Bartz U - Search Results

1

N-Sulfonyl dipeptide nitriles as inhibitors of human cathepsin S: In silico design, synthesis and biochemical characterization.

Lemke C, Cianni L, Feldmann C, Gilberg E, Yin J, Dos Reis Rocho F, de Vita D, Bartz U, Bajorath J, Montanari CA, Gütschow M. Lemke C, et al. Among authors: bartz u. Bioorg Med Chem Lett. 2020 Sep 15;30(18):127420. doi: 10.1016/j.bmcl.2020.127420. Epub 2020 Jul 17. Bioorg Med Chem Lett. 2020. PMID: 32763808

2

3-Cyano-3-aza-β-amino Acid Derivatives as Inhibitors of Human Cysteine Cathepsins.

Schmitz J, Beckmann AM, Dudic A, Li T, Sellier R, Bartz U, Gütschow M. Schmitz J, et al. Among authors: bartz u. ACS Med Chem Lett. 2014 Aug 11;5(10):1076-81. doi: 10.1021/ml500238q. eCollection 2014 Oct 9. ACS Med Chem Lett. 2014. PMID: 25313316 Free PMC article.

3

Active Site Mapping of Human Cathepsin F with Dipeptide Nitrile Inhibitors.

Schmitz J, Furtmann N, Ponert M, Frizler M, Löser R, Bartz U, Bajorath J, Gütschow M. Schmitz J, et al. Among authors: bartz u. ChemMedChem. 2015 Aug;10(8):1365-77. doi: 10.1002/cmdc.201500151. Epub 2015 Jun 26. ChemMedChem. 2015. PMID: 26119278

4

Design, characterization and cellular uptake studies of fluorescence-labeled prototypic cathepsin inhibitors.

Kohl F, Schmitz J, Furtmann N, Schulz-Fincke AC, Mertens MD, Küppers J, Benkhoff M, Tobiasch E, Bartz U, Bajorath J, Stirnberg M, Gütschow M. Kohl F, et al. Among authors: bartz u. Org Biomol Chem. 2015 Nov 7;13(41):10310-23. doi: 10.1039/c5ob01613d. Org Biomol Chem. 2015. PMID: 26307943

5

Cathepsin B Inhibitors: Combining Dipeptide Nitriles with an Occluding Loop Recognition Element by Click Chemistry.

Schmitz J, Li T, Bartz U, Gütschow M. Schmitz J, et al. Among authors: bartz u. ACS Med Chem Lett. 2015 Dec 28;7(3):211-6. doi: 10.1021/acsmedchemlett.5b00474. eCollection 2016 Mar 10. ACS Med Chem Lett. 2015. PMID: 26985300 Free PMC article.

6

Synthesis and kinetic evaluation of ethyl acrylate and vinyl sulfone derived inhibitors for human cysteine cathepsins.

Breuer C, Lemke C, Schmitz J, Bartz U, Gütschow M. Breuer C, et al. Among authors: bartz u. Bioorg Med Chem Lett. 2018 Jun 15;28(11):2008-2012. doi: 10.1016/j.bmcl.2018.05.005. Epub 2018 May 4. Bioorg Med Chem Lett. 2018. PMID: 29748052

7

Cathepsin B: Active site mapping with peptidic substrates and inhibitors.

Schmitz J, Gilberg E, Löser R, Bajorath J, Bartz U, Gütschow M. Schmitz J, et al. Among authors: bartz u. Bioorg Med Chem. 2019 Jan 1;27(1):1-15. doi: 10.1016/j.bmc.2018.10.017. Epub 2018 Oct 19. Bioorg Med Chem. 2019. PMID: 30473362 Review.

8

Chromenones as Multineurotargeting Inhibitors of Human Enzymes.

Lemke C, Christmann J, Yin J, Alonso JM, Serrano E, Chioua M, Ismaili L, Martínez-Grau MA, Beadle CD, Vetman T, Dato FM, Bartz U, Elsinghorst PW, Pietsch M, Müller CE, Iriepa I, Wille T, Marco-Contelles J, Gütschow M. Lemke C, et al. Among authors: bartz u. ACS Omega. 2019 Dec 11;4(26):22161-22168. doi: 10.1021/acsomega.9b03409. eCollection 2019 Dec 24. ACS Omega. 2019. PMID: 31891098 Free PMC article.

9

Coumarin as a structural component of substrates and probes for serine and cysteine proteases.

Breidenbach J, Bartz U, Gütschow M. Breidenbach J, et al. Among authors: bartz u. Biochim Biophys Acta Proteins Proteom. 2020 Sep;1868(9):140445. doi: 10.1016/j.bbapap.2020.140445. Epub 2020 May 13. Biochim Biophys Acta Proteins Proteom. 2020. PMID: 32405284 Free PMC article. Review.

10

An Activity-Based Probe for Cathepsin K Imaging with Excellent Potency and Selectivity.

Lemke C, Benýšek J, Brajtenbach D, Breuer C, Jílková A, Horn M, Buša M, Ulrychová L, Illies A, Kubatzky KF, Bartz U, Mareš M, Gütschow M. Lemke C, et al. Among authors: bartz u. J Med Chem. 2021 Sep 23;64(18):13793-13806. doi: 10.1021/acs.jmedchem.1c01178. Epub 2021 Sep 2. J Med Chem. 2021. PMID: 34473502

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