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Covalent Macrocyclic Proteasome Inhibitors Mitigate Resistance in Plasmodium falciparum.
Bennett JM, Ward KE, Muir RK, Kabeche S, Yoo E, Yeo T, Lam G, Zhang H, Almaliti J, Berger G, Faucher FF, Lin G, Gerwick WH, Yeh E, Fidock DA, Bogyo M. Bennett JM, et al. Among authors: gerwick wh. ACS Infect Dis. 2023 Oct 13;9(10):2036-2047. doi: 10.1021/acsinfecdis.3c00310. Epub 2023 Sep 15. ACS Infect Dis. 2023. PMID: 37712594 Free PMC article.
Development of Potent and Highly Selective Epoxyketone-Based Plasmodium Proteasome Inhibitors.
Almaliti J, Fajtová P, Calla J, LaMonte GM, Feng M, Rocamora F, Ottilie S, Glukhov E, Boura E, Suhandynata RT, Momper JD, Gilson MK, Winzeler EA, Gerwick WH, O'Donoghue AJ. Almaliti J, et al. Among authors: gerwick wh. Chemistry. 2023 Apr 6;29(20):e202203958. doi: 10.1002/chem.202203958. Epub 2023 Mar 6. Chemistry. 2023. PMID: 36617500 Free PMC article.
Mitigating the risk of antimalarial resistance via covalent dual-subunit inhibition of the Plasmodium proteasome.
Deni I, Stokes BH, Ward KE, Fairhurst KJ, Pasaje CFA, Yeo T, Akbar S, Park H, Muir R, Bick DS, Zhan W, Zhang H, Liu YJ, Ng CL, Kirkman LA, Almaliti J, Gould AE, Duffey M, O'Donoghue AJ, Uhlemann AC, Niles JC, da Fonseca PCA, Gerwick WH, Lin G, Bogyo M, Fidock DA. Deni I, et al. Among authors: gerwick wh. Cell Chem Biol. 2023 May 18;30(5):470-485.e6. doi: 10.1016/j.chembiol.2023.03.002. Epub 2023 Mar 23. Cell Chem Biol. 2023. PMID: 36963402 Free PMC article.
Methods in marine natural product drug discovery: what's new?
Almaliti J, Gerwick WH. Almaliti J, et al. Among authors: gerwick wh. Expert Opin Drug Discov. 2023 Jul;18(7):687-691. doi: 10.1080/17460441.2023.2214360. Epub 2023 May 16. Expert Opin Drug Discov. 2023. PMID: 37194298 No abstract available.
Structural elucidation of recombinant Trichomonas vaginalis 20S proteasome bound to covalent inhibitors.
Silhan J, Fajtova P, Bartosova J, Hurysz BM, Almaliti J, Miyamoto Y, Eckmann L, Gerwick WH, O'Donoghue AJ, Boura E. Silhan J, et al. Among authors: gerwick wh. bioRxiv [Preprint]. 2023 Aug 17:2023.08.17.553660. doi: 10.1101/2023.08.17.553660. bioRxiv. 2023. Update in: Nat Commun. 2024 Oct 4;15(1):8621. doi: 10.1038/s41467-024-53022-w PMID: 37645851 Free PMC article. Updated. Preprint.
Carmaphycin B-Based Proteasome Inhibitors to Treat Human African Trypanosomiasis: Structure-Activity Relationship and In Vivo Efficacy.
Liu LJ, Francisco KR, Sun YU, Serafim MSM, Amarasinghe DK, Teixeira TR, Lucero B, Kronenberger T, Elsayed W, Elwakeel H, Al-Hindy M, Almaliti J, Gerwick WH, O'Donoghue AJ, Caffrey CR. Liu LJ, et al. Among authors: gerwick wh. ACS Infect Dis. 2024 Dec 13;10(12):4182-4193. doi: 10.1021/acsinfecdis.4c00441. Epub 2024 Nov 26. ACS Infect Dis. 2024. PMID: 39589805 Free PMC article.
381 results