Carlino L - Search Results

1

Structure-Activity Relationships of Hexahydrocyclopenta[c]quinoline Derivatives as Allosteric Inhibitors of CDK2 and EGFR.

Carlino L, Christodoulou MS, Restelli V, Caporuscio F, Foschi F, Semrau MS, Costanzi E, Tinivella A, Pinzi L, Lo Presti L, Battistutta R, Storici P, Broggini M, Passarella D, Rastelli G. Carlino L, et al. ChemMedChem. 2018 Dec 20;13(24):2627-2634. doi: 10.1002/cmdc.201800687. Epub 2018 Nov 20. ChemMedChem. 2018. PMID: 30457710 Free article.

2

Molecular Dynamics Simulations and Classical Multidimensional Scaling Unveil New Metastable States in the Conformational Landscape of CDK2.

Pisani P, Caporuscio F, Carlino L, Rastelli G. Pisani P, et al. Among authors: carlino l. PLoS One. 2016 Apr 21;11(4):e0154066. doi: 10.1371/journal.pone.0154066. eCollection 2016. PLoS One. 2016. PMID: 27100206 Free PMC article.

3

Probing an Allosteric Pocket of CDK2 with Small Molecules.

Christodoulou MS, Caporuscio F, Restelli V, Carlino L, Cannazza G, Costanzi E, Citti C, Lo Presti L, Pisani P, Battistutta R, Broggini M, Passarella D, Rastelli G. Christodoulou MS, et al. Among authors: carlino l. ChemMedChem. 2017 Jan 5;12(1):33-41. doi: 10.1002/cmdc.201600474. Epub 2016 Dec 19. ChemMedChem. 2017. PMID: 27860401

4

Dual Kinase-Bromodomain Inhibitors in Anticancer Drug Discovery: A Structural and Pharmacological Perspective.

Carlino L, Rastelli G. Carlino L, et al. J Med Chem. 2016 Oct 27;59(20):9305-9320. doi: 10.1021/acs.jmedchem.6b00438. Epub 2016 Sep 7. J Med Chem. 2016. PMID: 27559828 Review.

5

Identification and Structure-Activity Relationship Studies of Small-Molecule Inhibitors of the Methyllysine Reader Protein Spindlin1.

Robaa D, Wagner T, Luise C, Carlino L, McMillan J, Flaig R, Schüle R, Jung M, Sippl W. Robaa D, et al. Among authors: carlino l. ChemMedChem. 2016 Oct 19;11(20):2327-2338. doi: 10.1002/cmdc.201600362. Epub 2016 Sep 16. ChemMedChem. 2016. PMID: 27634332

6

Structural basis of the effect of activating mutations on the EGF receptor.

Galdadas I, Carlino L, Ward RA, Hughes SJ, Haider S, Gervasio FL. Galdadas I, et al. Among authors: carlino l. Elife. 2021 Jul 28;10:e65824. doi: 10.7554/eLife.65824. Elife. 2021. PMID: 34319231 Free PMC article.

7

Computer- and structure-based lead design for epigenetic targets.

Heinke R, Carlino L, Kannan S, Jung M, Sippl W. Heinke R, et al. Among authors: carlino l. Bioorg Med Chem. 2011 Jun 15;19(12):3605-15. doi: 10.1016/j.bmc.2011.01.029. Epub 2011 Jan 22. Bioorg Med Chem. 2011. PMID: 21316248

8

Nonpeptidic propargylamines as inhibitors of lysine specific demethylase 1 (LSD1) with cellular activity.

Schmitt ML, Hauser AT, Carlino L, Pippel M, Schulz-Fincke J, Metzger E, Willmann D, Yiu T, Barton M, Schüle R, Sippl W, Jung M. Schmitt ML, et al. Among authors: carlino l. J Med Chem. 2013 Sep 26;56(18):7334-42. doi: 10.1021/jm400792m. Epub 2013 Sep 5. J Med Chem. 2013. PMID: 24007511 Free PMC article.

9

Heterogeneous Antibody-Based Activity Assay for Lysine Specific Demethylase 1 (LSD1) on a Histone Peptide Substrate.

Schmitt ML, Ladwein KI, Carlino L, Schulz-Fincke J, Willmann D, Metzger E, Schilcher P, Imhof A, Schüle R, Sippl W, Jung M. Schmitt ML, et al. Among authors: carlino l. J Biomol Screen. 2014 Jul;19(6):973-8. doi: 10.1177/1087057114529156. Epub 2014 Mar 31. J Biomol Screen. 2014. PMID: 24687155

10

The role of histone demethylases in cancer therapy.

Hoffmann I, Roatsch M, Schmitt ML, Carlino L, Pippel M, Sippl W, Jung M. Hoffmann I, et al. Among authors: carlino l. Mol Oncol. 2012 Dec;6(6):683-703. doi: 10.1016/j.molonc.2012.07.004. Epub 2012 Aug 7. Mol Oncol. 2012. PMID: 22902149 Free PMC article. Review.

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