Macchia M - Search Results

1

Design, synthesis and biological evaluation of second-generation benzoylpiperidine derivatives as reversible monoacylglycerol lipase (MAGL) inhibitors.

Granchi C, Bononi G, Ferrisi R, Gori E, Mantini G, Glasmacher S, Poli G, Palazzolo S, Caligiuri I, Rizzolio F, Canzonieri V, Perin T, Gertsch J, Sodi A, Giovannetti E, Macchia M, Minutolo F, Tuccinardi T, Chicca A. Granchi C, et al. Among authors: macchia m. Eur J Med Chem. 2021 Jan 1;209:112857. doi: 10.1016/j.ejmech.2020.112857. Epub 2020 Oct 7. Eur J Med Chem. 2021. PMID: 33045662

2

Conformationally restrained analogs of sympathomimetic catecholamines. Synthesis, conformational analysis, and adrenergic activity of isochroman derivatives.

Macchia B, Balsamo A, Breschi MC, Chiellini G, Lapucci A, Macchia M, Manera C, Martinelli A, Martini C, Scatizzi R, et al. Macchia B, et al. Among authors: macchia m. J Med Chem. 1993 Oct 15;36(21):3077-86. doi: 10.1021/jm00073a006. J Med Chem. 1993. PMID: 8230093

3

Geranylgeranyl diphosphate-based inhibitors of post-translational geranylgeranylation of cellular proteins.

Macchia M, Jannitti N, Gervasi G, Danesi R. Macchia M, et al. J Med Chem. 1996 Mar 29;39(7):1352-6. doi: 10.1021/jm960127s. J Med Chem. 1996. PMID: 8691464

4

Synthesis, inhibitory activity towards human leukocyte elastase and molecular modelling studies of 1-carbamoyl-4-methyleneaminoxyazetidinones.

Macchia B, Gentili D, Macchia M, Mamone F, Martinelli A, Orlandini E, Rossello A, Cercignani G, Pierotti R, Allegretti M, Asti C, Caselli G. Macchia B, et al. Among authors: macchia m. Eur J Med Chem. 2000 Jan;35(1):53-67. doi: 10.1016/s0223-5234(00)00111-2. Eur J Med Chem. 2000. PMID: 10733603

5

Synthesis and antiviral properties of 9-[(2-methyleneaminoxyethoxy)methyl]guanine derivatives as novel Acyclovir analogues.

Macchia M, Antonelli G, Calvani F, Di Bussolo V, Minutolo F, Orlandini E, Tesoro R, Turriziani O. Macchia M, et al. Farmaco. 2000 Feb;55(2):104-8. doi: 10.1016/s0014-827x(99)00129-9. Farmaco. 2000. PMID: 10782380

6

Synthesis and dopaminergic properties of the two enantiomers of 3-(3,4-dimethylphenyl)-1-propylpiperidine, a potent and selective dopamine D4 receptor ligand.

Macchia B, Cervetto L, Demontis GC, Domiano P, Longoni B, Macchia M, Minutolo F, Orlandini E, Ortore G, Papi C. Macchia B, et al. Among authors: macchia m. Bioorg Med Chem Lett. 2001 Jan 22;11(2):223-6. doi: 10.1016/s0960-894x(00)00633-8. Bioorg Med Chem Lett. 2001. PMID: 11206464

7

Synthesis and inhibitory activity towards human leukocyte elastase of new 7alpha-methoxy and 7alpha-chloro (2-acyloxymethyl) cephem derivatives.

Balsamo A, Cercignani G, Gentili D, Lapucci A, Macchia M, Orlandini E, Rapposelli S, Rossello A. Balsamo A, et al. Among authors: macchia m. Eur J Med Chem. 2001 Feb;36(2):185-93. doi: 10.1016/s0223-5234(01)01211-9. Eur J Med Chem. 2001. PMID: 11311749

8

Design, synthesis, and characterization of the antitumor activity of novel ceramide analogues.

Macchia M, Barontini S, Bertini S, Di Bussolo V, Fogli S, Giovannetti E, Grossi E, Minutolo F, Danesi R. Macchia M, et al. J Med Chem. 2001 Nov 8;44(23):3994-4000. doi: 10.1021/jm010947r. J Med Chem. 2001. PMID: 11689086

9

Salicylaldoxime moiety as a phenolic "A-Ring" substitute in estrogen receptor ligands.

Minutolo F, Bertini S, Papi C, Carlson KE, Katzenellenbogen JA, Macchia M. Minutolo F, et al. Among authors: macchia m. J Med Chem. 2001 Nov 22;44(24):4288-91. doi: 10.1021/jm010948j. J Med Chem. 2001. PMID: 11708930

10

7-Nitrobenzofurazan (NBD) derivatives of 5'-N-ethylcarboxamidoadenosine (NECA) as new fluorescent probes for human A(3) adenosine receptors.

Macchia M, Salvetti F, Bertini S, Di Bussolo V, Gattuso L, Gesi M, Hamdan M, Klotz KN, Laragione T, Lucacchini A, Minutolo F, Nencetti S, Papi C, Tuscano D, Martini C. Macchia M, et al. Bioorg Med Chem Lett. 2001 Dec 3;11(23):3023-6. doi: 10.1016/s0960-894x(01)00610-2. Bioorg Med Chem Lett. 2001. PMID: 11714602

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