Kormos CM - Search Results

1

Isolation of Hemiketal and Hydroxy Ketone Tautomers of Synthetic Intermediates Each Affording 18-Hydroxycortisol-1,6,7-d₃.

Lewin AH, Hayes JP, Zhong D, Zhang D, Kormos CM, Mascarella SW, Seltzman HH. Lewin AH, et al. Among authors: kormos cm. ACS Omega. 2023 Jul 26;8(31):28185-28195. doi: 10.1021/acsomega.3c01648. eCollection 2023 Aug 8. ACS Omega. 2023. PMID: 37576635 Free PMC article.

2

Synthesis and pharmacological validation of a novel radioligand for the orphan GPR88 receptor.

Decker AM, Rahman MT, Kormos CM, Hesk D, Darcq E, Kieffer BL, Jin C. Decker AM, et al. Among authors: kormos cm. Bioorg Med Chem Lett. 2023 Jan 15;80:129120. doi: 10.1016/j.bmcl.2022.129120. Epub 2022 Dec 29. Bioorg Med Chem Lett. 2023. PMID: 36587872 Free PMC article.

3

Identification of a Potent Human Trace Amine-Associated Receptor 1 Antagonist.

Decker AM, Brackeen MF, Mohammadkhani A, Kormos CM, Hesk D, Borgland SL, Blough BE. Decker AM, et al. Among authors: kormos cm. ACS Chem Neurosci. 2022 Apr 6;13(7):1082-1095. doi: 10.1021/acschemneuro.2c00086. Epub 2022 Mar 24. ACS Chem Neurosci. 2022. PMID: 35325532 Free PMC article.

4

Design, synthesis and biological evaluation of a bi-specific vaccine against α-pyrrolidinovalerophenone (α-PVP) and 3,4-methylenedioxypyrovalerone (MDPV) in rats.

McClenahan SJ, Kormos CM, Gunnell M, Hambuchen MD, Lamb P, Carroll FI, Lewin AH, Peterson EC, Owens SM. McClenahan SJ, et al. Among authors: kormos cm. Vaccine. 2020 Jan 10;38(2):336-344. doi: 10.1016/j.vaccine.2019.10.008. Epub 2019 Oct 16. Vaccine. 2020. PMID: 31629568 Free PMC article.

5

Potent and Selective Tetrahydroisoquinoline Kappa Opioid Receptor Antagonists of Lead Compound (3 R)-7-Hydroxy- N-[(1 S)-2-methyl-1-(piperidin-1-ylmethyl)propyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide (PDTic).

Ondachi PW, Kormos CM, Runyon SP, Thomas JB, Mascarella SW, Decker AM, Navarro HA, Fennell TR, Snyder RW, Carroll FI. Ondachi PW, et al. Among authors: kormos cm. J Med Chem. 2018 Sep 13;61(17):7525-7545. doi: 10.1021/acs.jmedchem.8b00673. Epub 2018 Aug 29. J Med Chem. 2018. PMID: 30117738 Free PMC article.

6

Potent and Selective Tetrahydroisoquinoline Kappa Opioid Receptor Antagonists of Lead Compound (3 R)- N-[1 R)-1-(Cyclohexylmethyl)-2-methylpropyl]-7-hydroxy-1,2,3,4-tetrahydroisoquinoline-3-carboxamide (CDTic).

Kormos CM, Ondachi PW, Runyon SP, Thomas JB, Mascarella SW, Decker AM, Navarro HA, Fennell TR, Snyder RW, Carroll FI. Kormos CM, et al. J Med Chem. 2018 Sep 13;61(17):7546-7559. doi: 10.1021/acs.jmedchem.8b00674. Epub 2018 Aug 29. J Med Chem. 2018. PMID: 30032602 Free PMC article.

7

Simple Tetrahydroisoquinolines Are Potent and Selective Kappa Opioid Receptor Antagonists.

Kormos CM, Ondachi PW, Runyon SP, Thomas JB, Mascarella SW, Decker AM, Navarro HA, Carroll FI. Kormos CM, et al. ACS Med Chem Lett. 2017 May 25;8(7):742-745. doi: 10.1021/acsmedchemlett.7b00115. eCollection 2017 Jul 13. ACS Med Chem Lett. 2017. PMID: 28740609 Free PMC article.

8

Design, Synthesis, and Biological Evaluation of Structurally Rigid Analogues of 4-(3-Hydroxyphenyl)piperidine Opioid Receptor Antagonists.

Runyon SP, Kormos CM, Gichinga MG, Mascarella SW, Navarro HA, Deschamps JR, Imler GH, Carroll FI. Runyon SP, et al. Among authors: kormos cm. J Org Chem. 2016 Nov 4;81(21):10383-10391. doi: 10.1021/acs.joc.6b01366. Epub 2016 Aug 2. J Org Chem. 2016. PMID: 27462910 Free PMC article.

9

Design, synthesis, and pharmacological evaluation of JDTic analogs to examine the significance of replacement of the 3-hydroxyphenyl group with pyridine or thiophene bioisosteres.

Kormos CM, Gichinga MG, Runyon SP, Thomas JB, Mascarella SW, Decker AM, Navarro HA, Carroll FI. Kormos CM, et al. Bioorg Med Chem. 2016 Aug 15;24(16):3842-8. doi: 10.1016/j.bmc.2016.06.029. Epub 2016 Jun 15. Bioorg Med Chem. 2016. PMID: 27364611 Free PMC article.

10

Design, synthesis, and pharmacological evaluation of JDTic analogs to examine the significance of the 3- and 4-methyl substituents.

Carroll FI, Gichinga MG, Kormos CM, Maitra R, Runyon SP, Thomas JB, Mascarella SW, Decker AM, Navarro HA. Carroll FI, et al. Among authors: kormos cm. Bioorg Med Chem. 2015 Oct 1;23(19):6379-88. doi: 10.1016/j.bmc.2015.08.025. Epub 2015 Aug 25. Bioorg Med Chem. 2015. PMID: 26342544 Free PMC article.

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