of hepatocellular carcinoma.

Boraei ATA, Ashour HK, El Tamany ESH, Abdelmoaty N, El-Falouji AI, Gomaa MS. Boraei ATA, et al. Among authors: gomaa ms. Bioorg Chem. 2019 Apr;85:293-307. doi: 10.1016/j.bioorg.2018.12.039. Epub 2018 Dec 31. Bioorg Chem. 2019. PMID: 30654221

8

Synthesis and biological evaluation of novel cYY analogues targeting Mycobacterium tuberculosis CYP121A1.

Kishk SM, McLean KJ, Sood S, Helal MA, Gomaa MS, Salama I, Mostafa SM, de Carvalho LPS, Munro AW, Simons C. Kishk SM, et al. Among authors: gomaa ms. Bioorg Med Chem. 2019 Apr 15;27(8):1546-1561. doi: 10.1016/j.bmc.2019.02.051. Epub 2019 Feb 27. Bioorg Med Chem. 2019. PMID: 30837169 Free PMC article.

9

Design and Synthesis of Imidazole and Triazole Pyrazoles as Mycobacterium Tuberculosis CYP121A1 Inhibitors.

Kishk SM, McLean KJ, Sood S, Smith D, Evans JWD, Helal MA, Gomaa MS, Salama I, Mostafa SM, de Carvalho LPS, Levy CW, Munro AW, Simons C. Kishk SM, et al. Among authors: gomaa ms. ChemistryOpen. 2019 Jul 23;8(7):995-1011. doi: 10.1002/open.201900227. eCollection 2019 Jul. ChemistryOpen. 2019. PMID: 31367508 Free PMC article.

10

Sulfadiazine Exerts Potential Anticancer Effect in HepG2 and MCF7 Cells by Inhibiting TNFα, IL1b, COX-1, COX-2, 5-LOX Gene Expression: Evidence from In Vitro and Computational Studies.

Gomaa M, Gad W, Hussein D, Pottoo FH, Tawfeeq N, Alturki M, Alfahad D, Alanazi R, Salama I, Aziz M, Zahra A, Hanafy A. Gomaa M, et al. Pharmaceuticals (Basel). 2024 Jan 31;17(2):189. doi: 10.3390/ph17020189. Pharmaceuticals (Basel). 2024. PMID: 38399404 Free PMC article.

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