Desai UR - Search Results

1

Dual Targeting of the PDZ1 and PDZ2 Domains of MDA-9/Syntenin Inhibits Melanoma Metastasis.

Pradhan AK, Modi J, Maji S, Kumar A, Bhoopathi P, Mannangatti P, Guo C, Afosah DK, Mochel MC, Mukhopadhyay ND, Kirkwood JM, Wang XY, Desai UR, Sarkar D, Emdad L, Das SK, Fisher PB. Pradhan AK, et al. Among authors: desai ur. Mol Cancer Ther. 2023 Oct 2;22(10):1115-1127. doi: 10.1158/1535-7163.MCT-22-0653. Mol Cancer Ther. 2023. PMID: 37721536

2

Allosteric Partial Inhibition of Monomeric Proteases. Sulfated Coumarins Induce Regulation, not just Inhibition, of Thrombin.

Verespy S 3rd, Mehta AY, Afosah D, Al-Horani RA, Desai UR. Verespy S 3rd, et al. Among authors: desai ur. Sci Rep. 2016 Apr 7;6:24043. doi: 10.1038/srep24043. Sci Rep. 2016. PMID: 27053426 Free PMC article.

3

Allosteric Inhibition of Factor XIIIa. Non-Saccharide Glycosaminoglycan Mimetics, but Not Glycosaminoglycans, Exhibit Promising Inhibition Profile.

Al-Horani RA, Karuturi R, Lee M, Afosah DK, Desai UR. Al-Horani RA, et al. Among authors: desai ur. PLoS One. 2016 Jul 28;11(7):e0160189. doi: 10.1371/journal.pone.0160189. eCollection 2016. PLoS One. 2016. PMID: 27467511 Free PMC article.

4

2-O, 3-O Desulfated Heparin Blocks High Mobility Group Box 1 Release by Inhibition of p300 Acetyltransferase Activity.

Zheng S, Kummarapurugu AB, Afosah DK, Sankaranarayanan NV, Boothello RS, Desai UR, Kennedy T, Voynow JA. Zheng S, et al. Among authors: desai ur. Am J Respir Cell Mol Biol. 2017 Jan;56(1):90-98. doi: 10.1165/rcmb.2016-0069OC. Am J Respir Cell Mol Biol. 2017. PMID: 27585400 Free PMC article.

5

Potent, Selective, Allosteric Inhibition of Human Plasmin by Sulfated Non-Saccharide Glycosaminoglycan Mimetics.

Afosah DK, Al-Horani RA, Sankaranarayanan NV, Desai UR. Afosah DK, et al. Among authors: desai ur. J Med Chem. 2017 Jan 26;60(2):641-657. doi: 10.1021/acs.jmedchem.6b01474. Epub 2017 Jan 5. J Med Chem. 2017. PMID: 27976897 Free PMC article.

6

A small group of sulfated benzofurans induces steady-state submaximal inhibition of thrombin.

Afosah DK, Verespy S 3rd, Al-Horani RA, Boothello RS, Karuturi R, Desai UR. Afosah DK, et al. Among authors: desai ur. Bioorg Med Chem Lett. 2018 Apr 1;28(6):1101-1105. doi: 10.1016/j.bmcl.2018.01.069. Epub 2018 Feb 3. Bioorg Med Chem Lett. 2018. PMID: 29459207 Free PMC article.

7

Molecular principles for heparin oligosaccharide-based inhibition of neutrophil elastase in cystic fibrosis.

Kummarapurugu AB, Afosah DK, Sankaranarayanan NV, Navaz Gangji R, Zheng S, Kennedy T, Rubin BK, Voynow JA, Desai UR. Kummarapurugu AB, et al. Among authors: desai ur. J Biol Chem. 2018 Aug 10;293(32):12480-12490. doi: 10.1074/jbc.RA118.002644. Epub 2018 Jun 14. J Biol Chem. 2018. PMID: 29903912 Free PMC article.

8

Inhibition of Herpes Simplex Virus-1 Entry into Human Cells by Nonsaccharide Glycosaminoglycan Mimetics.

Gangji RN, Sankaranarayanan NV, Elste J, Al-Horani RA, Afosah DK, Joshi R, Tiwari V, Desai UR. Gangji RN, et al. Among authors: desai ur. ACS Med Chem Lett. 2018 Jul 16;9(8):797-802. doi: 10.1021/acsmedchemlett.7b00364. eCollection 2018 Aug 9. ACS Med Chem Lett. 2018. PMID: 30128070 Free PMC article.

9

On the Process of Discovering Leads That Target the Heparin-Binding Site of Neutrophil Elastase in the Sputum of Cystic Fibrosis Patients.

Morla S, Sankaranarayanan NV, Afosah DK, Kumar M, Kummarapurugu AB, Voynow JA, Desai UR. Morla S, et al. Among authors: desai ur. J Med Chem. 2019 Jun 13;62(11):5501-5511. doi: 10.1021/acs.jmedchem.9b00379. Epub 2019 May 28. J Med Chem. 2019. PMID: 31074986 Free PMC article.

10

A synthetic heparin mimetic that allosterically inhibits factor XIa and reduces thrombosis in vivo without enhanced risk of bleeding.

Al-Horani RA, Abdelfadiel EI, Afosah DK, Morla S, Sistla JC, Mohammed B, Martin EJ, Sakagami M, Brophy DF, Desai UR. Al-Horani RA, et al. Among authors: desai ur. J Thromb Haemost. 2019 Dec;17(12):2110-2122. doi: 10.1111/jth.14606. Epub 2019 Sep 10. J Thromb Haemost. 2019. PMID: 31397071 Free PMC article.

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