Kaiser M - Search Results

1

Discovery of Novel Quinoline-Based Proteasome Inhibitors for Human African Trypanosomiasis (HAT).

Koester DC, Marx VM, Williams S, Jiricek J, Dauphinais M, René O, Miller SL, Zhang L, Patra D, Chen YL, Cheung H, Gable J, Lakshminarayana SB, Osborne C, Galarneau JR, Kulkarni U, Richmond W, Bretz A, Xiao L, Supek F, Wiesmann C, Honnappa S, Be C, Mäser P, Kaiser M, Ritchie R, Barrett MP, Diagana TT, Sarko C, Rao SPS. Koester DC, et al. Among authors: kaiser m. J Med Chem. 2022 Sep 8;65(17):11776-11787. doi: 10.1021/acs.jmedchem.2c00791. Epub 2022 Aug 22. J Med Chem. 2022. PMID: 35993839 Free PMC article.

2

DNA binding affinity of bisguanidine and bis(2-aminoimidazoline) derivatives with in vivo antitrypanosomal activity.

Dardonville C, Barrett MP, Brun R, Kaiser M, Tanious F, Wilson WD. Dardonville C, et al. Among authors: kaiser m. J Med Chem. 2006 Jun 15;49(12):3748-52. doi: 10.1021/jm060295c. J Med Chem. 2006. PMID: 16759117 Free article.

3

Synthesis and biological evaluation of phosphate prodrugs of 4-phospho-D-erythronohydroxamic acid, an inhibitor of 6-phosphogluconate dehydrogenase.

Ruda GF, Alibu VP, Mitsos C, Bidet O, Kaiser M, Brun R, Barrett MP, Gilbert IH. Ruda GF, et al. Among authors: kaiser m. ChemMedChem. 2007 Aug;2(8):1169-80. doi: 10.1002/cmdc.200700040. ChemMedChem. 2007. PMID: 17615587 Free PMC article.

4

New bis(2-aminoimidazoline) and bisguanidine DNA minor groove binders with potent in vivo antitrypanosomal and antiplasmodial activity.

Rodríguez F, Rozas I, Kaiser M, Brun R, Nguyen B, Wilson WD, García RN, Dardonville C. Rodríguez F, et al. Among authors: kaiser m. J Med Chem. 2008 Feb 28;51(4):909-23. doi: 10.1021/jm7013088. Epub 2008 Feb 5. J Med Chem. 2008. PMID: 18247550

5

Novel functionalized melamine-based nitroheterocycles: synthesis and activity against trypanosomatid parasites.

Baliani A, Peal V, Gros L, Brun R, Kaiser M, Barrett MP, Gilbert IH. Baliani A, et al. Among authors: kaiser m. Org Biomol Chem. 2009 Mar 21;7(6):1154-66. doi: 10.1039/b813394h. Epub 2009 Jan 28. Org Biomol Chem. 2009. PMID: 19262935

6

Adenosine Kinase of T. b. Rhodesiense identified as the putative target of 4-[5-(4-phenoxyphenyl)-2H-pyrazol-3-yl]morpholine using chemical proteomics.

Kuettel S, Mosimann M, Mäser P, Kaiser M, Brun R, Scapozza L, Perozzo R. Kuettel S, et al. Among authors: kaiser m. PLoS Negl Trop Dis. 2009 Aug 25;3(8):e506. doi: 10.1371/journal.pntd.0000506. PLoS Negl Trop Dis. 2009. PMID: 19707572 Free PMC article.

7

Antitrypanosomal activity of 1,2-dihydroquinolin-6-ols and their ester derivatives.

Fotie J, Kaiser M, Delfín DA, Manley J, Reid CS, Paris JM, Wenzler T, Maes L, Mahasenan KV, Li C, Werbovetz KA. Fotie J, et al. Among authors: kaiser m. J Med Chem. 2010 Feb 11;53(3):966-82. doi: 10.1021/jm900723w. J Med Chem. 2010. PMID: 20047276

8

Optimization of purine-nitrile TbcatB inhibitors for use in vivo and evaluation of efficacy in murine models.

Mallari JP, Zhu F, Lemoff A, Kaiser M, Lu M, Brun R, Guy RK. Mallari JP, et al. Among authors: kaiser m. Bioorg Med Chem. 2010 Dec 1;18(23):8302-9. doi: 10.1016/j.bmc.2010.09.073. Epub 2010 Oct 8. Bioorg Med Chem. 2010. PMID: 21051236

9

1-Aryl-4-nitro-1H-imidazoles, a new promising series for the treatment of human African trypanosomiasis.

Trunz BB, Jędrysiak R, Tweats D, Brun R, Kaiser M, Suwiński J, Torreele E. Trunz BB, et al. Among authors: kaiser m. Eur J Med Chem. 2011 May;46(5):1524-35. doi: 10.1016/j.ejmech.2011.01.071. Epub 2011 Feb 26. Eur J Med Chem. 2011. PMID: 21353728

10

Antiparasitic agents: new drugs on the horizon.

Mäser P, Wittlin S, Rottmann M, Wenzler T, Kaiser M, Brun R. Mäser P, et al. Among authors: kaiser m. Curr Opin Pharmacol. 2012 Oct;12(5):562-6. doi: 10.1016/j.coph.2012.05.001. Epub 2012 May 29. Curr Opin Pharmacol. 2012. PMID: 22652215 Review.

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