Gainetdinov RR - Search Results

1

Discovery of Novel Trace Amine-Associated Receptor 5 (TAAR5) Antagonists Using a Deep Convolutional Neural Network.

Bon C, Chern TR, Cichero E, O'Brien TE, Gustincich S, Gainetdinov RR, Espinoza S. Bon C, et al. Among authors: gainetdinov rr. Int J Mol Sci. 2022 Mar 14;23(6):3127. doi: 10.3390/ijms23063127. Int J Mol Sci. 2022. PMID: 35328548 Free PMC article.

2

Further insights into the pharmacology of the human trace amine-associated receptors: discovery of novel ligands for TAAR1 by a virtual screening approach.

Cichero E, Espinoza S, Franchini S, Guariento S, Brasili L, Gainetdinov RR, Fossa P. Cichero E, et al. Among authors: gainetdinov rr. Chem Biol Drug Des. 2014 Dec;84(6):712-20. doi: 10.1111/cbdd.12367. Epub 2014 Jun 30. Chem Biol Drug Des. 2014. PMID: 24894156

3

In-vivo pharmacology of Trace-Amine Associated Receptor 1.

Lam VM, Espinoza S, Gerasimov AS, Gainetdinov RR, Salahpour A. Lam VM, et al. Among authors: gainetdinov rr. Eur J Pharmacol. 2015 Sep 15;763(Pt B):136-42. doi: 10.1016/j.ejphar.2015.06.026. Epub 2015 Jun 17. Eur J Pharmacol. 2015. PMID: 26093041 Review.

4

Trace Amine Associate Receptor 1 (TAAR1) as a New Target for the Treatment of Cognitive Dysfunction in Alzheimer's Disease.

Leo D, Targa G, Espinoza S, Villers A, Gainetdinov RR, Ris L. Leo D, et al. Among authors: gainetdinov rr. Int J Mol Sci. 2022 Jul 15;23(14):7811. doi: 10.3390/ijms23147811. Int J Mol Sci. 2022. PMID: 35887159 Free PMC article.

5

Improved cognitive performance in trace amine-associated receptor 5 (TAAR5) knock-out mice.

Maggi S, Bon C, Gustincich S, Tucci V, Gainetdinov RR, Espinoza S. Maggi S, et al. Among authors: gainetdinov rr. Sci Rep. 2022 Aug 29;12(1):14708. doi: 10.1038/s41598-022-18924-z. Sci Rep. 2022. PMID: 36038766 Free PMC article.

6

Functional interaction between trace amine-associated receptor 1 and dopamine D2 receptor.

Espinoza S, Salahpour A, Masri B, Sotnikova TD, Messa M, Barak LS, Caron MG, Gainetdinov RR. Espinoza S, et al. Among authors: gainetdinov rr. Mol Pharmacol. 2011 Sep;80(3):416-25. doi: 10.1124/mol.111.073304. Epub 2011 Jun 13. Mol Pharmacol. 2011. PMID: 21670104 Free PMC article.

7

Insights into the structure and pharmacology of the human trace amine-associated receptor 1 (hTAAR1): homology modelling and docking studies.

Cichero E, Espinoza S, Gainetdinov RR, Brasili L, Fossa P. Cichero E, et al. Among authors: gainetdinov rr. Chem Biol Drug Des. 2013 Apr;81(4):509-16. doi: 10.1111/cbdd.12018. Chem Biol Drug Des. 2013. PMID: 22883051

8

BRET approaches to characterize dopamine and TAAR1 receptor pharmacology and signaling.

Espinoza S, Masri B, Salahpour A, Gainetdinov RR. Espinoza S, et al. Among authors: gainetdinov rr. Methods Mol Biol. 2013;964:107-22. doi: 10.1007/978-1-62703-251-3_8. Methods Mol Biol. 2013. PMID: 23296781

9

Design, Synthesis, and Evaluation of Thyronamine Analogues as Novel Potent Mouse Trace Amine Associated Receptor 1 (mTAAR1) Agonists.

Chiellini G, Nesi G, Digiacomo M, Malvasi R, Espinoza S, Sabatini M, Frascarelli S, Laurino A, Cichero E, Macchia M, Gainetdinov RR, Fossa P, Raimondi L, Zucchi R, Rapposelli S. Chiellini G, et al. Among authors: gainetdinov rr. J Med Chem. 2015 Jun 25;58(12):5096-107. doi: 10.1021/acs.jmedchem.5b00526. Epub 2015 Jun 5. J Med Chem. 2015. PMID: 26010728

10

Hit-to-Lead Optimization of Mouse Trace Amine Associated Receptor 1 (mTAAR1) Agonists with a Diphenylmethane-Scaffold: Design, Synthesis, and Biological Study.

Chiellini G, Nesi G, Sestito S, Chiarugi S, Runfola M, Espinoza S, Sabatini M, Bellusci L, Laurino A, Cichero E, Gainetdinov RR, Fossa P, Raimondi L, Zucchi R, Rapposelli S. Chiellini G, et al. Among authors: gainetdinov rr. J Med Chem. 2016 Nov 10;59(21):9825-9836. doi: 10.1021/acs.jmedchem.6b01092. Epub 2016 Oct 21. J Med Chem. 2016. PMID: 27731647

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