Scilimati A - Search Results

1

An attempt to chemically state the cross-talk between monomers of COX homodimers by double/hybrid inhibitors mofezolac-spacer-mofezolac and mofezolac-spacer-arachidonic acid.

Perrone MG, Miciaccia M, Vitale P, Ferorelli S, Araújo CDCB, de Almeida GS, Souza Domingos TF, da Silva LCRP, de Pádula M, Cabral LM, Sathler PC, Bonaccorso C, Fortuna CG, Scilimati A. Perrone MG, et al. Among authors: scilimati a. Eur J Med Chem. 2021 Jan 1;209:112919. doi: 10.1016/j.ejmech.2020.112919. Epub 2020 Oct 9. Eur J Med Chem. 2021. PMID: 33129592

2

Novel synthesis of 3,4-diarylisoxazole analogues of valdecoxib: reversal cyclooxygenase-2 selectivity by sulfonamide group removal.

Di Nunno L, Vitale P, Scilimati A, Tacconelli S, Patrignani P. Di Nunno L, et al. Among authors: scilimati a. J Med Chem. 2004 Sep 23;47(20):4881-90. doi: 10.1021/jm040782x. J Med Chem. 2004. PMID: 15369392

3

Synthesis and biological evaluation of new clofibrate analogues as potential PPARalpha agonists.

Perrone MG, Santandrea E, Dell'Uomo N, Giannessi F, Milazzo FM, Sciarroni AF, Scilimati A, Tortorella V. Perrone MG, et al. Among authors: scilimati a. Eur J Med Chem. 2005 Feb;40(2):143-54. doi: 10.1016/j.ejmech.2004.09.018. Eur J Med Chem. 2005. PMID: 15694649

4

A chemoenzymatic scalable route to optically active (R)-1-(pyridin-3-yl)-2-aminoethanol, valuable moiety of beta3-adrenergic receptor agonists.

Perrone MG, Santandrea E, Giorgio E, Bleve L, Scilimati A, Tortorella P. Perrone MG, et al. Among authors: scilimati a. Bioorg Med Chem. 2006 Feb 15;14(4):1207-14. doi: 10.1016/j.bmc.2005.09.046. Epub 2005 Oct 10. Bioorg Med Chem. 2006. PMID: 16216512

5

Stereospecific synthesis and bio-activity of novel beta(3)-adrenoceptor agonists and inverse agonists.

Perrone MG, Santandrea E, Bleve L, Vitale P, Colabufo NA, Jockers R, Milazzo FM, Sciarroni AF, Scilimati A. Perrone MG, et al. Among authors: scilimati a. Bioorg Med Chem. 2008 Mar 1;16(5):2473-88. doi: 10.1016/j.bmc.2007.11.060. Epub 2007 Nov 28. Bioorg Med Chem. 2008. PMID: 18083578

6

Constrained analogues of tocainide as potent skeletal muscle sodium channel blockers towards the development of antimyotonic agents.

Catalano A, Carocci A, Corbo F, Franchini C, Muraglia M, Scilimati A, De Bellis M, De Luca A, Camerino DC, Sinicropi MS, Tortorella V. Catalano A, et al. Among authors: scilimati a. Eur J Med Chem. 2008 Nov;43(11):2535-40. doi: 10.1016/j.ejmech.2008.01.023. Epub 2008 Jan 31. Eur J Med Chem. 2008. PMID: 18342401

7

Upregulation of beta3-adrenergic receptor mRNA in human colon cancer: a preliminary study.

Perrone MG, Notarnicola M, Caruso MG, Tutino V, Scilimati A. Perrone MG, et al. Among authors: scilimati a. Oncology. 2008;75(3-4):224-9. doi: 10.1159/000163851. Epub 2008 Oct 14. Oncology. 2008. PMID: 18852493

8

The tertiary amine nitrogen atom of piperazine sulfonamides as a novel determinant of potent and selective beta3-adrenoceptor agonists.

Perrone MG, Bleve L, Santandrea E, Vitale P, Niso M, Scilimati A. Perrone MG, et al. Among authors: scilimati a. ChemMedChem. 2009 Dec;4(12):2080-97. doi: 10.1002/cmdc.200900292. ChemMedChem. 2009. PMID: 19882697

9

Selective COX-1 inhibition: A therapeutic target to be reconsidered.

Perrone MG, Scilimati A, Simone L, Vitale P. Perrone MG, et al. Among authors: scilimati a. Curr Med Chem. 2010;17(32):3769-805. doi: 10.2174/092986710793205408. Curr Med Chem. 2010. PMID: 20858219 Review.

10

β(3)-Adrenoceptor ligand development history through patent review.

Perrone MG, Scilimati A. Perrone MG, et al. Among authors: scilimati a. Expert Opin Ther Pat. 2011 Apr;21(4):505-36. doi: 10.1517/13543776.2011.561316. Epub 2011 Mar 17. Expert Opin Ther Pat. 2011. PMID: 21410429 Review.

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