Endo Y - Search Results

1

Novel androgen receptor full antagonists: Design, synthesis, and a docking study of glycerol and aminoglycerol derivatives that contain p-carborane cages.

Kaise A, Ohta K, Fujii S, Oda A, Goto T, Endo Y. Kaise A, et al. Among authors: endo y. Bioorg Med Chem. 2018 Jul 30;26(13):3805-3811. doi: 10.1016/j.bmc.2018.06.007. Epub 2018 Jun 7. Bioorg Med Chem. 2018. PMID: 29903411

2

Acidic heterocycles as novel hydrophilic pharmacophore of androgen receptor ligands with a carborane core structure.

Fujii S, Ohta K, Goto T, Kagechika H, Endo Y. Fujii S, et al. Among authors: endo y. Bioorg Med Chem. 2009 Jan 1;17(1):344-50. doi: 10.1016/j.bmc.2008.10.060. Epub 2008 Oct 30. Bioorg Med Chem. 2009. PMID: 19022677

3

Synthesis and biological evaluation of p-carborane bisphenols and their derivatives: structure-activity relationship for estrogenic activity.

Ogawa T, Ohta K, Iijima T, Suzuki T, Ohta S, Endo Y. Ogawa T, et al. Among authors: endo y. Bioorg Med Chem. 2009 Feb 1;17(3):1109-17. doi: 10.1016/j.bmc.2008.12.044. Epub 2008 Dec 25. Bioorg Med Chem. 2009. PMID: 19141368

4

Novel estrogen receptor (ER) modulators: carbamate and thiocarbamate derivatives with m-carborane bisphenol structure.

Ohta K, Ogawa T, Suzuki T, Ohta S, Endo Y. Ohta K, et al. Among authors: endo y. Bioorg Med Chem. 2009 Dec 1;17(23):7958-63. doi: 10.1016/j.bmc.2009.10.018. Epub 2009 Oct 13. Bioorg Med Chem. 2009. PMID: 19857971

5

Design and synthesis of androgen receptor full antagonists bearing a p-carborane cage: promising ligands for anti-androgen withdrawal syndrome.

Goto T, Ohta K, Fujii S, Ohta S, Endo Y. Goto T, et al. Among authors: endo y. J Med Chem. 2010 Jul 8;53(13):4917-26. doi: 10.1021/jm100316f. J Med Chem. 2010. PMID: 20521823

6

Crystal structure, docking study and structure-activity relationship of carborane-containing androgen receptor antagonist 3-(12-hydroxymethyl-1,12-dicarba-closo-dodecaboran-1-yl)benzonitrile.

Ohta K, Goto T, Fujii S, Kawahata M, Oda A, Ohta S, Yamaguchi K, Hirono S, Endo Y. Ohta K, et al. Among authors: endo y. Bioorg Med Chem. 2011 Jun 1;19(11):3540-8. doi: 10.1016/j.bmc.2011.04.017. Epub 2011 Apr 20. Bioorg Med Chem. 2011. PMID: 21536446

7

Estrogenic activity of B-fluorinated o-carborane-1,2-bisphenol synthesized via S(N)Ar reaction.

Ohta K, Ogawa T, Endo Y. Ohta K, et al. Among authors: endo y. Bioorg Med Chem Lett. 2012 Jul 15;22(14):4728-30. doi: 10.1016/j.bmcl.2012.05.068. Epub 2012 May 30. Bioorg Med Chem Lett. 2012. PMID: 22695130

8

Enhanced estrogen receptor beta (ERβ) selectivity of fluorinated carborane-containing ER modulators.

Ohta K, Ogawa T, Kaise A, Endo Y. Ohta K, et al. Among authors: endo y. Bioorg Med Chem Lett. 2013 Dec 15;23(24):6555-8. doi: 10.1016/j.bmcl.2013.10.067. Epub 2013 Nov 7. Bioorg Med Chem Lett. 2013. PMID: 24268550

9

Novel estrogen receptor (ER) modulators containing various hydrophobic bent-core structures.

Ohta K, Ogawa T, Kaise A, Endo Y. Ohta K, et al. Among authors: endo y. Bioorg Med Chem. 2014 Jul 1;22(13):3508-14. doi: 10.1016/j.bmc.2014.04.022. Epub 2014 Apr 20. Bioorg Med Chem. 2014. PMID: 24837157

10

Structure-activity relationship study of diphenylamine-based estrogen receptor (ER) antagonists.

Ohta K, Chiba Y, Kaise A, Endo Y. Ohta K, et al. Among authors: endo y. Bioorg Med Chem. 2015 Feb 15;23(4):861-7. doi: 10.1016/j.bmc.2014.12.022. Epub 2015 Jan 6. Bioorg Med Chem. 2015. PMID: 25614118

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