Umezawa Y - Search Results

1

Structure-activity relationships of natural quinone vegfrecine analogs with potent activity against VEGFR-1 and -2 tyrosine kinases.

Adachi H, Nosaka C, Atsumi S, Nakae K, Umezawa Y, Sawa R, Kubota Y, Nakane C, Shibuya M, Nishimura Y. Adachi H, et al. Among authors: umezawa y. J Antibiot (Tokyo). 2021 Oct;74(10):734-742. doi: 10.1038/s41429-021-00445-y. Epub 2021 Jul 20. J Antibiot (Tokyo). 2021. PMID: 34282315

2

Synthesis and inhibitory activity of 8-substituted 2-deoxy-beta-KDO against CMP-KDO synthetase.

Adachi H, Kondo K, Kojima F, Umezawa Y, Ishino K, Hotta K, Nishimura Y. Adachi H, et al. Among authors: umezawa y. Nat Prod Res. 2006 Apr;20(4):361-70. doi: 10.1080/14756360500183699. Nat Prod Res. 2006. PMID: 16644531

3

Synthesis of boronic acid derivatives of tyropeptin: proteasome inhibitors.

Watanabe T, Momose I, Abe M, Abe H, Sawa R, Umezawa Y, Ikeda D, Takahashi Y, Akamatsu Y. Watanabe T, et al. Among authors: umezawa y. Bioorg Med Chem Lett. 2009 Apr 15;19(8):2343-5. doi: 10.1016/j.bmcl.2009.02.117. Epub 2009 Mar 4. Bioorg Med Chem Lett. 2009. PMID: 19307118

4

Flexible Enantiodivergent Synthesis and Biological Activity of Mannostatin Analogues, New Cyclitol Glycosidase Inhibitors.

Nishimura Y, Umezawa Y, Adachi H, Kondo S, Takeuchi T. Nishimura Y, et al. Among authors: umezawa y. J Org Chem. 1996 Jan 26;61(2):480-488. doi: 10.1021/jo951126v. J Org Chem. 1996. PMID: 11666964

5

Discovery of incednine as a potent modulator of the anti-apoptotic function of Bcl-xL from microbial origin.

Futamura Y, Sawa R, Umezawa Y, Igarashi M, Nakamura H, Hasegawa K, Yamasaki M, Tashiro E, Takahashi Y, Akamatsu Y, Imoto M. Futamura Y, et al. Among authors: umezawa y. J Am Chem Soc. 2008 Feb 13;130(6):1822-3. doi: 10.1021/ja710124p. Epub 2008 Jan 19. J Am Chem Soc. 2008. PMID: 18205364 No abstract available.

6

Structure-based design of derivatives of tyropeptin A as the potent and selective inhibitors of mammalian 20S proteasome.

Momose I, Umezawa Y, Hirosawa S, Iinuma H, Ikeda D. Momose I, et al. Among authors: umezawa y. Bioorg Med Chem Lett. 2005 Apr 1;15(7):1867-71. doi: 10.1016/j.bmcl.2005.02.013. Bioorg Med Chem Lett. 2005. PMID: 15780623

7

Synthesis and activity of tyropeptin A derivatives as potent and selective inhibitors of mammalian 20S proteasome.

Momose I, Umezawa Y, Hirosawa S, Iijima M, Iinuma H, Ikeda D. Momose I, et al. Among authors: umezawa y. Biosci Biotechnol Biochem. 2005 Sep;69(9):1733-42. doi: 10.1271/bbb.69.1733. Biosci Biotechnol Biochem. 2005. PMID: 16195592 Free article.

8

Novel pyrrole- and 1,2,3-triazole-based 2,3-oxidosqualene cyclase inhibitors.

Watanabe T, Umezawa Y, Takahashi Y, Akamatsu Y. Watanabe T, et al. Among authors: umezawa y. Bioorg Med Chem Lett. 2010 Oct 1;20(19):5807-10. doi: 10.1016/j.bmcl.2010.07.131. Epub 2010 Aug 3. Bioorg Med Chem Lett. 2010. PMID: 20728352

9

Synthesis and biological activity of sulphostin analogues, novel dipeptidyl peptidase IV inhibitors.

Abe M, Akiyama T, Umezawa Y, Yamamoto K, Nagai M, Yamazaki H, Ichikawa Y, Muraoka Y. Abe M, et al. Among authors: umezawa y. Bioorg Med Chem. 2005 Feb 1;13(3):785-97. doi: 10.1016/j.bmc.2004.10.036. Bioorg Med Chem. 2005. PMID: 15653346

10

Inhibitors of human 2,3-oxidosqualene cyclase (OSC) discovered by virtual screening.

Watanabe T, Kurata I, Umezawa Y, Takahashi Y, Akamatsu Y. Watanabe T, et al. Among authors: umezawa y. Bioorg Med Chem Lett. 2012 Jan 1;22(1):231-4. doi: 10.1016/j.bmcl.2011.11.021. Epub 2011 Nov 12. Bioorg Med Chem Lett. 2012. PMID: 22137785

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