Hassan AHE - Search Results

1

First-in-class DAPK1/CSF1R dual inhibitors: Discovery of 3,5-dimethoxy-N-(4-(4-methoxyphenoxy)-2-((6-morpholinopyridin-3-yl)amino)pyrimidin-5-yl)benzamide as a potential anti-tauopathies agent.

Farag AK, Hassan AHE, Jeong H, Kwon Y, Choi JG, Oh MS, Park KD, Kim YK, Roh EJ. Farag AK, et al. Among authors: hassan ahe. Eur J Med Chem. 2019 Jan 15;162:161-175. doi: 10.1016/j.ejmech.2018.10.057. Epub 2018 Nov 2. Eur J Med Chem. 2019. PMID: 30445265

2

Synthesis and biological evaluation of picolinamides and thiazole-2-carboxamides as mGluR5 (metabotropic glutamate receptor 5) antagonists.

Vu HN, Kim JY, Hassan AH, Choi K, Park JH, Park KD, Lee JK, Pae AN, Choo H, Min SJ, Cho YS. Vu HN, et al. Bioorg Med Chem Lett. 2016 Jan 1;26(1):140-4. doi: 10.1016/j.bmcl.2015.11.012. Epub 2015 Nov 5. Bioorg Med Chem Lett. 2016. PMID: 26598462

3

Discovery of 1-(3-(benzyloxy)pyridin-2-yl)-3-(2-(piperazin-1-yl)ethyl)urea: A new modulator for amyloid beta-induced mitochondrial dysfunction.

Elkamhawy A, Park JE, Hassan AHE, Ra H, Pae AN, Lee J, Park BG, Moon B, Park HM, Roh EJ. Elkamhawy A, et al. Among authors: hassan ahe. Eur J Med Chem. 2017 Mar 10;128:56-69. doi: 10.1016/j.ejmech.2016.12.057. Epub 2016 Dec 29. Eur J Med Chem. 2017. PMID: 28152427

4

Design, synthesis, biological evaluation and molecular modelling of 2-(2-aryloxyphenyl)-1,4-dihydroisoquinolin-3(2H)-ones: A novel class of TSPO ligands modulating amyloid-β-induced mPTP opening.

Elkamhawy A, Park JE, Hassan AHE, Pae AN, Lee J, Park BG, Paik S, Do J, Park JH, Park KD, Moon B, Park WK, Cho H, Jeong DY, Roh EJ. Elkamhawy A, et al. Among authors: hassan ahe. Eur J Pharm Sci. 2017 Jun 15;104:366-381. doi: 10.1016/j.ejps.2017.04.015. Epub 2017 Apr 21. Eur J Pharm Sci. 2017. PMID: 28435076

5

Synthesis and evaluation of new pyridyl/pyrazinyl thiourea derivatives: Neuroprotection against amyloid-β-induced toxicity.

Park JE, Elkamhawy A, Hassan AHE, Pae AN, Lee J, Paik S, Park BG, Roh EJ. Park JE, et al. Among authors: hassan ahe. Eur J Med Chem. 2017 Dec 1;141:322-334. doi: 10.1016/j.ejmech.2017.09.043. Epub 2017 Sep 22. Eur J Med Chem. 2017. PMID: 29031076

6

Hit discovery of 4-amino-N-(4-(3-(trifluoromethyl)phenoxy)pyrimidin-5-yl)benzamide: A novel EGFR inhibitor from a designed small library.

Elkamhawy A, Paik S, Hassan AHE, Lee YS, Roh EJ. Elkamhawy A, et al. Among authors: hassan ahe. Bioorg Chem. 2017 Dec;75:393-405. doi: 10.1016/j.bioorg.2017.10.009. Epub 2017 Nov 5. Bioorg Chem. 2017. PMID: 29102722

7

Synthesis and evaluation of 2-(3-arylureido)pyridines and 2-(3-arylureido)pyrazines as potential modulators of Aβ-induced mitochondrial dysfunction in Alzheimer's disease.

Elkamhawy A, Park JE, Hassan AHE, Pae AN, Lee J, Park BG, Roh EJ. Elkamhawy A, et al. Among authors: hassan ahe. Eur J Med Chem. 2018 Jan 20;144:529-543. doi: 10.1016/j.ejmech.2017.12.045. Epub 2017 Dec 14. Eur J Med Chem. 2018. PMID: 29288949

8

Repositioning of the antipsychotic trifluoperazine: Synthesis, biological evaluation and in silico study of trifluoperazine analogs as anti-glioblastoma agents.

Kang S, Lee JM, Jeon B, Elkamhawy A, Paik S, Hong J, Oh SJ, Paek SH, Lee CJ, Hassan AHE, Kang SS, Roh EJ. Kang S, et al. Among authors: hassan ahe. Eur J Med Chem. 2018 May 10;151:186-198. doi: 10.1016/j.ejmech.2018.03.055. Epub 2018 Mar 23. Eur J Med Chem. 2018. PMID: 29614416

9

Pyrazinyl ureas revisited: 1-(3-(Benzyloxy)pyrazin-2-yl)-3-(3,4-dichlorophenyl)urea, a new blocker of Aβ-induced mPTP opening for Alzheimer's disease.

Elkamhawy A, Park JE, Hassan AHE, Pae AN, Lee J, Paik S, Park BG, Roh EJ. Elkamhawy A, et al. Among authors: hassan ahe. Eur J Med Chem. 2018 Sep 5;157:268-278. doi: 10.1016/j.ejmech.2018.07.068. Epub 2018 Jul 31. Eur J Med Chem. 2018. PMID: 30098482

10

Design, synthesis and biological evaluation of novel thiazolidinedione derivatives as irreversible allosteric IKK-β modulators.

Elkamhawy A, Kim NY, Hassan AHE, Park JE, Yang JE, Oh KS, Lee BH, Lee MY, Shin KJ, Lee KT, Hur W, Roh EJ. Elkamhawy A, et al. Among authors: hassan ahe. Eur J Med Chem. 2018 Sep 5;157:691-704. doi: 10.1016/j.ejmech.2018.08.020. Epub 2018 Aug 8. Eur J Med Chem. 2018. PMID: 30130718

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