Bianchini G - Search Results

1

Discovery of Novel TRPM8 Blockers Suitable for the Treatment of Somatic and Ocular Painful Conditions: A Journey through pK_a and LogD Modulation.

Bianchini G, Tomassetti M, Lillini S, Sirico A, Bovolenta S, Za L, Liberati C, Novelli R, Aramini A. Bianchini G, et al. J Med Chem. 2021 Nov 25;64(22):16820-16837. doi: 10.1021/acs.jmedchem.1c01647. Epub 2021 Nov 11. J Med Chem. 2021. PMID: 34762442

2

Targeting the minor pocket of C5aR for the rational design of an oral allosteric inhibitor for inflammatory and neuropathic pain relief.

Moriconi A, Cunha TM, Souza GR, Lopes AH, Cunha FQ, Carneiro VL, Pinto LG, Brandolini L, Aramini A, Bizzarri C, Bianchini G, Beccari AR, Fanton M, Bruno A, Costantino G, Bertini R, Galliera E, Locati M, Ferreira SH, Teixeira MM, Allegretti M. Moriconi A, et al. Among authors: bianchini g. Proc Natl Acad Sci U S A. 2014 Nov 25;111(47):16937-42. doi: 10.1073/pnas.1417365111. Epub 2014 Nov 10. Proc Natl Acad Sci U S A. 2014. PMID: 25385614 Free PMC article.

3

DFL23448, A Novel Transient Receptor Potential Melastin 8-Selective Ion Channel Antagonist, Modifies Bladder Function and Reduces Bladder Overactivity in Awake Rats.

Mistretta FA, Russo A, Castiglione F, Bettiga A, Colciago G, Montorsi F, Brandolini L, Aramini A, Bianchini G, Allegretti M, Bovolenta S, Russo R, Benigni F, Hedlund P. Mistretta FA, et al. Among authors: bianchini g. J Pharmacol Exp Ther. 2016 Jan;356(1):200-11. doi: 10.1124/jpet.115.228684. Epub 2015 Nov 6. J Pharmacol Exp Ther. 2016. PMID: 26546575

4

DF2755A, a novel non-competitive allosteric inhibitor of CXCR1/2, reduces inflammatory and post-operative pain.

Lopes AH, Brandolini L, Aramini A, Bianchini G, Silva RL, Zaperlon AC, Verri WA Jr, Alves-Filho JC, Cunha FQ, Teixeira MM, Allegretti M, Cunha TM. Lopes AH, et al. Among authors: bianchini g. Pharmacol Res. 2016 Jan;103:69-79. doi: 10.1016/j.phrs.2015.11.005. Epub 2015 Nov 28. Pharmacol Res. 2016. PMID: 26592483 Free article.

5

Antinociceptive effect of two novel transient receptor potential melastatin 8 antagonists in acute and chronic pain models in rat.

De Caro C, Russo R, Avagliano C, Cristiano C, Calignano A, Aramini A, Bianchini G, Allegretti M, Brandolini L. De Caro C, et al. Among authors: bianchini g. Br J Pharmacol. 2018 May;175(10):1691-1706. doi: 10.1111/bph.14177. Epub 2018 Apr 14. Br J Pharmacol. 2018. PMID: 29485712 Free PMC article.

6

DF2726A, a new IL-8 signalling inhibitor, is able to counteract chemotherapy-induced neuropathic pain.

Brandolini L, Castelli V, Aramini A, Giorgio C, Bianchini G, Russo R, De Caro C, d'Angelo M, Catanesi M, Benedetti E, Giordano A, Cimini A, Allegretti M. Brandolini L, et al. Among authors: bianchini g. Sci Rep. 2019 Aug 13;9(1):11729. doi: 10.1038/s41598-019-48231-z. Sci Rep. 2019. PMID: 31409858 Free PMC article.

7

Catalyst-Free Synthesis of Polysubstituted 5-Acylamino-1,3-Thiazoles via Hantzsch Cyclization of α-Chloroglycinates.

Tomassetti M, Lupidi G, Piermattei P, Rossi FV, Lillini S, Bianchini G, Aramini A, Ciufolini MA, Marcantoni E. Tomassetti M, et al. Among authors: bianchini g. Molecules. 2019 Oct 25;24(21):3846. doi: 10.3390/molecules24213846. Molecules. 2019. PMID: 31731437 Free PMC article.

8

Ergogenic Effect of BCAAs and L-Alanine Supplementation: Proof-of-Concept Study in a Murine Model of Physiological Exercise.

Mantuano P, Bianchini G, Cappellari O, Boccanegra B, Conte E, Sanarica F, Mele A, Camerino GM, Brandolini L, Allegretti M, De Bellis M, Aramini A, De Luca A. Mantuano P, et al. Among authors: bianchini g. Nutrients. 2020 Jul 30;12(8):2295. doi: 10.3390/nu12082295. Nutrients. 2020. PMID: 32751732 Free PMC article.

9

A new synthetic dual agonist of GPR120/GPR40 induces GLP-1 secretion and improves glucose homeostasis in mice.

Bianchini G, Nigro C, Sirico A, Novelli R, Prevenzano I, Miele C, Beguinot F, Aramini A. Bianchini G, et al. Biomed Pharmacother. 2021 Jul;139:111613. doi: 10.1016/j.biopha.2021.111613. Epub 2021 Apr 22. Biomed Pharmacother. 2021. PMID: 33895521 Free article.

10

Unexpected Salt/Cocrystal Polymorphism of the Ketoprofen-Lysine System: Discovery of a New Ketoprofen-l-Lysine Salt Polymorph with Different Physicochemical and Pharmacokinetic Properties.

Aramini A, Bianchini G, Lillini S, Bordignon S, Tomassetti M, Novelli R, Mattioli S, Lvova L, Paolesse R, Chierotti MR, Allegretti M. Aramini A, et al. Among authors: bianchini g. Pharmaceuticals (Basel). 2021 Jun 10;14(6):555. doi: 10.3390/ph14060555. Pharmaceuticals (Basel). 2021. PMID: 34200917 Free PMC article.

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