Hassan AHE - Search Results

1

EGFR inhibitors from cancer to inflammation: Discovery of 4-fluoro-N-(4-(3-(trifluoromethyl)phenoxy)pyrimidin-5-yl)benzamide as a novel anti-inflammatory EGFR inhibitor.

Elkamhawy A, Hassan AHE, Paik S, Sup Lee Y, Lee HH, Shin JS, Lee KT, Roh EJ. Elkamhawy A, et al. Among authors: hassan ahe. Bioorg Chem. 2019 May;86:112-118. doi: 10.1016/j.bioorg.2019.01.017. Epub 2019 Jan 12. Bioorg Chem. 2019. PMID: 30685642

2

Synthesis and biological evaluation of picolinamides and thiazole-2-carboxamides as mGluR5 (metabotropic glutamate receptor 5) antagonists.

Vu HN, Kim JY, Hassan AH, Choi K, Park JH, Park KD, Lee JK, Pae AN, Choo H, Min SJ, Cho YS. Vu HN, et al. Bioorg Med Chem Lett. 2016 Jan 1;26(1):140-4. doi: 10.1016/j.bmcl.2015.11.012. Epub 2015 Nov 5. Bioorg Med Chem Lett. 2016. PMID: 26598462

3

Discovery of 1-(3-(benzyloxy)pyridin-2-yl)-3-(2-(piperazin-1-yl)ethyl)urea: A new modulator for amyloid beta-induced mitochondrial dysfunction.

Elkamhawy A, Park JE, Hassan AHE, Ra H, Pae AN, Lee J, Park BG, Moon B, Park HM, Roh EJ. Elkamhawy A, et al. Among authors: hassan ahe. Eur J Med Chem. 2017 Mar 10;128:56-69. doi: 10.1016/j.ejmech.2016.12.057. Epub 2016 Dec 29. Eur J Med Chem. 2017. PMID: 28152427

4

Design, synthesis, biological evaluation and molecular modelling of 2-(2-aryloxyphenyl)-1,4-dihydroisoquinolin-3(2H)-ones: A novel class of TSPO ligands modulating amyloid-β-induced mPTP opening.

Elkamhawy A, Park JE, Hassan AHE, Pae AN, Lee J, Park BG, Paik S, Do J, Park JH, Park KD, Moon B, Park WK, Cho H, Jeong DY, Roh EJ. Elkamhawy A, et al. Among authors: hassan ahe. Eur J Pharm Sci. 2017 Jun 15;104:366-381. doi: 10.1016/j.ejps.2017.04.015. Epub 2017 Apr 21. Eur J Pharm Sci. 2017. PMID: 28435076

5

Synthesis and evaluation of new pyridyl/pyrazinyl thiourea derivatives: Neuroprotection against amyloid-β-induced toxicity.

Park JE, Elkamhawy A, Hassan AHE, Pae AN, Lee J, Paik S, Park BG, Roh EJ. Park JE, et al. Among authors: hassan ahe. Eur J Med Chem. 2017 Dec 1;141:322-334. doi: 10.1016/j.ejmech.2017.09.043. Epub 2017 Sep 22. Eur J Med Chem. 2017. PMID: 29031076

6

Design, synthesis and evaluation of alkylphosphocholine-gefitinib conjugates as multitarget anticancer agents.

Alam MM, Hassan AHE, Kwon YH, Lee HJ, Kim NY, Min KH, Lee SY, Kim DH, Lee YS. Alam MM, et al. Among authors: hassan ahe. Arch Pharm Res. 2018 Jan;41(1):35-45. doi: 10.1007/s12272-017-0977-z. Epub 2017 Nov 1. Arch Pharm Res. 2018. PMID: 29094267

7

Hit discovery of 4-amino-N-(4-(3-(trifluoromethyl)phenoxy)pyrimidin-5-yl)benzamide: A novel EGFR inhibitor from a designed small library.

Elkamhawy A, Paik S, Hassan AHE, Lee YS, Roh EJ. Elkamhawy A, et al. Among authors: hassan ahe. Bioorg Chem. 2017 Dec;75:393-405. doi: 10.1016/j.bioorg.2017.10.009. Epub 2017 Nov 5. Bioorg Chem. 2017. PMID: 29102722

8

Synthesis and evaluation of 2-(3-arylureido)pyridines and 2-(3-arylureido)pyrazines as potential modulators of Aβ-induced mitochondrial dysfunction in Alzheimer's disease.

Elkamhawy A, Park JE, Hassan AHE, Pae AN, Lee J, Park BG, Roh EJ. Elkamhawy A, et al. Among authors: hassan ahe. Eur J Med Chem. 2018 Jan 20;144:529-543. doi: 10.1016/j.ejmech.2017.12.045. Epub 2017 Dec 14. Eur J Med Chem. 2018. PMID: 29288949

9

Repositioning of the antipsychotic trifluoperazine: Synthesis, biological evaluation and in silico study of trifluoperazine analogs as anti-glioblastoma agents.

Kang S, Lee JM, Jeon B, Elkamhawy A, Paik S, Hong J, Oh SJ, Paek SH, Lee CJ, Hassan AHE, Kang SS, Roh EJ. Kang S, et al. Among authors: hassan ahe. Eur J Med Chem. 2018 May 10;151:186-198. doi: 10.1016/j.ejmech.2018.03.055. Epub 2018 Mar 23. Eur J Med Chem. 2018. PMID: 29614416

10

Pyrazinyl ureas revisited: 1-(3-(Benzyloxy)pyrazin-2-yl)-3-(3,4-dichlorophenyl)urea, a new blocker of Aβ-induced mPTP opening for Alzheimer's disease.

Elkamhawy A, Park JE, Hassan AHE, Pae AN, Lee J, Paik S, Park BG, Roh EJ. Elkamhawy A, et al. Among authors: hassan ahe. Eur J Med Chem. 2018 Sep 5;157:268-278. doi: 10.1016/j.ejmech.2018.07.068. Epub 2018 Jul 31. Eur J Med Chem. 2018. PMID: 30098482

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