Horenstein NA - Search Results

1

Novel 5-(quinuclidin-3-ylmethyl)-1,2,4-oxadiazoles to investigate the activation of the α7 nicotinic acetylcholine receptor subtype: Synthesis and electrophysiological evaluation.

Quadri M, Silnović A, Matera C, Horenstein NA, Stokes C, De Amici M, Papke RL, Dallanoce C. Quadri M, et al. Among authors: horenstein na. Eur J Med Chem. 2018 Dec 5;160:207-228. doi: 10.1016/j.ejmech.2018.10.015. Epub 2018 Oct 11. Eur J Med Chem. 2018. PMID: 30342362 Free PMC article.

2

Effects at a distance in alpha 7 nAChR selective agonists: benzylidene substitutions that regulate potency and efficacy.

Papke RL, Meyer EM, Lavieri S, Bollampally SR, Papke TA, Horenstein NA, Itoh Y, Porter Papke JK. Papke RL, et al. Among authors: horenstein na. Neuropharmacology. 2004 Jun;46(7):1023-38. doi: 10.1016/j.neuropharm.2004.01.005. Neuropharmacology. 2004. PMID: 15081799

3

The structural basis for GTS-21 selectivity between human and rat nicotinic alpha7 receptors.

Stokes C, Papke JK, Horenstein NA, Kem WR, McCormack TJ, Papke RL. Stokes C, et al. Among authors: horenstein na. Mol Pharmacol. 2004 Jul;66(1):14-24. doi: 10.1124/mol.66.1.14. Mol Pharmacol. 2004. PMID: 15213292

4

The effects of subunit composition on the inhibition of nicotinic receptors by the amphipathic blocker 2,2,6,6-tetramethylpiperidin-4-yl heptanoate.

Papke RL, Buhr JD, Francis MM, Choi KI, Thinschmidt JS, Horenstein NA. Papke RL, et al. Among authors: horenstein na. Mol Pharmacol. 2005 Jun;67(6):1977-90. doi: 10.1124/mol.105.011676. Epub 2005 Mar 10. Mol Pharmacol. 2005. PMID: 15761116

5

Molecular dissection of tropisetron, an alpha7 nicotinic acetylcholine receptor-selective partial agonist.

Papke RL, Schiff HC, Jack BA, Horenstein NA. Papke RL, et al. Among authors: horenstein na. Neurosci Lett. 2005 Apr 22;378(3):140-4. doi: 10.1016/j.neulet.2004.12.025. Epub 2005 Jan 5. Neurosci Lett. 2005. PMID: 15781147

6

The characterization of a novel rigid nicotine analog with alpha7-selective nAChR agonist activity and modulation of agonist properties by boron inclusion.

Papke RL, Zheng G, Horenstein NA, Dwoskin LP, Crooks PA. Papke RL, et al. Among authors: horenstein na. Bioorg Med Chem Lett. 2005 Sep 1;15(17):3874-80. doi: 10.1016/j.bmcl.2005.05.118. Bioorg Med Chem Lett. 2005. PMID: 16005216 Free PMC article.

7

Reversal of agonist selectivity by mutations of conserved amino acids in the binding site of nicotinic acetylcholine receptors.

Horenstein NA, McCormack TJ, Stokes C, Ren K, Papke RL. Horenstein NA, et al. J Biol Chem. 2007 Feb 23;282(8):5899-909. doi: 10.1074/jbc.M609202200. Epub 2006 Dec 21. J Biol Chem. 2007. PMID: 17189260 Free article.

8

Quinuclidines as selective agonists for alpha-7 nicotinic acetylcholine receptors.

Leonik FM, Papke RL, Horenstein NA. Leonik FM, et al. Among authors: horenstein na. Bioorg Med Chem Lett. 2007 Mar 15;17(6):1520-2. doi: 10.1016/j.bmcl.2007.01.003. Epub 2007 Jan 12. Bioorg Med Chem Lett. 2007. PMID: 17276680

9

Multiple pharmacophores for the selective activation of nicotinic alpha7-type acetylcholine receptors.

Horenstein NA, Leonik FM, Papke RL. Horenstein NA, et al. Mol Pharmacol. 2008 Dec;74(6):1496-511. doi: 10.1124/mol.108.048892. Epub 2008 Sep 2. Mol Pharmacol. 2008. PMID: 18768388 Free PMC article.

10

Synthesis of H-bonding probes of alpha7 nAChR agonist selectivity.

Wang J, Papke RL, Horenstein NA. Wang J, et al. Among authors: horenstein na. Bioorg Med Chem Lett. 2009 Jan 15;19(2):474-6. doi: 10.1016/j.bmcl.2008.11.044. Epub 2008 Nov 18. Bioorg Med Chem Lett. 2009. PMID: 19081250 Free PMC article.

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