D'hooghe M - Search Results

1

Synthesis of Novel Nitroxoline Analogs with Potent Cathepsin B Exopeptidase Inhibitory Activity.

Van de Walle T, Briand M, Mitrović A, Sosič I, Gobec S, Kos J, Persoons L, Daelemans D, De Jonghe S, Ubiparip Z, Desmet T, Van Hecke K, Mangelinckx S, D'hooghe M. Van de Walle T, et al. ChemMedChem. 2020 Dec 15;15(24):2477-2490. doi: 10.1002/cmdc.202000402. Epub 2020 Sep 21. ChemMedChem. 2020. PMID: 32744405

2

Synthesis of 1-arylmethyl-2-(cyanomethyl)aziridines and their ring transformation into methyl N-(2-cyanocyclopropyl)benzimidates.

D'hooghe M, Mangelinckx S, Persyn E, Van Brabandt W, De Kimpe N. D'hooghe M, et al. J Org Chem. 2006 May 26;71(11):4232-6. doi: 10.1021/jo060425p. J Org Chem. 2006. PMID: 16709066

3

Biocatalytic production of novel glycolipids with cellodextrin phosphorylase.

Tran HG, Desmet T, Saerens K, Waegeman H, Vandekerckhove S, D'hooghe M, Van Bogaert I, Soetaert W. Tran HG, et al. Bioresour Technol. 2012 Jul;115:84-7. doi: 10.1016/j.biortech.2011.09.085. Epub 2011 Sep 25. Bioresour Technol. 2012. PMID: 22000964

4

Synthesis of 2-aminomethyl-4-phenyl-1-azabicyclo[2.2.1]heptanes via LiAlH₄-induced reductive cyclization of 2-(4-chloro-2-cyano-2-phenylbutyl)aziridines and evaluation of their antimalarial activity.

D'hooghe M, Vervisch K, Törnroos KW, Verhaeghe T, Desmet T, Lategan C, Smith PJ, Chibale K, De Kimpe N. D'hooghe M, et al. Bioorg Med Chem Lett. 2013 Mar 1;23(5):1507-10. doi: 10.1016/j.bmcl.2012.12.029. Epub 2012 Dec 20. Bioorg Med Chem Lett. 2013. PMID: 23347684

5

Potent and selective HDAC6 inhibitory activity of N-(4-hydroxycarbamoylbenzyl)-1,2,4,9-tetrahydro-3-thia-9-azafluorenes as novel sulfur analogues of Tubastatin A.

De Vreese R, Verhaeghe T, Desmet T, D'hooghe M. De Vreese R, et al. Chem Commun (Camb). 2013 May 8;49(36):3775-7. doi: 10.1039/c3cc41422a. Epub 2013 Mar 28. Chem Commun (Camb). 2013. PMID: 23538448

6

Evaluation of (4-aminobutyloxy)quinolines as a novel class of antifungal agents.

Vandekerckhove S, Tran HG, Desmet T, D'hooghe M. Vandekerckhove S, et al. Bioorg Med Chem Lett. 2013 Aug 15;23(16):4641-3. doi: 10.1016/j.bmcl.2013.06.014. Epub 2013 Jun 13. Bioorg Med Chem Lett. 2013. PMID: 23838261

7

Synthesis of halogenated 4-quinolones and evaluation of their antiplasmodial activity.

Vandekerckhove S, Desmet T, Tran HG, de Kock C, Smith PJ, Chibale K, D'hooghe M. Vandekerckhove S, et al. Bioorg Med Chem Lett. 2014 Feb 15;24(4):1214-7. doi: 10.1016/j.bmcl.2013.12.067. Epub 2014 Jan 4. Bioorg Med Chem Lett. 2014. PMID: 24468411

8

Selective synthesis of functionalized trifluoromethylated pyrrolidines, piperidines, and azepanes starting from 1-tosyl-2-(trifluoromethyl)aziridine.

Dolfen J, Kenis S, Van Hecke K, De Kimpe N, D'hooghe M. Dolfen J, et al. Chemistry. 2014 Aug 18;20(34):10650-3. doi: 10.1002/chem.201304759. Epub 2014 Feb 12. Chemistry. 2014. PMID: 24523231

9

Engineering the specificity of trehalose phosphorylase as a general strategy for the production of glycosyl phosphates.

Chen C, Van der Borght J, De Vreese R, D'hooghe M, Soetaert W, Desmet T. Chen C, et al. Chem Commun (Camb). 2014 Jul 25;50(58):7834-6. doi: 10.1039/c4cc02202e. Chem Commun (Camb). 2014. PMID: 24909572

10

Synthesis of functionalized 3-, 5-, 6- and 8-aminoquinolines via intermediate (3-pyrrolin-1-yl)- and (2-oxopyrrolidin-1-yl)quinolines and evaluation of their antiplasmodial and antifungal activity.

Vandekerckhove S, Van Herreweghe S, Willems J, Danneels B, Desmet T, de Kock C, Smith PJ, Chibale K, D'hooghe M. Vandekerckhove S, et al. Eur J Med Chem. 2015 Mar 6;92:91-102. doi: 10.1016/j.ejmech.2014.12.020. Epub 2014 Dec 12. Eur J Med Chem. 2015. PMID: 25544689

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