Deprez B - Search Results

1

Fragment-Based Optimized EthR Inhibitors with in Vivo Ethionamide Boosting Activity.

Villemagne B, Machelart A, Tran NC, Flipo M, Moune M, Leroux F, Piveteau C, Wohlkönig A, Wintjens R, Li X, Gref R, Brodin P, Deprez B, Baulard AR, Willand N. Villemagne B, et al. Among authors: deprez b. ACS Infect Dis. 2020 Mar 13;6(3):366-378. doi: 10.1021/acsinfecdis.9b00277. Epub 2020 Mar 2. ACS Infect Dis. 2020. PMID: 32011115

2

A library of novel hydroxamic acids targeting the metallo-protease family: design, parallel synthesis and screening.

Flipo M, Beghyn T, Charton J, Leroux VA, Deprez BP, Deprez-Poulain RF. Flipo M, et al. Bioorg Med Chem. 2007 Jan 1;15(1):63-76. doi: 10.1016/j.bmc.2006.10.010. Epub 2006 Oct 12. Bioorg Med Chem. 2007. PMID: 17070058

3

Novel selective inhibitors of the zinc plasmodial aminopeptidase PfA-M1 as potential antimalarial agents.

Flipo M, Beghyn T, Leroux V, Florent I, Deprez BP, Deprez-Poulain RF. Flipo M, et al. J Med Chem. 2007 Mar 22;50(6):1322-34. doi: 10.1021/jm061169b. Epub 2007 Feb 28. J Med Chem. 2007. PMID: 17326615

4

Natural compounds: leads or ideas? Bioinspired molecules for drug discovery.

Beghyn T, Deprez-Poulain R, Willand N, Folleas B, Deprez B. Beghyn T, et al. Among authors: deprez poulain r, deprez b. Chem Biol Drug Des. 2008 Jul;72(1):3-15. doi: 10.1111/j.1747-0285.2008.00673.x. Epub 2008 Jun 11. Chem Biol Drug Des. 2008. PMID: 18554253

5

Synthesis of a 200-member library of squaric acid N-hydroxylamide amides.

Charton J, Leroux F, Delaroche S, Landry V, Déprez BP, Déprez-Poulain RF. Charton J, et al. Bioorg Med Chem Lett. 2008 Sep 15;18(18):4968-71. doi: 10.1016/j.bmcl.2008.08.025. Epub 2008 Aug 14. Bioorg Med Chem Lett. 2008. PMID: 18760922

6

Synthetic EthR inhibitors boost antituberculous activity of ethionamide.

Willand N, Dirié B, Carette X, Bifani P, Singhal A, Desroses M, Leroux F, Willery E, Mathys V, Déprez-Poulain R, Delcroix G, Frénois F, Aumercier M, Locht C, Villeret V, Déprez B, Baulard AR. Willand N, et al. Among authors: deprez poulain r, deprez b. Nat Med. 2009 May;15(5):537-44. doi: 10.1038/nm.1950. Epub 2009 May 3. Nat Med. 2009. PMID: 19412174

7

Hydroxamates: relationships between structure and plasma stability.

Flipo M, Charton J, Hocine A, Dassonneville S, Deprez B, Deprez-Poulain R. Flipo M, et al. Among authors: deprez poulain r, deprez b. J Med Chem. 2009 Nov 12;52(21):6790-802. doi: 10.1021/jm900648x. J Med Chem. 2009. PMID: 19821586

8

Designing focused chemical libraries enriched in protein-protein interaction inhibitors using machine-learning methods.

Reynès C, Host H, Camproux AC, Laconde G, Leroux F, Mazars A, Deprez B, Fahraeus R, Villoutreix BO, Sperandio O. Reynès C, et al. Among authors: deprez b. PLoS Comput Biol. 2010 Mar 5;6(3):e1000695. doi: 10.1371/journal.pcbi.1000695. PLoS Comput Biol. 2010. PMID: 20221258 Free PMC article.

9

Exploring drug target flexibility using in situ click chemistry: application to a mycobacterial transcriptional regulator.

Willand N, Desroses M, Toto P, Dirié B, Lens Z, Villeret V, Rucktooa P, Locht C, Baulard A, Deprez B. Willand N, et al. Among authors: deprez b. ACS Chem Biol. 2010 Nov 19;5(11):1007-13. doi: 10.1021/cb100177g. ACS Chem Biol. 2010. PMID: 20704273

10

New non-hydroxamic ADAMTS-5 inhibitors based on the 1,2,4-triazole-3-thiol scaffold.

Maingot L, Leroux F, Landry V, Dumont J, Nagase H, Villoutreix B, Sperandio O, Deprez-Poulain R, Deprez B. Maingot L, et al. Among authors: deprez poulain r, deprez b. Bioorg Med Chem Lett. 2010 Nov 1;20(21):6213-6. doi: 10.1016/j.bmcl.2010.08.108. Epub 2010 Aug 27. Bioorg Med Chem Lett. 2010. PMID: 20846863

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