Jacobson AE - Search Results

1

A Journey through Diastereomeric Space: The Design, Synthesis, In Vitro and In Vivo Pharmacological Activity, and Molecular Modeling of Novel Potent Diastereomeric MOR Agonists and Antagonists.

Chambers DR, Sulima A, Luo D, Prisinzano TE, Goldberg A, Xie B, Shi L, Paronis CA, Bergman J, Nassehi N, Selley DE, Imler GH, Jacobson AE, Rice KC. Chambers DR, et al. Among authors: jacobson ae. Molecules. 2022 Sep 30;27(19):6455. doi: 10.3390/molecules27196455. Molecules. 2022. PMID: 36234992 Free PMC article.

2

Optical resolution of (+/-)-2,5-dimethyl-2'-hydroxy-9alpha- and -9beta-propyl-6,7-benzomorphans and their pharmacological properties.

Rice KC, Jacobson AE. Rice KC, et al. Among authors: jacobson ae. J Med Chem. 1976 Mar;19(3):430-2. doi: 10.1021/jm00225a021. J Med Chem. 1976. PMID: 815550

3

Preparation and analgesic activity of 3,6-diacetylnormorphine and 6-acetylnormorphine.

Rice KC, Jacobson AE. Rice KC, et al. Among authors: jacobson ae. J Med Chem. 1975 Oct;18(10):1033-5. doi: 10.1021/jm00244a019. J Med Chem. 1975. PMID: 1159685

4

Probes for narcotic receptor mediated phenomena. 18. Epimeric 6 alpha- and 6 beta-iodo-3,14-dihydroxy-17-(cyclopropylmethyl)-4,5 alpha-epoxymorphinans as potential ligands for opioid receptor single photon emission computed tomography: synthesis, evaluation, and radiochemistry of [125I]-6 beta-iodo-3,14-dihydroxy-17-(cyclopropylmethyl)-4,5 alpha-epoxymorphinan.

de Costa BR, Iadarola MJ, Rothman RB, Berman KF, George C, Newman AH, Mahboubi A, Jacobson AE, Rice KC. de Costa BR, et al. Among authors: jacobson ae. J Med Chem. 1992 Jul 24;35(15):2826-35. doi: 10.1021/jm00093a016. J Med Chem. 1992. PMID: 1322988

5

Novel kappa opioid receptor and sigma ligands.

de Costa B, Rothman RB, Bowen WD, Radesca L, Band L, Reid A, Paolo LD, Walker JM, Jacobson AE, Rice KC. de Costa B, et al. Among authors: jacobson ae. NIDA Res Monogr. 1992;119:76-80. NIDA Res Monogr. 1992. PMID: 1331800 Review. No abstract available.

6

A study of the effect of the irreversible delta receptor antagonist [D-Ala2,Leu5,Cys6]-enkephalin on delta cx and delta ncx opioid binding sites in vitro and in vivo.

Rothman RB, Bykov V, Jacobson AE, Rice KC, Long JE, Bowen WD. Rothman RB, et al. Among authors: jacobson ae. Peptides. 1992 Jul-Aug;13(4):691-4. doi: 10.1016/0196-9781(92)90174-2. Peptides. 1992. PMID: 1331996

7

Probing the opioid receptor complex with (+)-trans-SUPERFIT. II. Evidence that mu ligands are noncompetitive inhibitors of the delta cx opioid peptide binding site.

Rothman RB, Mahboubi A, Bykov V, Kim CH, de Costa BR, Jacobson AE, Rice KC. Rothman RB, et al. Among authors: jacobson ae. Peptides. 1992 Nov-Dec;13(6):1137-43. doi: 10.1016/0196-9781(92)90020-4. Peptides. 1992. PMID: 1337378

8

Analogues of the dioxolanes dexoxadrol and etoxadrol as potential phencyclidine-like agents. Synthesis and structure-activity relationships.

Thurkauf A, Mattson MV, Richardson S, Mirsadeghi S, Ornstein PL, Harrison EA Jr, Rice KC, Jacobson AE, Monn JA. Thurkauf A, et al. Among authors: jacobson ae. J Med Chem. 1992 Apr 17;35(8):1323-9. doi: 10.1021/jm00086a001. J Med Chem. 1992. PMID: 1349351

9

The continuing interrelationship of CPDD and NIDDK.

Jacobson AE, Rice KC. Jacobson AE, et al. NIDA Res Monogr. 1992;119:49-53. NIDA Res Monogr. 1992. PMID: 1435982 No abstract available.

10

Potent analgesia, respiratory depression, dependence, abuse liability-clue to separability.

Newman AH, Rice KC, Jacobson AE. Newman AH, et al. Among authors: jacobson ae. NIDA Res Monogr. 1992;119:54-8. NIDA Res Monogr. 1992. PMID: 1435985 Review. No abstract available.

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