Silvestri R - Search Results

1

Structure-activity relationship studies and in vitro and in vivo anticancer activity of novel 3-aroyl-1,4-diarylpyrroles against solid tumors and hematological malignancies.

Puxeddu M, Shen H, Bai R, Coluccia A, Nalli M, Mazzoccoli C, Da Pozzo E, Cavallini C, Martini C, Orlando V, Biagioni S, Mazzoni C, Coluccia AML, Hamel E, Liu T, Silvestri R, La Regina G. Puxeddu M, et al. Among authors: silvestri r. Eur J Med Chem. 2020 Jan 1;185:111828. doi: 10.1016/j.ejmech.2019.111828. Epub 2019 Nov 2. Eur J Med Chem. 2020. PMID: 31727471

2

1-[2-(Diphenylmethoxy)ethyl]-2-methyl-5-nitroimidazole: a potent lead for the design of novel NNRTIs.

Silvestri R, Artico M, Massa S, Marceddu T, De Montis F, La Colla P. Silvestri R, et al. Bioorg Med Chem Lett. 2000 Feb 7;10(3):253-6. doi: 10.1016/s0960-894x(99)00664-2. Bioorg Med Chem Lett. 2000. PMID: 10698447

3

Structure-based design, synthesis, and biological evaluation of novel pyrrolyl aryl sulfones: HIV-1 non-nucleoside reverse transcriptase inhibitors active at nanomolar concentrations.

Artico M, Silvestri R, Pagnozzi E, Bruno B, Novellino E, Greco G, Massa S, Ettorre A, Loi AG, Scintu F, La Colla P. Artico M, et al. Among authors: silvestri r. J Med Chem. 2000 May 4;43(9):1886-91. doi: 10.1021/jm9901125. J Med Chem. 2000. PMID: 10794705

4

Synthesis, biological evaluation, and binding mode of novel 1-[2-(diarylmethoxy)ethyl]-2-methyl-5-nitroimidazoles targeted at the HIV-1 reverse transcriptase.

Silvestri R, Artico M, De Martino G, Ragno R, Massa S, Loddo R, Murgioni C, Loi AG, La Colla P, Pani A. Silvestri R, et al. J Med Chem. 2002 Apr 11;45(8):1567-76. doi: 10.1021/jm010904a. J Med Chem. 2002. PMID: 11931611

5

Simple, potent, and selective pyrrole inhibitors of monoamine oxidase types A and B.

Silvestri R, La Regina G, De Martino G, Artico M, Befani O, Palumbo M, Agostinelli E, Turini P. Silvestri R, et al. J Med Chem. 2003 Mar 13;46(6):917-20. doi: 10.1021/jm0256124. J Med Chem. 2003. PMID: 12620068

6

Novel indolyl aryl sulfones active against HIV-1 carrying NNRTI resistance mutations: synthesis and SAR studies.

Silvestri R, De Martino G, La Regina G, Artico M, Massa S, Vargiu L, Mura M, Loi AG, Marceddu T, La Colla P. Silvestri R, et al. J Med Chem. 2003 Jun 5;46(12):2482-93. doi: 10.1021/jm0211063. J Med Chem. 2003. PMID: 12773052

7

Anti-HIV-1 activity of pyrryl aryl sulfone (PAS) derivatives: synthesis and SAR studies of novel esters and amides at the position 2 of the pyrrole nucleus.

Silvestri R, Artico M, La Regina G, De Martino G, La Colla M, Loddo R, La Colla P. Silvestri R, et al. Farmaco. 2004 Mar;59(3):201-10. doi: 10.1016/j.farmac.2003.11.004. Farmaco. 2004. PMID: 14987983

8

Simple, short peptide derivatives of a sulfonylindolecarboxamide (L-737,126) active in vitro against HIV-1 wild type and variants carrying non-nucleoside reverse transcriptase inhibitor resistance mutations.

Silvestri R, Artico M, De Martino G, La Regina G, Loddo R, La Colla M, Mura M, La Colla P. Silvestri R, et al. J Med Chem. 2004 Jul 15;47(15):3892-6. doi: 10.1021/jm031147e. J Med Chem. 2004. PMID: 15239667

9

Imidazole analogues of fluoxetine, a novel class of anti-Candida agents.

Silvestri R, Artico M, La Regina G, Di Pasquali A, De Martino G, D'Auria FD, Nencioni L, Palamara AT. Silvestri R, et al. J Med Chem. 2004 Jul 29;47(16):3924-6. doi: 10.1021/jm049856v. J Med Chem. 2004. PMID: 15267229

10

Arylthioindoles, potent inhibitors of tubulin polymerization.

De Martino G, La Regina G, Coluccia A, Edler MC, Barbera MC, Brancale A, Wilcox E, Hamel E, Artico M, Silvestri R. De Martino G, et al. Among authors: silvestri r. J Med Chem. 2004 Dec 2;47(25):6120-3. doi: 10.1021/jm049360d. J Med Chem. 2004. PMID: 15566282

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