Kaise A - Search Results

1

Novel androgen receptor full antagonists: Design, synthesis, and a docking study of glycerol and aminoglycerol derivatives that contain p-carborane cages.

Kaise A, Ohta K, Fujii S, Oda A, Goto T, Endo Y. Kaise A, et al. Bioorg Med Chem. 2018 Jul 30;26(13):3805-3811. doi: 10.1016/j.bmc.2018.06.007. Epub 2018 Jun 7. Bioorg Med Chem. 2018. PMID: 29903411

2

Enhanced estrogen receptor beta (ERβ) selectivity of fluorinated carborane-containing ER modulators.

Ohta K, Ogawa T, Kaise A, Endo Y. Ohta K, et al. Among authors: kaise a. Bioorg Med Chem Lett. 2013 Dec 15;23(24):6555-8. doi: 10.1016/j.bmcl.2013.10.067. Epub 2013 Nov 7. Bioorg Med Chem Lett. 2013. PMID: 24268550

3

Novel estrogen receptor (ER) modulators containing various hydrophobic bent-core structures.

Ohta K, Ogawa T, Kaise A, Endo Y. Ohta K, et al. Among authors: kaise a. Bioorg Med Chem. 2014 Jul 1;22(13):3508-14. doi: 10.1016/j.bmc.2014.04.022. Epub 2014 Apr 20. Bioorg Med Chem. 2014. PMID: 24837157

4

Structure-activity relationship study of diphenylamine-based estrogen receptor (ER) antagonists.

Ohta K, Chiba Y, Kaise A, Endo Y. Ohta K, et al. Among authors: kaise a. Bioorg Med Chem. 2015 Feb 15;23(4):861-7. doi: 10.1016/j.bmc.2014.12.022. Epub 2015 Jan 6. Bioorg Med Chem. 2015. PMID: 25614118

5

Synthesis and biological evaluation of novel m-carborane-containing estrogen receptor partial agonists as SERM candidates.

Ohta K, Ogawa T, Kaise A, Endo Y. Ohta K, et al. Among authors: kaise a. Bioorg Med Chem Lett. 2015 Aug 15;25(16):3213-6. doi: 10.1016/j.bmcl.2015.05.083. Epub 2015 Jun 3. Bioorg Med Chem Lett. 2015. PMID: 26077489

6

Design and synthesis of carborane-containing estrogen receptor-beta (ERβ)-selective ligands.

Ohta K, Ogawa T, Oda A, Kaise A, Endo Y. Ohta K, et al. Among authors: kaise a. Bioorg Med Chem Lett. 2015 Oct 1;25(19):4174-8. doi: 10.1016/j.bmcl.2015.08.007. Epub 2015 Aug 7. Bioorg Med Chem Lett. 2015. PMID: 26298498

7

Symmetric 4,4'-(piperidin-4-ylidenemethylene)bisphenol derivatives as novel tunable estrogen receptor (ER) modulators.

Sato M, Ohta K, Kaise A, Aoto S, Endo Y. Sato M, et al. Among authors: kaise a. Bioorg Med Chem. 2016 Mar 1;24(5):1089-94. doi: 10.1016/j.bmc.2016.01.035. Epub 2016 Jan 18. Bioorg Med Chem. 2016. PMID: 26822566

8

Design, synthesis, and anti-proliferative activity of 1-(4-methoxyphenyl)-12-hydroxymethyl-p-carborane derivatives.

Kaise A, Ohta K, Endo Y. Kaise A, et al. Eur J Med Chem. 2016 Oct 21;122:257-263. doi: 10.1016/j.ejmech.2016.06.029. Epub 2016 Jun 18. Eur J Med Chem. 2016. PMID: 27371927

9

Novel p-carborane-containing multitarget anticancer agents inspired by the metabolism of 17β-estradiol.

Kaise A, Ohta K, Endo Y. Kaise A, et al. Bioorg Med Chem. 2017 Dec 15;25(24):6371-6378. doi: 10.1016/j.bmc.2017.10.006. Epub 2017 Oct 12. Bioorg Med Chem. 2017. PMID: 29054710

10

Design and synthesis of p-carborane-containing sulfamates as multitarget anti-breast cancer agents.

Kaise A, Ohta K, Shirata C, Endo Y. Kaise A, et al. Bioorg Med Chem. 2017 Dec 15;25(24):6417-6426. doi: 10.1016/j.bmc.2017.10.013. Epub 2017 Oct 16. Bioorg Med Chem. 2017. PMID: 29102082

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