Aso K - Search Results

1

Pharmacological evaluation of a novel corticotropin-releasing factor 1 receptor antagonist T-3047928 in stress-induced animal models in a comparison with alosetron.

Itomi Y, Tanaka T, Matsushita K, Kawamura T, Kojima T, Aso K, Matsumoto-Okano S, Tsukimi Y. Itomi Y, et al. Among authors: aso k. Neurogastroenterol Motil. 2020 May;32(5):e13795. doi: 10.1111/nmo.13795. Epub 2020 Jan 22. Neurogastroenterol Motil. 2020. PMID: 31970891

2

Discovery of 1,2,3,4-tetrahydropyrimido[1,2-a]benzimidazoles as novel class of corticotropin releasing factor 1 receptor antagonists.

Kojima T, Mochizuki M, Takai T, Hoashi Y, Morimoto S, Seto M, Nakamura M, Kobayashi K, Sako Y, Tanaka M, Kanzaki N, Kosugi Y, Yano T, Aso K. Kojima T, et al. Among authors: aso k. Bioorg Med Chem. 2018 May 15;26(9):2229-2250. doi: 10.1016/j.bmc.2018.01.020. Epub 2018 Feb 8. Bioorg Med Chem. 2018. PMID: 29459145

3

Discovery of 4-chloro-2-(2,4-dichloro-6-methylphenoxy)-1-methyl-7-(pentan-3-yl)-1H-benzimidazole, a novel CRF₁ receptor antagonist.

Mochizuki M, Kojima T, Kobayashi K, Kotani E, Ishichi Y, Kanzaki N, Nakagawa H, Okuda T, Kosugi Y, Yano T, Sako Y, Tanaka M, Aso K. Mochizuki M, et al. Among authors: aso k. Bioorg Med Chem. 2017 Mar 1;25(5):1556-1570. doi: 10.1016/j.bmc.2016.11.011. Epub 2016 Nov 8. Bioorg Med Chem. 2017. PMID: 28174066

4

Characterization of CRF₁ receptor antagonists with differential peripheral vs central actions in CRF challenge in rats.

Tanaka M, Tomimatsu Y, Sakimura K, Ootani Y, Sako Y, Kojima T, Aso K, Yano T, Hirai K. Tanaka M, et al. Among authors: aso k. Peptides. 2017 Sep;95:40-50. doi: 10.1016/j.peptides.2017.06.009. Epub 2017 Jul 6. Peptides. 2017. PMID: 28689880

5

Design and Synthesis of Benzimidazoles As Novel Corticotropin-Releasing Factor 1 Receptor Antagonists.

Mochizuki M, Kori M, Kobayashi K, Yano T, Sako Y, Tanaka M, Kanzaki N, Gyorkos AC, Corrette CP, Cho SY, Pratt SA, Aso K. Mochizuki M, et al. Among authors: aso k. J Med Chem. 2016 Mar 24;59(6):2551-66. doi: 10.1021/acs.jmedchem.5b01715. Epub 2016 Mar 7. J Med Chem. 2016. PMID: 26901666

6

Discovery of a 7-arylaminobenzimidazole series as novel CRF1 receptor antagonists.

Mochizuki M, Kori M, Kono M, Yano T, Sako Y, Tanaka M, Kanzaki N, Gyorkos AC, Corrette CP, Aso K. Mochizuki M, et al. Among authors: aso k. Bioorg Med Chem. 2016 Oct 1;24(19):4675-4691. doi: 10.1016/j.bmc.2016.08.005. Epub 2016 Aug 4. Bioorg Med Chem. 2016. PMID: 27567079

7

Discovery of pyrrolo[2,3-d]pyrimidin-4-ones as corticotropin-releasing factor 1 receptor antagonists with a carbonyl-based hydrogen bonding acceptor.

Aso K, Kobayashi K, Mochizuki M, Kanzaki N, Sako Y, Yano T. Aso K, et al. Bioorg Med Chem Lett. 2011 Apr 15;21(8):2365-71. doi: 10.1016/j.bmcl.2011.02.086. Epub 2011 Feb 26. Bioorg Med Chem Lett. 2011. PMID: 21414781

8

Design, synthesis, and pharmacological evaluation of 4-azolyl-benzamide derivatives as novel GPR52 agonists.

Tokumaru K, Ito Y, Nomura I, Nakahata T, Shimizu Y, Kurimoto E, Aoyama K, Aso K. Tokumaru K, et al. Among authors: aso k. Bioorg Med Chem. 2017 Jun 15;25(12):3098-3115. doi: 10.1016/j.bmc.2017.03.064. Epub 2017 Apr 1. Bioorg Med Chem. 2017. PMID: 28433511

9

Identification of a novel series of potent and selective CCR6 inhibitors as biological probes.

Tawaraishi T, Sakauchi N, Hidaka K, Yoshikawa K, Okui T, Kuno H, Chisaki I, Aso K. Tawaraishi T, et al. Among authors: aso k. Bioorg Med Chem Lett. 2018 Oct 1;28(18):3067-3072. doi: 10.1016/j.bmcl.2018.07.042. Epub 2018 Jul 30. Bioorg Med Chem Lett. 2018. PMID: 30098865

10

Design and synthesis of 1-(1-benzothiophen-7-yl)-1H-pyrazole, a novel series of G protein-coupled receptor 52 (GPR52) agonists.

Nakahata T, Tokumaru K, Ito Y, Ishii N, Setoh M, Shimizu Y, Harasawa T, Aoyama K, Hamada T, Kori M, Aso K. Nakahata T, et al. Among authors: aso k. Bioorg Med Chem. 2018 May 1;26(8):1598-1608. doi: 10.1016/j.bmc.2018.02.005. Epub 2018 Feb 10. Bioorg Med Chem. 2018. PMID: 29478803

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