Haupenthal J - Search Results

1

Rapid Discovery of Aspartyl Protease Inhibitors Using an Anchoring Approach.

Konstantinidou M, Magari F, Sutanto F, Haupenthal J, Jumde VR, Ünver MY, Heine A, Camacho CJ, Hirsch AKH, Klebe G, Dömling A. Konstantinidou M, et al. Among authors: haupenthal j. ChemMedChem. 2020 Apr 20;15(8):680-684. doi: 10.1002/cmdc.202000024. Epub 2020 Mar 18. ChemMedChem. 2020. PMID: 32187447 Free PMC article.

2

Discovery of novel bacterial RNA polymerase inhibitors: pharmacophore-based virtual screening and hit optimization.

Hinsberger S, Hüsecken K, Groh M, Negri M, Haupenthal J, Hartmann RW. Hinsberger S, et al. Among authors: haupenthal j. J Med Chem. 2013 Nov 14;56(21):8332-8. doi: 10.1021/jm400485e. Epub 2013 Oct 31. J Med Chem. 2013. PMID: 24112046

3

Discovery and Structure-Based Optimization of 2-Ureidothiophene-3-carboxylic Acids as Dual Bacterial RNA Polymerase and Viral Reverse Transcriptase Inhibitors.

Elgaher WA, Sharma KK, Haupenthal J, Saladini F, Pires M, Real E, Mély Y, Hartmann RW. Elgaher WA, et al. Among authors: haupenthal j. J Med Chem. 2016 Aug 11;59(15):7212-22. doi: 10.1021/acs.jmedchem.6b00730. Epub 2016 Jul 7. J Med Chem. 2016. PMID: 27339173

4

Biophysical Screening of a Focused Library for the Discovery of CYP121 Inhibitors as Novel Antimycobacterials.

Brengel C, Thomann A, Schifrin A, Allegretta G, Kamal AAM, Haupenthal J, Schnorr I, Cho SH, Franzblau SG, Empting M, Eberhard J, Hartmann RW. Brengel C, et al. Among authors: haupenthal j. ChemMedChem. 2017 Oct 9;12(19):1616-1626. doi: 10.1002/cmdc.201700363. Epub 2017 Sep 26. ChemMedChem. 2017. PMID: 28815923 Free article.

5

Spray-drying of inhalable, multifunctional formulations for the treatment of biofilms formed in cystic fibrosis.

Lababidi N, Ofosu Kissi E, Elgaher WAM, Sigal V, Haupenthal J, Schwarz BC, Hirsch AKH, Rades T, Schneider M. Lababidi N, et al. Among authors: haupenthal j. J Control Release. 2019 Nov 28;314:62-71. doi: 10.1016/j.jconrel.2019.10.038. Epub 2019 Oct 22. J Control Release. 2019. PMID: 31654686

6

From Wood to Tetrahydro-2-benzazepines in Three Waste-Free Steps: Modular Synthesis of Biologically Active Lignin-Derived Scaffolds.

Elangovan S, Afanasenko A, Haupenthal J, Sun Z, Liu Y, Hirsch AKH, Barta K. Elangovan S, et al. Among authors: haupenthal j. ACS Cent Sci. 2019 Oct 23;5(10):1707-1716. doi: 10.1021/acscentsci.9b00781. Epub 2019 Oct 11. ACS Cent Sci. 2019. PMID: 31660439 Free PMC article.

7

N-Aryl-3-mercaptosuccinimides as Antivirulence Agents Targeting Pseudomonas aeruginosa Elastase and Clostridium Collagenases.

Konstantinović J, Yahiaoui S, Alhayek A, Haupenthal J, Schönauer E, Andreas A, Kany AM, Müller R, Koehnke J, Berger FK, Bischoff M, Hartmann RW, Brandstetter H, Hirsch AKH. Konstantinović J, et al. Among authors: haupenthal j. J Med Chem. 2020 Aug 13;63(15):8359-8368. doi: 10.1021/acs.jmedchem.0c00584. Epub 2020 Jun 17. J Med Chem. 2020. PMID: 32470298 Free PMC article.

8

Evaluation of Bacterial RNA Polymerase Inhibitors in a Staphylococcus aureus-Based Wound Infection Model in SKH1 Mice.

Haupenthal J, Kautz Y, Elgaher WAM, Pätzold L, Röhrig T, Laschke MW, Tschernig T, Hirsch AKH, Molodtsov V, Murakami KS, Hartmann RW, Bischoff M. Haupenthal J, et al. ACS Infect Dis. 2020 Oct 9;6(10):2573-2581. doi: 10.1021/acsinfecdis.0c00034. Epub 2020 Sep 21. ACS Infect Dis. 2020. PMID: 32886885 Free PMC article.

9

Phosphonate as a Stable Zinc-Binding Group for "Pathoblocker" Inhibitors of Clostridial Collagenase H (ColH).

Voos K, Schönauer E, Alhayek A, Haupenthal J, Andreas A, Müller R, Hartmann RW, Brandstetter H, Hirsch AKH, Ducho C. Voos K, et al. Among authors: haupenthal j. ChemMedChem. 2021 Apr 20;16(8):1257-1267. doi: 10.1002/cmdc.202000994. Epub 2021 Mar 16. ChemMedChem. 2021. PMID: 33506625 Free PMC article.

10

Assessment of the rules related to gaining activity against Gram-negative bacteria.

Ropponen HK, Diamanti E, Siemens A, Illarionov B, Haupenthal J, Fischer M, Rottmann M, Witschel M, Hirsch AKH. Ropponen HK, et al. Among authors: haupenthal j. RSC Med Chem. 2021 Mar 3;12(4):593-601. doi: 10.1039/d0md00409j. eCollection 2021 Apr 28. RSC Med Chem. 2021. PMID: 34046630 Free PMC article.

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